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RX-3117

Phase 1

Metastatic Pancreatic Cancer | Small molecule | Oncology |Processa Pharmaceuticals, Inc.|Last Updated: Dec 6, 2023

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment46

FDA Designations

No designations recorded

Clinical trial landscape

RX-3117 · 2 trials · 3 indications

Phase 1 2
NCT03189914RX-3117 in Combination With Abraxane® in Subjects With Metastatic Pancreatic CancerMetastatic Pancreatic Cancer
COMPLETED46 Analytics
NCT02030067Dose-Finding and Safety Study for Oral Single-Agent to Treat Advanced MalignanciesSolid Tumor
COMPLETED127 Analytics
PHASE1COMPLETED
RX-3117 in Combination With Abraxane® in Subjects With Metastatic Pancreatic Cancer
Metastatic Pancreatic CancerUnlock trial analytics
PHASE1COMPLETED
Dose-Finding and Safety Study for Oral Single-Agent to Treat Advanced Malignancies
Solid TumorUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of Participants With Treatment-related Adverse Events as Assessed by CTCAE v4.0 (Phase 1 and 2)
9 months

Number of participants who experienced a treatment-related adverse event

Number of Participants With Clinical Laboratory Abnormalities (Phase 1 and 2)
9 months

Participants with adverse events coded using the MedDRA Dictionary (Version 20.0) to Investigations. Due to the underlying disease, not all abnormal labs are reported.

Number of Participants With Vital Sign Abnormalities (Phase 1 and 2)
9 months

Number of participants with clinically significant vital sign abnormalities (Phase 1 and 2) including heart rate, respiration rate, and blood pressure

Number of Participants With Electrocardiogram (ECG) Abnormalities (Phase 1 and 2)
1 month

Number of participants with clinically significant ECG abnormalities (Phase 1 and 2)

Number of Dose-limiting Toxicities (DLTs) (Phase 1)
4 weeks
Number of Participants With Progression Free Survival (PFS) and/or Objective Clinical Response (Phase 2)
9 months

Participants must have progression Free Survival (PFS) \> 4 months or objective clinical response (complete or partial response).

Overall Safety Profile Characterized by # of Subjects With Dose-limiting Toxicities (DLTs) in Phase 1
28 days

Number of subjects participating in Phase 1 that experienced a DLT during the first cycle of treatment (28 days)

Overall Safety Profile Characterized by Number of Subjects Experiencing Serious Adverse Events in Phase 1
through study completion, up to 224 days (8 cycles of treatment)

Number of subjects participating in Phase 1 that experience any SAEs

Overall Safety Profile Characterized by the Number of Subjects That Discontinue Study Treatment - Phase 1
through study completion, up to 224 days (8 cycles of treatment)

Number of subjects participating in Phase 1 of study that discontinued study treatment due to a treatment emergent adverse event.

Overall Safety Profile Characterized by Number of Subjects Experiencing a Treatment Emergent Adverse Event- Phase 1
through study completion, up to 224 days (8 cycles of treatment)

Number of subjects that experience any treatment-related adverse event.

Progression Free Survival (Phase 2)
4 months

Progression Free Survival in Phase 2 of the study for pancreatic and bladder cancer subjects.

Secondary Endpoints

Area Under the Plasma Concentration Versus Time Curve (AUC) of RX-3117 (Phase 1 and Phase 2) - Day 1
Cycle 1 Day 1 (pre-infusion, post-infusion, pre-dose RX-3117, and 0.5, 1, 2, 4, 6, and 24 hours after administration)
Time to Maximum Observed Concentration [Tmax] of RX-3117 (Phase 1 and Phase 2) - Day 1
Cycle 1 Days 1 (pre-infusion, post-infusion, pre-dose RX-3117, and 0.5, 1, 2, 4, 6, and 24 hours after administration)
Maximum Observed Concentration [Cmax] of RX-3117 (Phase 1 and Phase 2) - Day 1
Cycle 1 Days 1 (pre-infusion, post-infusion, pre-dose RX-3117, and 0.5, 1, 2, 4, 6, and 24 hours after administration)
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
RX-3117 + AbraxaneEXPERIMENTALRX-3117: oral, 500 - 700 mg/ day for 5 days on/ 2 days off for 3 weeks. 1 washout week/ cycle. Abraxane: 75 - 125 mg/m\^2, infused once per week for 3 weeks. 1 washout week/ cycle.
RX-3117EXPERIMENTALAll subjects will receive RX-3117.

