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SPC ezetimibe/rosuvastatin

Phase 3

Hypercholesterolemia | Small molecule | Metabolic |Sanofi|Last Updated: Sep 22, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindACTIVE_CONTROLLEDBiomarker
Total Trials1
Total Enrollment305
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04669041A Study to Evaluate the Efficacy and the Safety of Single Pill Combination (SPC) Ezetimibe/Rosuvastatin in Chinese Adult Patients With Primary Hypercholesterolemia Not Adequately Controlled on Statin TherapyPHASE3 COMPLETED 305Dec 8, 2020Jun 15, 2022Sep 22, 202540 China
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Study Endpoints
Primary Endpoints
Percent change in measured LDL-C from baseline (the last available measured LDL-C value obtained up to randomization) to Week 8
Baseline to Week 8

The percent change from baseline in measured LDL-C at Week 8 will be analyzed in the modified intent-to-treat (mITT) population using a mixed effect model with repeated measures (MMRM) approach.

Secondary Endpoints
Proportion of patients who attain lipid goal (measured LDL-C <2.6 mmol/L [100 mg/dL]) at Week 8
Week 8
Percent change in measured LDL-C plasma level from baseline to Week 4
Baseline to Week 4
Percent change in total cholesterol (TC) from baseline to Week 8
Baseline to Week 8
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Single pill combination (SPC)EXPERIMENTALOnce daily rosuvastatin 10 mg for 4 weeks, then once daily SPC ezetimibe 10 mg /rosuvastatin 10 mg (E10/R10) for 8 weeks
RosuvastatinACTIVE_COMPARATOROnce daily rosuvastatin 10 mg for 4 weeks, then once daily rosuvastatin 10 mg (R10) for 8 weeks
Interventions
NameTypeDescription
RosuvastatinDRUGPharmaceutical form:Tablet Route of administration: Oral
SPC ezetimibe/rosuvastatinDRUGPharmaceutical form:Tablet Route of administration: Oral
Rosuvastatin active capsuleDRUGPharmaceutical form:Capsule Route of administration: Oral
PlaceboDRUGPharmaceutical form:Tablet Route of administration: Oral
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites40

Inclusion criteria : * Participant must be at least 18 years of age inclusive, at the time of signing the informed consent. * Patients with primary hypercholesterolemia. * Inclusion criteria in the run-in period: Participants who are not adequately controlled (defined by screening LDL-C \>2.6 mmol/...

Countries:China
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