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NNC0487-0111 A

Phase 1

Obesity | Small molecule | Metabolic |Novo Nordisk A/S|Last Updated: Jun 15, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials2
Total Enrollment187
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT06461039A Research Study Looking at How the Compound NNC0487-0111 Works With Birth Control Pills and Affects Emptying of the Stomach in Women Not Able to Become PregnantPHASE1 COMPLETED 43Jun 14, 2024Apr 4, 2025May 8, 20251 Canada
NCT05369390A Research Study on How NNC0487-0111 Works in People With Overweight or ObesityPHASE1 COMPLETED 144May 11, 2022Jan 9, 2024Jun 15, 20252 United States
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Study Endpoints
Primary Endpoints
The area under the ethinylestradiol plasma concentration time curve at steady state
Day 8 and Day 193

Measured as hours picograms per milliliter (h\*pg/mL).

The area under the levonorgestrel plasma concentration time curve at steady state
Day 8 and Day 193

Measured as hours picograms per milliliter (h\*pg/mL).

Number of treatment emergent adverse events (TEAE)
Part A: From pre-dose on Day 1 to 22 days; Part B: From pre-dose on Day 1 to 31 days; Part C and D: From pre-dose on Day 1 to 105 days

Number of events

Secondary Endpoints
Maximum ethinylestradiol plasma concentration at steady state
Day 8 and Day 193
Maximum levonorgestrel plasma concentration at steady state
Day 8 and Day 193
The area under the ethinylestradiol plasma concentration time curve at steady state
Day 8 and Day 135
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Study Design & Arms
AllocationNA
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
NNC0487-0111EXPERIMENTALParticipants will receive oral dosing of NNC0487-0111 and gradually will escalate from dose 1 to dose 2. The oral NNC0487-0111 treatment will be followed by s.c. NNC0487-0111 treatment with dose escalating from dose 3 to dose 4.
Part A: Single ascending dose (SAD)EXPERIMENTALParticipants will receive a single dose of any of the six different dose levels (1, 3, 6, 12, 25 and 50 milligrams (mg)) of NNC0487-0111 A or matching placebo in a sequential manner with the dose increasing between cohorts.
Part B: Multiple ascending dose (MAD)EXPERIMENTALParticipants will receive NNC0487-0111 once daily for 10 days at any of the five different dose levels (3, 6, 12, 25 and 50 milligrams (mg)) of NNC0487-0111 A or matching placebo in a sequential manner with the dose increasing between cohorts.
Part CEXPERIMENTALParticipants will receive NNC0487-0111 A or matching placebo once-daily for 12 weeks: 3 or 6 mg for weeks 1-2, 6 or 12 mg for weeks 3-4, 12 or 25 mg for weeks 5-6, 25 or 50 mg for weeks 7-8, 25 or 50 mg for weeks 9-10 and 50 or 2\*50 mg for weeks 11-12.
Part DEXPERIMENTALParticipants will receive NNC0487-0111 B or matching placebo once-daily for 12 weeks: 3 or 6 mg for weeks 1-2, 6 or 12 mg for weeks 3-4, 12 or 25 mg for weeks 5-6, 25 or 50 mg for weeks 7-8, 25 or 50 mg for weeks 9-10 and 50 or 2\*50 mg for weeks 11-12.
Interventions
NameTypeDescription
NNC0487-0111 ADRUGNNC0487-0111 A will be administered subcutaneously.
NNC0487-0111 CDRUGNNC0487-0111 C will be taken orally.
Levonorgestrel 150 μg + Ethinylestradiol 30 μg (Oral contraceptive OC)DRUGLevonorgestrel 150 μg + Ethinylestradiol 30 μg (Oral contraceptive OC) will be taken orally.
Acetaminophen - 500 mg/15 mlDRUGAcetaminophen - 500 mg/15 ml will be taken orally.
NNC0487-0111 BDRUGParticipants will receive NNC0487-0111 B tablet once daily.
Placebo B (NNC0487-0111 B)OTHERParticipants will receive placebo matched to NNC0487-0111 B tablet once daily.
Placebo A (NNC0487-0111 A)OTHERParticipants will receive placebo matched to NNC0487-0111 A tablet once daily.
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Eligibility Criteria
Age Range18 Years — 65 Years
SexFEMALE
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Females of non-childbearing potential. * Age 18 - 65 years (both inclusive) at the time of signing the informed consent. * Body mass index (BMI) between 25.0 and 39.9 kg/m\^2 (both inclusive) at screening. * Considered to be generally healthy based on the medical history, phys...

Countries:CanadaUnited States
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