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SPC ezetimibe/rosuvastatin

Phase 3

Hypercholesterolemia | Small molecule | Metabolic |Sanofi|Last Updated: Sep 22, 2025

Success Probability

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials1
Total Enrollment305

FDA Designations

No designations recorded

Clinical trial landscape

SPC ezetimibe/rosuvastatin · 1 trial · 1 indication

Phase 3 1
NCT04669041A Study to Evaluate the Efficacy and the Safety of Single Pill Combination (SPC) Ezetimibe/Rosuvastatin in Chinese Adult Patients With Primary Hypercholesterolemia Not Adequately Controlled on Statin TherapyHypercholesterolemia
COMPLETED305 Analytics
PHASE3COMPLETED
A Study to Evaluate the Efficacy and the Safety of Single Pill Combination (SPC) Ezetimibe/Rosuvastatin in Chinese Adult Patients With Primary Hypercholesterolemia Not Adequately Controlled on Statin Therapy
HypercholesterolemiaUnlock trial analytics

Study Endpoints

Primary Endpoints

Percent change in measured LDL-C from baseline (the last available measured LDL-C value obtained up to randomization) to Week 8
Baseline to Week 8

The percent change from baseline in measured LDL-C at Week 8 will be analyzed in the modified intent-to-treat (mITT) population using a mixed effect model with repeated measures (MMRM) approach.

Secondary Endpoints

Proportion of patients who attain lipid goal (measured LDL-C <2.6 mmol/L [100 mg/dL]) at Week 8
Week 8
Percent change in measured LDL-C plasma level from baseline to Week 4
Baseline to Week 4
Percent change in total cholesterol (TC) from baseline to Week 8
Baseline to Week 8
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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Single pill combination (SPC)EXPERIMENTALOnce daily rosuvastatin 10 mg for 4 weeks, then once daily SPC ezetimibe 10 mg /rosuvastatin 10 mg (E10/R10) for 8 weeks
RosuvastatinACTIVE_COMPARATOROnce daily rosuvastatin 10 mg for 4 weeks, then once daily rosuvastatin 10 mg (R10) for 8 weeks

Interventions

NameTypeDescription
RosuvastatinDRUGPharmaceutical form:Tablet Route of administration: Oral
SPC ezetimibe/rosuvastatinDRUGPharmaceutical form:Tablet Route of administration: Oral
Rosuvastatin active capsuleDRUGPharmaceutical form:Capsule Route of administration: Oral
PlaceboDRUGPharmaceutical form:Tablet Route of administration: Oral
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites40

Inclusion criteria : * Participant must be at least 18 years of age inclusive, at the time of signing the informed consent. * Patients with primary hypercholesterolemia. * Inclusion criteria in the run-in period: Participants who are not adequately controlled (defined by screening LDL-C \>2.6 mmol/...

Countries:China
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Frequently asked questions about SPC ezetimibe/rosuvastatin

What is SPC ezetimibe/rosuvastatin used for?

SPC ezetimibe/rosuvastatin is a single pill combination used for hypercholesterolemia, specifically in Chinese adult patients with primary hypercholesterolemia not adequately controlled on statin therapy. It is a small molecule being developed by Sanofi and is currently in Phase 3 clinical development.

What does SPC ezetimibe/rosuvastatin target?

SPC ezetimibe/rosuvastatin combines two active ingredients: ezetimibe, which inhibits cholesterol absorption in the intestine, and rosuvastatin, a statin that inhibits HMG-CoA reductase to reduce cholesterol synthesis. Together they lower LDL cholesterol levels in patients with hypercholesterolemia.

Who makes SPC ezetimibe/rosuvastatin?

SPC ezetimibe/rosuvastatin is being developed by Sanofi, a multinational pharmaceutical company listed on the stock exchange under the ticker SNY. The drug is currently in Phase 3 clinical development for the treatment of hypercholesterolemia.

What phase is SPC ezetimibe/rosuvastatin in?

SPC ezetimibe/rosuvastatin is in Phase 3 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 3 trial has been completed, with 305 participants enrolled.

What clinical trials is SPC ezetimibe/rosuvastatin in?

SPC ezetimibe/rosuvastatin has one completed Phase 3 trial, NCT04669041, which evaluated its efficacy and safety in Chinese adult patients with primary hypercholesterolemia not adequately controlled on statin therapy. The trial enrolled 305 participants and was randomized, double-blind, and active-controlled.

Is SPC ezetimibe/rosuvastatin the same as ezetimibe/rosuvastatin?

SPC ezetimibe/rosuvastatin is a single pill combination (SPC) of ezetimibe and rosuvastatin. It is a fixed-dose combination product that contains both active ingredients in one tablet, as opposed to taking them as separate medications.