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zosuquidar trihydrochloride

Phase 3

Leukemia | Small molecule | Oncology |Eli Lilly and Company|Last Updated: Jul 5, 2023

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLEDDMC
Total Trials1
Total Enrollment449

FDA Designations

No designations recorded

Clinical trial landscape

zosuquidar trihydrochloride · 1 trial · 2 indications

Phase 3 1
NCT00046930Daunorubicin & Cytarabine +/- Zosuquidar inTreating Older Patients With Newly Diagnosed Acute Myeloid Leukemia or Refractory AnemiaLeukemia
COMPLETED449 Analytics
PHASE3COMPLETED
Daunorubicin & Cytarabine +/- Zosuquidar inTreating Older Patients With Newly Diagnosed Acute Myeloid Leukemia or Refractory Anemia
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Study Endpoints

Primary Endpoints

Overall Survival (OS)
Assessed every 3 months for 2 years, then every 6 months for 3 years, then annually thereafter

Time from randomization to death. Patients alive at last follow-up were censored.

Secondary Endpoints

Progression-free Survival (PFS)
Assessed every 3 months for 2 years, then every 6 months for 3 years, then annually thereafter
Response
Assessed at the end of induction
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ZosuquidarEXPERIMENTALInduction treatment with daunorubicin, cytarabine and zosuquidar (details provided in Intervention section), followed by consolidation with Cytarabine (1500 mg/m2 every 12 hours for 6 days), then additional consolidation with the same regimen as received during induction.
PlaceboACTIVE_COMPARATORInduction treatment with daunorubicin, cytarabine and placebo (details provided in Intervention section), followed by consolidation with Cytarabine (1500 mg/m2 every 12 hours for 6 days), then additional consolidation with the same regimen as received during induction.

Interventions

NameTypeDescription
filgrastimBIOLOGICAL250 μg/m2/day by either intravenous or subcutaneous injection starting day 12, provided marrow aplasia is achieved, through recovery of absolute neutrophil count (ANC) to \> 500 cells/μl, sustained for 3 consecutive days. The dose may be rounded to the nearest vial size.
sargramostimBIOLOGICAL5 μg/kg/day by either intravenous or subcutaneous injection starting day 12, provided marrow aplasia is achieved, through recovery of absolute neutrophil count (ANC) to \> 500 cells/μl, sustained for 3 consecutive days. The dose may be rounded to the nearest vial size.
cytarabineDRUG100 mg/m²/day by continuous intravenous infusion for 7 days (days 1-7).
daunorubicin hydrochlorideDRUG45 mg/m²/day by 10 - 15 minute intravenous infusion for 3 days (days 1, 2, and 3).
zosuquidar trihydrochlorideDRUGZosuquidar 550 mg/day by continuous intravenous infusion through a central venous catheter over approximately 6 hours on days 1, 2, and 3. The infusion will begin approximately one hour prior to daunorubicin on days 1, 2 and 3.
PlaceboDRUGPlacebo 550 mg/day by continuous intravenous infusion through a central venous catheter over approximately 6 hours on days 1, 2, and 3. The infusion will begin approximately one hour prior to daunorubicin on days 1, 2 and 3. Placebo consisted of a 1:1000 dilution of Infuvite, appropriately colored.
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Eligibility Criteria

Age Range60 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites92

Inclusion Criteria: One of the following disorders: * Acute myeloid leukemia (AML), defined as \>30% myeloblasts on the marrow aspirate or peripheral blood differential and any French-American-British (FAB) subtype except M3 (i.e., acute promyelocytic leukemia) * Refractory anemia with excess blas...

Countries:United StatesIsrael
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