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BMF-650

Phase 1

Obesity | Small molecule | Metabolic |Biomea Fusion, Inc.|Last Updated: Apr 9, 2026

Target and mechanism

Molecular targetGLP-1
Target classReceptor
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLEDDMC
Total Trials1
Total Enrollment80

FDA Designations

No designations recorded

Clinical trial landscape

BMF-650 · 1 trial · 1 indication

Phase 1 1
NCT07223216Study of BMF-650 in Otherwise Healthy Overweight or Obese Adult ParticipantsObesity
ACTIVE NOT_RECRUITING80 Analytics
PHASE1ACTIVE NOT_RECRUITING
Study of BMF-650 in Otherwise Healthy Overweight or Obese Adult Participants
ObesityUnlock trial analytics

Study Endpoints

Primary Endpoints

Assess safety and tolerability of BMF-650
6 weeks (Part 1) and 11 weeks (Part 2)

Incidence of adverse events (AEs)

Secondary Endpoints

Evaluate PK and food effect of BMF-650 in fed and fasted states
2 weeks (Part 1) and 6 weeks (Part 2)
Assess the impact of multiple ascending doses of BMF-650 on weight (Part 2 only)
6 weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part 1 SAD Cohort 1 (Regimen A)EXPERIMENTALBMF-650 Tablets 10 mg or matching placebo in fasted state
Part 1 SAD Cohort 2 (Regimen B and C)EXPERIMENTALRegimen B: BMF-650 Tablets 25 mg or matching placebo in fasted state Regimen C: BMF-650 Tablets 25 mg or matching placebo in fed state (high-fat breakfast 30 minutes before BMF-650 or placebo is administered)
Part 1 SAD Cohort 3 (Regimen D)EXPERIMENTALBMF-650 Tablets 50 mg or matching placebo in fasted state
Part 1 SAD Cohort 4 (Regimen E and F) (Optional)EXPERIMENTALRegimen E: BMF-650 Tablets 100 mg or matching placebo in fasted state Regimen F: BMF-650 Tablets 100 mg or matching placebo in fed state (high-fat breakfast 30 minutes before BMF-650 or placebo is administered)
Part 1 SAD Cohort 5 (Regimen G) (Optional)EXPERIMENTALBMF-650 Tablets 200 mg or matching placebo in fasted state
Part 2 MAD Cohort 1 (Regimen H)EXPERIMENTALBMF-650 Tablets or matching placebo in fasted state 10 mg QD for 7 days; 25 mg QD for 7 days; 50 mg QD for 7 days; 100 mg QD for 21 days.
Part 2 MAD Cohort 2 (Regimen I)EXPERIMENTALBMF-650 Tablets or matching placebo in fasted state 50 mg QD for 7 days; 100 mg QD for 7 days; 200 mg QD for 28 days.
Part 2 MAD Cohort 3 (Regimen J)EXPERIMENTALBMF-650 Tablets or matching placebo in fasted state 75 mg QD for 7 days; 150 mg QD for 7 days; 300 mg QD for 28 days.
Part 2 MAD Cohort 4 (Regimen K) (Optional)EXPERIMENTALBMF-650 Tablets or matching placebo in fasted state 75 mg QD for 7 days; 200 mg QD for 7 days; 400 mg QD for 28 days.

Interventions

NameTypeDescription
BMF-650DRUGInterventional Product
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Must be able to understand a written informed consent, which must be obtained prior to initiation of study procedures. 2. Must be willing and able to comply with all study requirements 3. Healthy males or non-pregnant, non-lactating healthy females with obesity or overweight....

Countries:United States
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Frequently asked questions about BMF-650

What is BMF-650 used for?

BMF-650 is an investigational small molecule being developed for the treatment of obesity. It is currently in Phase 1 clinical development and has not been approved by the FDA. The drug is being studied in otherwise healthy overweight or obese adult participants.

What does BMF-650 target?

BMF-650 targets the GLP-1 receptor. GLP-1 receptor agonists are known to help regulate appetite and blood sugar, which is relevant for obesity treatment. As a small molecule targeting this receptor, BMF-650 is being investigated for its potential effects in overweight or obese individuals.

Who is developing BMF-650?

BMF-650 is being developed by Biomea Fusion, Inc., a biopharmaceutical company traded on the stock exchange under the ticker symbol BMEA. The company is conducting clinical research on this small molecule for obesity.

What phase is BMF-650 in?

BMF-650 is in Phase 1 clinical development. It is an investigational drug, meaning it has not yet been approved by regulatory authorities. The ongoing Phase 1 trial is active but not recruiting participants, and the drug is being studied in the United States.

What clinical trials is BMF-650 in?

BMF-650 is being studied in a Phase 1 clinical trial with the identifier NCT07223216, titled "Study of BMF-650 in Otherwise Healthy Overweight or Obese Adult Participants." This randomized, double-blind, controlled trial has an enrollment of 80 participants and is being conducted in the United States.