Recent Updates
Recently added Catalysts

AMG 181

Phase 1

Ulcerative Colitis | Small molecule | Gastrointestinal |Amgen Inc.|Last Updated: Mar 17, 2015

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials1
Total Enrollment43

FDA Designations

No designations recorded

Clinical trial landscape

AMG 181 · 1 trial · 2 indications

Phase 1 1
NCT01290042Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of AMG 181.Ulcerative Colitis
COMPLETED43 Analytics
PHASE1COMPLETED
Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of AMG 181.
Ulcerative ColitisUnlock trial analytics

Study Endpoints

Primary Endpoints

To assess the number of adverse events per subject, after multiple subcutaneous doses of AMG 181 in in healthy subjects, in subjects with active ulcerative colitis, and in subjects with active Crohn's disease.
40 Weeks

Secondary Endpoints

To measure the area under the plasma concentration curve versus time of drug AMG 181.
29 Weeks
To assess receptor saturation percentages relative to baseline after multiple doses of AMG 181.
29 Weeks
To evaluate changes in peripheral blood T lymphocyte subsets counts relative to baseline after multiple doses of AMG 181.
29 weeks
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Placebo armACTIVE_COMPARATORFour escalating dose levels of AMG 181 administered as multiple doses of AMG 181 in healthy subjects, in subjects with active ulcerative colitis, and in subjects with active Crohn's disease.
Active armACTIVE_COMPARATORFour escalating dose levels of AMG 181 administered as multiple doses of AMG 181 in healthy subjects, in subjects with active ulcerative colitis, and in subjects with active Crohn's disease.

Interventions

NameTypeDescription
AMG 181DRUGFour escalating dose levels of AMG 181 administered as multiple doses of AMG 181 in healthy subjects, in subjects with active ulcerative colitis, and in subjects with active Crohn's disease.
Placebo for AMG 181OTHERFour escalating dose levels of AMG 181 administered as multiple doses of AMG 181 in healthy subjects, in subjects with active ulcerative colitis, and in subjects with active Crohn's disease.
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites8

Inclusion Criteria: * Body Mass Index (BMI) between 18 and 34 kg/m2 * Normal physical and neurological examination, clinical laboratory values and ECG * Ulcerative Colitis Disease Activity Index (UCDAI, aka Mayo score) score of 4 to 10 (inclusive), with a minimum sigmoidoscopy score of 1; (for subj...

Countries:United StatesAustralia
Unlock Eligibility Criteria

Frequently asked questions about AMG 181

What is AMG 181 used for?

AMG 181 is an investigational small molecule being developed for ulcerative colitis, a form of inflammatory bowel disease. It was studied in a Phase 1 clinical trial that also included patients with Crohn's disease, another inflammatory bowel condition. The drug is not approved and remains in clinical development.

Who makes AMG 181?

AMG 181 is being developed by Amgen Inc., a biopharmaceutical company traded on the NASDAQ under the ticker symbol AMGN. The company sponsored a Phase 1 clinical trial of the drug in patients with ulcerative colitis and Crohn's disease.

What phase is AMG 181 in?

AMG 181 is in Phase 1 clinical development. A Phase 1 study of the drug has been completed, and it is not approved for any use. The drug remains investigational, and no later-phase trials have been reported.

What clinical trials is AMG 181 in?

AMG 181 has one completed clinical trial, identified as NCT01290042, titled "Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of AMG 181." This Phase 1 study enrolled 43 participants with ulcerative colitis or Crohn's disease, as well as healthy volunteers, at sites in the United States and Australia.

Is AMG 181 the same as another drug?

AMG 181 is the only name provided for this drug, and no alternative names have been reported. It is an investigational small molecule developed by Amgen Inc. for ulcerative colitis and Crohn's disease.