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RO7616789

Phase 1

Small Cell Lung Cancer | Small molecule | Oncology |Roche Holding AG|Last Updated: Mar 10, 2025

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment41

FDA Designations

No designations recorded

Clinical trial landscape

RO7616789 · 1 trial · 2 indications

Phase 1 1
NCT05619744A Study to Evaluate Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Preliminary Anti-tumor Activity of RO7616789 in Advanced Small Cell Lung Cancer and Other Neuroendocrine CarcinomasSmall Cell Lung Cancer
COMPLETED41 Analytics
PHASE1COMPLETED
A Study to Evaluate Safety, Tolerability, Pharmacokinetics, Pharmacodynamics, and Preliminary Anti-tumor Activity of RO7616789 in Advanced Small Cell Lung Cancer and Other Neuroendocrine Carcinomas
Small Cell Lung CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Part 1, 2 and 3: Number of Participants with Adverse Events and Serious Adverse Events
Up to approximately 26 months

Adverse events were reported according to the National Cancer Institute Common Terminology Criteria for Adverse Events, Version 5.0 (NCI CTCAE v5.0), and Cytokine release syndrome (CRS), will be graded based on the American Society for Transplantation and Cell Therapy (ASTCT) criteria.

Part 1 and 2: Number of Participants with Dose Limiting Toxicities (DLTs)
Day 1 through Day 21 in cycle 1 (Cycle is 21 days)
Part 3: Objective Response Rate (ORR) as determined by Investigator
Up to approximately 26 months
Part 3: Disease Control Rates as Determined by the Investigator
Up to approximately 26 months
Part 3: Duration of Response (DOR) as Determined by the Investigator
Up to approximately 26 months
Part 3: Progression Free Survival (PFS) as Determined by the Investigator
Up to approximately 26 months
Part 3: Overall Survival (OS)
Up to approximately 26 months

Secondary Endpoints

Part 1, 2 and 3: Serum Concentration of RO7616789
Up to approximately 26 months
Part 1, 2 and 3: Maximum Serum Concentration (Cmax) of RO7616789
Up to approximately 26 months
Part 1, 2 and 3: Area Under the Concentration-Time Curve (AUC) of RO7616789
Up to approximately 26 months
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part 1: RO7616789 QW: Dose EscalationEXPERIMENTALParticipants will receive a fixed dose of RO7616789 intravenously once weekly (QW) per dose level on Day 1, 8, and 15 of each 21-day cycle. In case of toxicity, step-up (single or double) dosing may be explored.
Part 2: RO7616789 Q3W: Dose EscalationEXPERIMENTALParticipants will receive a fixed dose of RO7616789, at a dose determined in Part 1, intravenously once every 3 weeks (Q3W) on Day 1 of each 21-day cycle. In case of toxicity, step-up (single or double) dosing may be explored.
Part 3: Dose ExpansionEXPERIMENTALBased on emerging data from Part 1 and 2, one or more dosing regimens will be further investigated in Part 3.

Interventions

NameTypeDescription
RO7616789DRUGRO7616789 solution for infusion will be administered intravenously at a dose and per schedule as specified for the respective part.
TocilizumabDRUGTocilizumab will be used as rescue therapy, in case of clinical presentation of cytokine release syndrome (CRS). Tocilizumab solution for infusion will be administered intravenously at 8 mg/kg for participants \>/= 30 kg or at 12 mg/kg for participants \< 30 kg.
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites17

Inclusion Criteria: * Life expectancy at least 12 weeks * Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1 * Adequate hematologic and end organ function * Negative serum pregnancy test. * Adequate contraception and no or interruption of breastfeeding * Histologically confirmed...

Countries:United StatesDenmarkJapanPolandSpain
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Competitive Landscape -Non-Small Cell Lung Cancer 389 trials (matched to "Small Cell Lung Cancer")

Frequently asked questions about RO7616789

What is RO7616789 used for?

RO7616789 is an investigational small molecule being studied for the treatment of advanced small cell lung cancer and other neuroendocrine carcinomas. It is currently in Phase 1 clinical development and has not been approved by regulatory authorities.

What does RO7616789 target?

The molecular target of RO7616789 has not been disclosed in available information. It is being evaluated for its safety, tolerability, pharmacokinetics, pharmacodynamics, and preliminary anti-tumor activity in patients with advanced small cell lung cancer and other neuroendocrine carcinomas.

Who makes RO7616789?

RO7616789 is being developed by Roche Holding AG, which trades on the OTC market under the ticker RHHBY. The company is conducting clinical trials to evaluate the drug's safety and preliminary efficacy in oncology indications.

What phase is RO7616789 in?

RO7616789 is in Phase 1 clinical development. It is an investigational drug and has not been approved by the FDA or other regulatory agencies. The drug is being studied for safety, tolerability, and preliminary anti-tumor activity in advanced small cell lung cancer and neuroendocrine carcinomas.

What clinical trials is RO7616789 in?

RO7616789 has been studied in one completed Phase 1 clinical trial, NCT05619744. This trial evaluated the drug in 41 patients with advanced small cell lung cancer and neuroendocrine carcinomas across the United States, Denmark, Japan, Poland, and Spain.