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BIIB021

Phase 2

Breast Cancer | Small molecule | Oncology |Biogen Inc.|Last Updated: Dec 29, 2016

Success Probability

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment54

FDA Designations

No designations recorded

Clinical trial landscape

BIIB021 · 4 trials · 3 indications

Phase 2 2Phase 1 2
NCT01004081Hormone Receptor Positive Metastatic Breast Cancer (HR+ mBC) BIIB021 Plus Aromasin Schedule FindingBreast Cancer
COMPLETED54 Analytics
NCT00618319An Open-Label, 18FDG-PET Pharmacodynamic Assessment of the Effect of BIIB021 in Subjects With Gastrointestinal Stromal Tumors (GIST)GIST
COMPLETED20 Analytics
PHASE2COMPLETED
Hormone Receptor Positive Metastatic Breast Cancer (HR+ mBC) BIIB021 Plus Aromasin Schedule Finding
Breast CancerUnlock trial analytics
PHASE2COMPLETED
An Open-Label, 18FDG-PET Pharmacodynamic Assessment of the Effect of BIIB021 in Subjects With Gastrointestinal Stromal Tumors (GIST)
GISTUnlock trial analytics

Study Endpoints

Primary Endpoints

The primary objective of this study is to assess the efficacy of 2 dosing regimens of BIIB021 in combination with exemestane in women whose HR+ breast cancer had progressed following treatment with a nonsteroidal AI.
As specified in protocol
Changes in FDG-PET imaging
28 days
The primary objective of the study is to assess the pharmacokinetics of BIIB021 taken under fed conditions compared to BIIB021 taken under fasting conditions in subjects with advanced solid tumors.
Cycle 1, Day 3
Safety and tolerability of BIIB021
As specified in protocol

Secondary Endpoints

The secondary objective of this study is to evaluate the safety and tolerability of BIIB021 in combination with exemestane in this study population.
As specified in protocol
Characterize the safety profile of BIIB021
Duration of study
To assess the pharmacokinetics of BIIB021 taken with an antacid (ranitidine) compared to BIIB021 taken with no antacid, both under fasting conditions
Cycle 1, Day 8 and Day 10
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BIIB021 BID + exemestaneEXPERIMENTALBIIB021 100 mg BID + exemestane 25 mg QD
BIIB021 TIW + exemestaneEXPERIMENTALBIIB021 450 mg TIW + exemestane 25 mg QD
1EXPERIMENTALBIIB021
BIIB021 and FoodEXPERIMENTALThe food phase will assess the effect of a high fat meal on the pharmacokinetics of BIIB021.
BIIB021 and AntacidEXPERIMENTALAntacid phase will assess the effect of an antacid on the pharmacokinetics of BIIB021.
2EXPERIMENTALSubjects in Schedule B will take BIIB021 in the morning at approximately 0800 with at least 6 ounces of water following an overnight fast (beginning at midnight). The second dose will be taken, following at least a 2-hour fast, 12 hours (+/- 2 hours) after the first dose, except on Day 1 of Cycle 1 and Day 1 of Cycle 2.

Interventions

NameTypeDescription
BIIB021DRUGBID orally for 28 days
exemestane (Aromasin)DRUGDaily in tablet form for 28 days
BIIB021 and FoodDRUGAssessing the effect of food use on BIIB021
BIIB0121 and AntacidDRUGAssessing the effect of antacid use on BIIB021
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Eligibility Criteria

Age Range18 Years to N/A
SexFEMALE
Healthy VolunteersNo
Study Sites34

Inclusion Criteria: * Age 18 years of age * Must have histologically or cytologically confirmed estrogen receptor- positive or progesterone receptor-positive, incurable, locally advanced, or metastatic breast cancer. * Must have disease progression during treatment with a nonsteroidal AI for locall...

Countries:United StatesAustraliaBelgiumRussia
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Competitive Landscape -Breast Cancer 402 trials

Top 20 of 92 competitors

CompanyTickerTrialsLead PhaseDrugs
AstraZeneca PLCAZN47PHASE3Fulvestrant, Capivasertib
Merck & Co., Inc.MRK12PHASE3Pembrolizumab, Paclitaxel, Doxorubicin, Epirubicin, Cyclophosphamide
Eli Lilly and CompanyLLY27PHASE3Abemaciclib, Standard Adjuvant Endocrine Therapy
BioNTech SE Sponsored ADRBNTX7PHASE3DB-1303/BNT323, T-DM1
Gilead Sciences, Inc.GILD13PHASE3Sacituzumab Govitecan-hziy, Eribulin, Capecitabine Product, Gemcitabine, Vinorelbine
Novartis AG Sponsored ADRNVS30PHASE3Ribociclib
Pfizer Inc.PFE34PHASE3ARV-471, Fulvestrant
BeOne Medicines Ltd. Sponsored ADRONC5PHASE3BGB-43395, Letrozole, Abemaciclib, Palbociclib, Ribociclib
Olema Pharmaceuticals, Inc.OLMA5PHASE3Palazestrant, Fulvestrant, Anastrozole, Letrozole, Exemestane
Jazz Pharmaceuticals Public Limited CompanyJAZZ3PHASE3Zanidatamab, Trastuzumab, Eribulin, Vinorelbine, Gemcitabine
Celcuity Inc.CELC3PHASE3Gedatolisib, Palbociclib, Fulvestrant, Alpelisib
Relay Therapeutics, Inc.RLAY2PHASE3Zovegalisib, Capivasertib, Fulvestrant
GSK plc Sponsored ADRGSK2PHASE3Niraparib
Greenwich LifeSciences, Inc.GLSI1PHASE3GLSI-100
Bristol-Myers Squibb CompanyBMY5PHASE2Iza-bren, Nab-paclitaxel, Paclitaxel, Capecitabine, Carboplatin
BriaCell Therapeutics CorpBCTX2PHASE3SV-BR-1-GM, Cyclophosphamide, Interferon infiltration of the inoculation site, Retifanlimab, Treatment of Physician's Choice
Incyte CorporationINCY4PHASE2Ruxolitinib, Capecitabine, Regorafenib
Natera, Inc.NTRA3PHASE2Discontinuation of the anti-HER2 maintenance therapy
Puma Biotechnology, Inc.PBYI3PHASE2Neratinib, Loperamide, Colesevelam
Atossa Therapeutics, Inc.ATOS1PHASE2endoxifen, goserelin
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Frequently asked questions about BIIB021

What is BIIB021 used for?

BIIB021 is an investigational small molecule being studied for the treatment of breast cancer, gastrointestinal stromal tumors (GIST), and advanced solid tumors. It is developed by Biogen Inc. and has been evaluated in clinical trials for these oncology indications.

Who makes BIIB021?

BIIB021 is developed by Biogen Inc., a biotechnology company traded on the NASDAQ under the ticker symbol BIIB. The drug has been studied in clinical trials for oncology indications including breast cancer, GIST, and advanced solid tumors.

What phase is BIIB021 in?

BIIB021 is an investigational drug that has completed Phase 1 and Phase 2 clinical trials. It is not FDA approved and remains in clinical development. The trials have been completed, with no active trials currently ongoing for this asset.

What clinical trials has BIIB021 been in?

BIIB021 has been studied in four completed clinical trials. These include NCT00618319 for GIST, NCT00618735 for advanced solid tumors, NCT01004081 for hormone receptor positive metastatic breast cancer, and NCT01017198 for advanced solid tumors. The trials were conducted in the United States and other countries.

Is BIIB021 the same as any other drug?

BIIB021 is the investigational name for this small molecule developed by Biogen Inc. No alternative names have been reported for this compound in the available clinical trial information.