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Obicetrapib

Phase 3

Atherosclerotic Cardiovascular Disease | Small molecule | Cardiovascular |NewAmsterdam Pharma Company N.V.|Last Updated: Oct 19, 2025

Target and mechanism

Molecular targetCETP
Target classInhibitor
ModalitySmall molecule

Also known as Obicetrapib 10mg

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment9,541

FDA Designations

No designations recorded

Clinical trial landscape

Obicetrapib · 14 trials · 17 indications

Phase 3 3Phase 2 6Phase 1 5
NCT05425745Evaluate the Effect of Obicetrapib in Patients With HeFH on Top of Maximum Tolerated Lipid-Modifying Therapies.Dyslipidemias
COMPLETED354 Analytics
NCT05202509Cardiovascular Outcome Study to Evaluate the Effect of Obicetrapib in Patients With Cardiovascular DiseaseAtherosclerotic Cardiovascular Disease
ACTIVE NOT_RECRUITING9,541 Analytics
NCT05142722Randomized Study to Evaluate the Effect of Obicetrapib on Top of Maximum Tolerated Lipid-Modifying TherapiesDyslipidemias
COMPLETED2,530 Analytics
PHASE3COMPLETED
Evaluate the Effect of Obicetrapib in Patients With HeFH on Top of Maximum Tolerated Lipid-Modifying Therapies.
DyslipidemiasUnlock trial analytics
PHASE3ACTIVE NOT_RECRUITING
Cardiovascular Outcome Study to Evaluate the Effect of Obicetrapib in Patients With Cardiovascular Disease
Atherosclerotic Cardiovascular DiseaseUnlock trial analytics
PHASE3COMPLETED
Randomized Study to Evaluate the Effect of Obicetrapib on Top of Maximum Tolerated Lipid-Modifying Therapies
DyslipidemiasUnlock trial analytics

Study Design & Arms

Interventions

NameTypeDescription
ObicetrapibDRUG10 mg Obicetrapib tablet
PlaceboDRUGplacebo tablet made to resemble active
Obicetrapib 10mgDRUGActive Drug
Ezetimibe 10mgDRUGcapsules; 10 mg ezetimibe tablets filled into capsule shells, 1 tablet per capsule.
Obicetrapib placeboOTHERtablets; no active ingredient
Ezetimibe placeboOTHERcapsules; no active ingredient
Obicetrapib 5mgDRUGtablet
Obicetrapib + Drospirenone / Ethinyl Estradiol (COC)DRUGoral administration
Drospirenone / Ethinyl Estradiol (COC)DRUGoral administration
Atorvastatin CalciumDRUGAtorvastatin 80 mg
Rosuvastatin CalciumDRUGRosuvastatin 40 mg
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Frequently asked questions about Obicetrapib

What is Obicetrapib used for?

Obicetrapib is an investigational small molecule being studied for dyslipidemia, high cholesterol, and hypercholesterolemia, as well as early Alzheimer's disease, antioxidant absorption, hepatic impairment, and lipid metabolism. It is also evaluated in healthy volunteers. The drug is in Phase 2 clinical development and is not yet approved.

What does Obicetrapib target?

Obicetrapib targets cholesteryl ester transfer protein (CETP) and acts as a CETP inhibitor. By inhibiting CETP, it is designed to affect lipid metabolism, which is relevant to its study in dyslipidemia and related cholesterol conditions.

Who makes Obicetrapib?

Obicetrapib is being developed by NewAmsterdam Pharma Company N.V., a biopharmaceutical company. The company's stock is listed under the ticker symbol NAMS.

What phase is Obicetrapib in?

Obicetrapib is in Phase 2 clinical development. It is an investigational drug and has not received FDA approval. Several Phase 2 trials have been completed, and the drug continues to be studied for various indications.

What clinical trials is Obicetrapib in?

Obicetrapib has been studied in several Phase 2 trials, including NCT04753606, a randomized study as an adjunct to statin therapy; NCT05161715, a proof-of-concept study in early Alzheimer's disease; NCT05266586, a study combining obicetrapib with ezetimibe; and NCT05421078, a dose-finding study in Japanese patients.

Is Obicetrapib the same as other formulations?

Obicetrapib is known by several names, including obicetrapib 10mg, obicetrapib 10 mg plus obicetrapib/evolocumab 140 mg every 2 weeks, obicetrapib 10 mg plus ezetimibe 10 mg fixed-dose combination daily, and obicetrapib plus ezetimibe daily. These refer to different dosing regimens or combinations being studied.