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Beloranib

Phase 2

Obesity | Small molecule | Metabolic |Larimar Therapeutics, Inc.|Last Updated: Jul 14, 2016

Success Probability

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLEDDMC
Total Trials1
Total Enrollment160

FDA Designations

No designations recorded

Clinical trial landscape

Beloranib · 1 trial · 1 indication

Phase 2 1
NCT01666691An Efficacy, Safety and Pharmacokinetics Study of Beloranib (ZGN-440 for Injectable Suspension) in Obese SubjectsObesity
COMPLETED160 Analytics
PHASE2COMPLETED
An Efficacy, Safety and Pharmacokinetics Study of Beloranib (ZGN-440 for Injectable Suspension) in Obese Subjects
ObesityUnlock trial analytics

Study Endpoints

Primary Endpoints

Safety and tolerability of beloranib (ZGN-440 for injectable suspension) administered subcutaneously for 12 weeks
Up to 26 weeks

Safety and tolerability of beloranib will be assessed by comparing frequency and severity of adverse events as well as changes in physical examinations, ECGs, vital signs and laboratory evaluations. Other safety oriented questionnaires and parameters (e.g. sleep quality, hemodynamic parameters) will be measured and evaluated.

Weight loss and responses in metabolic biomarkers over a dose range of ZGN-440
Up to 13 weeks

Change from baseline in body weight and body composition (bioimpedance assessments), and scores of hunger/appetite over the dosing period will be evaluated to document beloranib's effect on obesity. Biomarkers of lipid metabolism will be measured to assess possible mechanisms of loss of body fat, as well as endocrinologic or anti-inflammatory markers.

Secondary Endpoints

Pharmacodynamics over a dose range of beloranib
Up to 12 weeks
Compare the plasma pharmacokinetic profile of beloranib administered subcutaneously with the profiles obtained previously using an alternative formulation administered subcutaneously and with ZGN-433 (beloranib hemioxalate) administered intravenously
Up to 12 weeks
Apparent bioavailability over a dose range of beloranib
Up to 12 weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
PlaceboPLACEBO_COMPARATORZGN-440 sterile diluent
0.3 mg BeloranibEXPERIMENTAL0.3 mg ZGN-440 for injectable suspension
0.6 mg BeloranibEXPERIMENTAL0.6 mg ZGN-440 for injectable suspension
1.2 mg BeloranibEXPERIMENTAL1.2 mg ZGN-440 for injectable suspension
2.4 mg BeloranibEXPERIMENTAL2.4 mg ZGN-440 for injectable suspension
3.2 mg BeloranibEXPERIMENTAL3.2 mg ZGN-440 for injectable suspension

Interventions

NameTypeDescription
BeloranibDRUGSubjects will receive ZGN-440 twice-weekly subcutaneous injections for up to 12 weeks and a total of 24 doses. A range of doses will be evaluated.
PlaceboDRUGSubjects will receive placebo twice-weekly subcutaneous injections for up to 12 weeks and a total of 24 doses.
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites3

Inclusion Criteria: * Obese volunteers weighing ≥ 50 kg * BMI ≥ 30 and ≤ 50 kg/m2 * Stable body weight during the past 2 months * Type 2 diabetes mellitus is allowed Exclusion Criteria: * Use of weight loss agents in the past month * Current, clinically significant eating disorder * Type 1 diabet...

Countries:Australia
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Frequently asked questions about Beloranib

What is Beloranib used for?

Beloranib is an investigational small molecule being developed for the treatment of obesity. It is a metabolic therapeutic that has been studied in a Phase 2 clinical trial. The drug is not approved and remains in clinical development.

Who makes Beloranib?

Beloranib is being developed by Larimar Therapeutics, Inc., a biopharmaceutical company traded on the Nasdaq under the ticker symbol LRMR. The company is conducting clinical research to evaluate the drug's safety and efficacy in obese subjects.

What phase is Beloranib in?

Beloranib is in Phase 2 clinical development. It has completed a Phase 2 trial in obese subjects. The drug is investigational and has not been approved by regulatory authorities for any use.

What clinical trials is Beloranib in?

Beloranib has been studied in one completed Phase 2 clinical trial, identified as NCT01666691. This randomized, double-blind, placebo-controlled study enrolled 160 obese subjects in Australia to evaluate the efficacy, safety, and pharmacokinetics of the drug.

Is Beloranib the same as ZGN-440?

Beloranib is also known as ZGN-440 for injectable suspension, as referenced in the clinical trial NCT01666691. This alternative name may be used in research publications and trial registries to refer to the same drug candidate.