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OSI-774

Phase 2

Head and Neck Cancer | Small molecule | Oncology |Roche Holding AG|Last Updated: Jul 22, 2026

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLEDBiomarker
Total Trials1
Total Enrollment50

FDA Designations

No designations recorded

Clinical trial landscape

OSI-774 · 1 trial · 1 indication

Phase 2 1
NCT00076310OSI-774/Cisplatin/Taxotere in Head & Neck Squamous Cell CancerHead and Neck Cancer
COMPLETED50 Analytics
PHASE2COMPLETED
OSI-774/Cisplatin/Taxotere in Head & Neck Squamous Cell Cancer
Head and Neck CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Overall Response Assessment (Radiographic RECIST)
after 2 cycles of treatment (6 weeks) and confirmed 4-6 weeks thereafter

Per Response Evaluation Criteria in Solid Tumors Criteria (RECIST v.1.0) for target lesions and assessed by CT or MRI: Complete Response (CR), disappearance of all target lesions; Partial Response (PR), \>= 30% decrease in the sum of the longest diameter of target lesions; Stable Disease (SD), neither sufficient shrinkage to qualify for PR nor sufficient growth to qualify for PD; Progressive Disease (PD), \>= 20% increase in the sum of the longest diameter from the smallest sum diameter recorded, NE = not evaluable

Secondary Endpoints

Progression Free Survival and Overall Survival Duration Assessments
From treatment initiation until 150 months after initiation of treatment
Toxicity -- Number of Adverse Events
time of first drug administration to 30 days after last drug administration (maximum of 6 months)
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Cisplatin + Docetaxel + OSI-774EXPERIMENTALCisplatin 75 mg/m\^2 IV every 21 days. Docetaxel 60 mg/m\^2 IV repeated every 21 days. OSI-774 100 mg oral administered daily. May have a dose escalation of 150 mg pending on prior dose toleration. Patients will continue on daily OSI-774 until a study endpoint or removal from study is reached.

Interventions

NameTypeDescription
DocetaxelDRUG60 mg/m\^2 IV repeated every 21 days.
OSI-774DRUG100 mg oral administered daily. May have a dose escalation of 150 mg pending on prior dose toleration. Patients will continue on daily OSI-774 until a study endpoint or removal from study is reached.
CisplatinDRUG75 mg/m\^2 IV every 21 days.
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. Have histologically or cytologically confirmed metastatic or recurrent head and neck squamous cell carcinoma from the primary lesion and/or lymph nodes of the oral cavity, oropharynx, hypopharynx, or larynx. 2. Have measurable disease, defined as at least one lesion that can ...

Countries:United States
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Recent Changes (Last 90 Days)

MEDIUMAug 22, 2026NCT00076310TRIAL_REMOVED: changed
MEDIUMAug 22, 2026NCT00076310TRIAL_REMOVED: changed
MEDIUMAug 22, 2026NCT00076310TRIAL_REMOVED: changed
MEDIUMAug 22, 2026NCT00076310TRIAL_REMOVED: changed

Frequently asked questions about OSI-774

What is OSI-774 used for in Head and Neck Cancer?

OSI-774 is an investigational small molecule being studied for the treatment of Head and Neck Cancer, specifically head and neck squamous cell carcinoma. It is currently in Phase 2 clinical development and has not been approved by regulatory authorities.

What does OSI-774 target?

OSI-774 is a small molecule that targets the epidermal growth factor receptor (EGFR) pathway. By inhibiting this receptor, it aims to interfere with cancer cell growth and survival in head and neck squamous cell carcinoma.

Who makes OSI-774?

OSI-774 is being developed by Roche Holding AG, a multinational healthcare company. Roche's stock is traded on the OTC market under the ticker symbol RHHBY.

What phase is OSI-774 in?

OSI-774 is currently in Phase 2 clinical development for Head and Neck Cancer. It is an investigational drug, meaning it has not yet been approved by the FDA or other regulatory bodies for commercial use.

What clinical trials is OSI-774 in?

OSI-774 has one completed Phase 2 clinical trial, identified as NCT00076310, titled 'OSI-774/Cisplatin/Taxotere in Head & Neck Squamous Cell Cancer'. This trial enrolled 50 participants in the United States and was an uncontrolled, non-randomized study.

Is OSI-774 the same as erlotinib?

OSI-774 is also known as erlotinib, a small molecule EGFR inhibitor. In the context of this development program, OSI-774 refers to the same compound being evaluated for head and neck cancer.