Recent Updates
Recently added Catalysts

AZD4248

Phase 1

Chronic Kidney Disease | Small molecule | Nephrology |AstraZeneca PLC|Last Updated: Aug 12, 2026

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedDouble-BlindNO_TREATMENT_CONTROLLEDDMC
Total Trials1
Total Enrollment124

FDA Designations

No designations recorded

Clinical trial landscape

AZD4248 · 1 trial · 1 indication

Phase 1 1
NCT07024823A Study to Investigate Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of AZD4248 in Healthy Participants and Participants With Chronic Kidney Disease and Type 2 Diabetes and to Assess Home Measurements of Creatinine in a Non Interventional CohortChronic Kidney Disease
RECRUITING124 Analytics
PHASE1RECRUITING
A Study to Investigate Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of AZD4248 in Healthy Participants and Participants With Chronic Kidney Disease and Type 2 Diabetes and to Assess Home Measurements of Creatinine in a Non Interventional Cohort
Chronic Kidney DiseaseUnlock trial analytics

Study Endpoints

Primary Endpoints

Parts A, B, and C: Number of Participants with Adverse Events (AEs) and Serious Adverse Events (SAEs)
From Day 1 to Follow Up visit (Part A: up to 12 days; Part B and C: up to 19 days)

To assess the safety and tolerability of AZD4248 following single oral ascending doses or single IV administration to healthy participants and multiple oral ascending doses to healthy participants and participants with CKD and T2D (DKD).

Part D: Intra- and inter-participant variability of estimated glomerular filtration rate (eGFR) derived from home self-testing device measurements
Day 1 to Day 169

To assess intra- and inter-participant variability of twice weekly home-based serum creatinine measurements.

Secondary Endpoints

Area under concentration-time curve from time 0 to infinity (AUCinf)
Part A1 and A2: Days 1-7, Part A3: Days 1-3, Part B: Days 1-17. Part C: Days 1-17
Area under concentration-curve from time 0 to the last quantifiable concentration (AUClast)
Part A1 and A2: Days 1-7, Part A3: Days 1-3, Part B: Days 1-17. Part C: Days 1-17
Dose normalized AUClast (AUClast/D)
Part A1 and A2: Days 1-7, Part A3: Days 1-3, Part B: Days 1-17. Part C: Days 1-17
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part A1 SADEXPERIMENTALParticipants will receive single ascending oral dose of AZD4248 or placebo.
Part A2 SAD Chinese CohortEXPERIMENTALParticipants will receive single oral dose of AZD4248 or placebo.
Part A3 SAD IV CohortEXPERIMENTALParticipants will receive single IV infusion of AZD4248 or placebo.
Part B1 MADEXPERIMENTALParticipants will receive multiple ascending oral doses of AZD4248 or placebo.
Part B2 MAD JapaneseEXPERIMENTALParticipants will receive multiple ascending oral doses of AZD4248 or placebo.
Part C Multiple Dosing DKDEXPERIMENTALParticipants will receive multiple oral doses of AZD4248 or placebo.
Part D Observational CohortNO_INTERVENTIONParticipants will participate in home-based creatinine self-measurement.

Interventions

NameTypeDescription
AZD4248DRUGAZD4248 will be administered orally.
PlaceboDRUGPlacebo will be administered orally.
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 75 Years
SexALL
Healthy VolunteersYes
Study Sites5

Key Inclusion Criteria: \- Healthy participants with suitable veins for cannulation or repeated venipuncture. Parts A and B: * Have a body mass index (BMI) between 18 and 30 kilograms per millimeter (kg/m2), inclusive. * For Chinese participants (Part A2): participants are to be Chinese, defined ...

Countries:United States
Unlock Eligibility Criteria

Recent Changes (Last 90 Days)

LOWAug 12, 2026NCT07024823lastUpdatePostDate: changed
LOWAug 12, 2026NCT07024823lastUpdatePostDate: changed
MEDIUMJul 2, 2026NCT07024823primaryCompletionDate: changed
MEDIUMJul 2, 2026NCT07024823primaryCompletionDate: changed
MEDIUMJul 2, 2026NCT07024823primaryCompletionDate: changed
MEDIUMJul 2, 2026NCT07024823primaryCompletionDate: changed

Frequently asked questions about AZD4248

What is AZD4248 used for?

AZD4248 is an investigational small molecule being developed for the treatment of Chronic Kidney Disease. It is currently in Phase 1 clinical development, meaning it has not yet been approved by regulatory authorities and is still being studied for safety and efficacy in clinical trials.

Who makes AZD4248?

AZD4248 is being developed by AstraZeneca PLC, a biopharmaceutical company listed on the stock exchange under the ticker symbol AZN. The company is conducting clinical trials to evaluate the safety, tolerability, pharmacokinetics, and pharmacodynamics of this investigational drug.

What phase is AZD4248 in?

AZD4248 is currently in Phase 1 clinical development. This is the earliest stage of testing in humans, focused primarily on assessing the drug's safety, tolerability, and how it is processed by the body. It is not yet approved for any use and remains an investigational agent.

What clinical trials is AZD4248 in?

AZD4248 is being studied in a Phase 1 clinical trial registered as NCT07024823. This trial is recruiting participants and aims to investigate the safety, tolerability, pharmacokinetics, and pharmacodynamics of AZD4248 in healthy participants and in those with Chronic Kidney Disease and Type 2 Diabetes.

Is AZD4248 being tested in healthy volunteers?

Yes, the Phase 1 clinical trial of AZD4248, NCT07024823, includes healthy volunteers as well as participants with Chronic Kidney Disease and Type 2 Diabetes. The study is designed to evaluate the drug's safety and how it behaves in the body across these different groups.