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Etrozulimab

Phase 3

Ulcerative Colitis | Small molecule | Gastrointestinal |Roche Holding AG|Last Updated: Aug 13, 2021

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment609

FDA Designations

No designations recorded

Clinical trial landscape

Etrozulimab · 1 trial · 1 indication

Phase 3 1
NCT02100696A Study of the Efficacy and Safety of Etrolizumab in Participants With Ulcerative Colitis Who Have Been Previously Exposed to Tumor Necrosis Factor (TNF) InhibitorsUlcerative Colitis
COMPLETED609 Analytics
PHASE3COMPLETED
A Study of the Efficacy and Safety of Etrolizumab in Participants With Ulcerative Colitis Who Have Been Previously Exposed to Tumor Necrosis Factor (TNF) Inhibitors
Ulcerative ColitisUnlock trial analytics

Study Endpoints

Primary Endpoints

Induction Phase: Percentage of Participants With Remission at Week 14, as Determined by the Mayo Clinic Score (MCS)
Week 14

The Mayo Clinic Score (MCS) ranges from 0 to 12 and is a composite of 4 assessments (each rated from 0-3): stool frequency, rectal bleeding, endoscopy, and physician's global assessment. Higher scores represent greater disease severity. Remission was defined as MCS less than or equal to (≤)2 with individual subscores ≤1 and a rectal bleeding subscore of 0.

Maintenance Phase: Percentage of Participants With Remission at Week 66 Among Participants Who Had Achieved a Clinical Response at Week 14, as Determined by the MCS
Week 66

The MCS ranges from 0 to 12 and is a composite of 4 assessments (each rated from 0-3): stool frequency, rectal bleeding, endoscopy, and physician's global assessment. Higher scores represent greater disease severity. Remission was defined as MCS less than or equal to (≤)2 with individual subscores ≤1 and a rectal bleeding subscore of 0. Clinical Response is MCS with ≥3-point decrease and 30% reduction from baseline as well as ≥1-point decrease in rectal bleeding subscore or an absolute rectal bleeding score of 0 or 1.

Secondary Endpoints

Induction Phase: Percentage of Participants With Clinical Remission at Week 14, as Determined by the MCS
Week 14
Induction Phase: Percentage of Participants With Clinical Response at Week 14, as Determined by the MCS
Week 14
Induction Phase: Percentage of Participants With Improvement From Baseline in Endoscopic Appearance of the Mucosa at Week 14, as Determined by the MCS Endoscopic Subscore
Baseline and Week 14
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Cohort 1: Etrolizumab (Open-Label Induction (OLI) Phase)EXPERIMENTALParticipants assigned to this arm will receive treatment with open-label etrolizumab 105 milligrams (mg) subcutaneous (SC) injection once every 4 weeks (Q4W) for 14 weeks during the induction phase.
Cohort 2: Placebo (Double-Blind Induction Phase)PLACEBO_COMPARATORParticipants randomized to this arm will receive treatment with double-blind placebo SC injection Q4W for 14 weeks during the induction phase.
Cohort 2: Etrolizumab (Double-Blind Induction Phase)EXPERIMENTALParticipants randomized to this arm will receive treatment with double-blind etrolizumab 105 mg SC injection Q4W for 14 weeks during the induction phase.
Placebo Responders: Placebo (Maintenance Phase)PLACEBO_COMPARATORParticipants who received placebo during the induction phase, Cohort 2: Placebo (Double-Blind Induction Phase), and achieve a clinical response with placebo at Week 14 will continue to receive blinded placebo from Week 16 up to Week 66 during the maintenance phase.
Etrolizumab Responders: Placebo (Maintenance Phase)PLACEBO_COMPARATORParticipants who received etrolizumab during the induction phase, Cohort 1: Etrolizumab (Open-Label Induction Phase) and Cohort 2: Etrolizumab (Double-Blind Induction Phase), and achieved a clinical response at Week 14 will be re-randomized by Week 16 for the double-blind maintenance phase. Clinical responders re-randomized to this arm will receive placebo SC injection Q4W from Week 16 up to Week 66.
Etrolizumab Responders: Etrolizumab (Maintenance Phase)EXPERIMENTALParticipants who received etrolizumab during the induction phase, Cohort 1: Etrolizumab (Open-Label Induction Phase) and Cohort 2: Etrolizumab (Double-Blind Induction Phase), and achieved a clinical response at Week 14 will be re-randomized by Week 16 for the double-blind maintenance phase. Clinical responders re-randomized to this arm will receive etrolizumab 105 mg SC injection Q4W from Week 16 up to Week 66.

Interventions

NameTypeDescription
EtrozulimabDRUGParticipants will receive 105 mg etrolizumab administered by SC injection Q4W.
PlaceboDRUGParticipants will receive placebo (matched with etrolizumab) administered by SC injection Q4W.
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Eligibility Criteria

Age Range18 Years to 80 Years
SexALL
Healthy VolunteersNo
Study Sites184

Inclusion Criteria: * Diagnosis of UC established at least 3 months prior to Day 1 * Moderately to severely active UC as determined by the Mayo Clinic Score (MCS) assessment * Treatment within 5 years prior to screening with one or two induction regimens that contain TNF inhibitors (including TNF i...

Countries:United StatesArgentinaAustraliaAustriaBelgiumBrazilCanadaCzechiaDenmarkFranceGermanyGreeceHungaryIsraelItalyLithuaniaMexicoNetherlandsPolandRomaniaSouth KoreaSpainSwitzerlandUnited Kingdom
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Frequently asked questions about Etrozulimab

What is Etrozulimab used for?

Etrozulimab is an investigational small molecule being studied for the treatment of ulcerative colitis, a form of inflammatory bowel disease. It is being developed by Roche Holding AG. The drug is currently in Phase 3 clinical development, meaning it is still being tested and is not yet approved for use.

What does Etrozulimab target?

The specific molecular target of Etrozulimab has not been disclosed in available information. The drug is a small molecule being developed by Roche Holding AG for ulcerative colitis. It is currently in Phase 3 clinical trials, but its mechanism of action has not been publicly detailed.

Who makes Etrozulimab?

Etrozulimab is being developed by Roche Holding AG, a multinational healthcare company. Roche is conducting clinical trials to evaluate the drug's safety and efficacy in patients with ulcerative colitis. The drug is currently in Phase 3 development, and Roche is the sponsor of the ongoing research.

What phase is Etrozulimab in?

Etrozulimab is in Phase 3 clinical development. It is an investigational drug being studied for the treatment of ulcerative colitis. The drug is not yet approved by regulatory authorities, and its safety and efficacy are still being evaluated in clinical trials.

What clinical trials is Etrozulimab in?

Etrozulimab has been studied in one Phase 3 clinical trial with the identifier NCT02100696. This completed trial enrolled 609 participants with ulcerative colitis who had previously been exposed to TNF inhibitors. The study was randomized, double-blind, and placebo-controlled, and it took place across multiple countries including the United States.

Is Etrozulimab the same as etrolizumab?

Yes, Etrozulimab is the same as etrolizumab. The drug is also known by the name etrolizumab, and both names refer to the same investigational therapy being developed by Roche Holding AG for ulcerative colitis. It is currently in Phase 3 clinical development.