Interventions

NameTypeDescription
RX-3117DRUGRX-3117 will be administered orally in combination with Abraxane.
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites10

Inclusion Criteria: Disease Related 1. Subject has confirmed histologic or cytologic evidence of metastatic pancreatic cancer and has no prior treatment for metastatic pancreatic cancer. 2. Subject has measurable disease using Response Evaluation Criteria in Solid Tumors (RECIST) v 1.1. 3. Subject...

Countries:United States
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Competitive Landscape -Pancreatic Cancer 179 trials (matched to "Metastatic Pancreatic Cancer")

Top 20 of 68 competitors

CompanyTickerTrialsLead PhaseDrugs
Revolution Medicines, Inc.RVMD9PHASE3RMC-6236, Gemcitabine, nab-paclitaxel, Irinotecan, Liposomal irinotecan
Arcus Biosciences, Inc.RCUS3PHASE3Quemliclustat, Nab-paclitaxel, Gemcitabine
Pfizer Inc.PFE7PHASE2tisotumab vedotin, pembrolizumab, carboplatin, cisplatin
AstraZeneca PLCAZN9PHASE2AZD0901, 5-Fluorouracil, Leucovorin, l-leucovorin, Irinotecan
AbbVie, Inc.ABBV4PHASE2TTX-030, nab-paclitaxel and gemcitabine, Nab-Paclitaxel and gemcitabine
AngioDynamics, Inc.ANGO2PHASE3Modified FOLFIRINOX Regimen
Bristol-Myers Squibb CompanyBMY4PHASE2Navlimetostat, Gemcitabine, Nab-paclitaxel
Immuneering Corp. Class AIMRX2PHASE3Atebimetinib, GnP, mGnP
RenovoRx, Inc.RNXT1PHASE3Gemcitabine, nab-paclitaxel
BioNTech SE Sponsored ADRBNTX2PHASE2Pumitamig, Nab-paclitaxel, Gemcitabine, mFOLFIRINOX
Veracyte, Inc.VCYT1PHASE3Tislelizumab
ArriVent BioPharma, Inc.AVBP3PHASE2JAB-21822
Merck & Co., Inc.MRK2PHASE2Belzutifan
Eli Lilly and CompanyLLY7PHASE1LY4101174
Exelixis, Inc.EXEL1PHASE2Zanzalintinib, Everolimus
Agenus Inc.AGEN4PHASE2AGEN1423, Botensilimab, Gemcitabine, Nab-paclitaxel
HUTCHMED (China) Limited Sponsored ADRHCM1PHASE2Surufatinib Combined With Camrelizumab, Nab-paclitaxel, and Gemcitabine, Nab-paclitaxel Plus Gemcitabine, Surufatinib with Nab-paclitaxel, and Gemcitabine
Incyte CorporationINCY3PHASE2Ruxolitinib, Capecitabine, Regorafenib
Jazz Pharmaceuticals Public Limited CompanyJAZZ1PHASE2Zanidatamab
ImmunityBio IncIBRX1PHASE2N-803, Aldoxorubicin, PD-L1 t-haNK, Nab-paclitaxel, Gemcitabine
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Frequently asked questions about RX-3117

What is RX-3117 used for?

RX-3117 is an investigational small molecule being developed for the treatment of metastatic pancreatic cancer and solid tumors. It is currently in Phase 1 clinical development and has not been approved by the FDA. The drug is being studied in patients with advanced malignancies, including metastatic bladder cancer.

What does RX-3117 target?

RX-3117 is a small molecule, but its specific molecular target has not been disclosed. The drug is being evaluated in Phase 1 clinical trials for its safety and efficacy in treating solid tumors and metastatic pancreatic cancer. Its mechanism of action is not publicly detailed in the available information.

Who makes RX-3117?

RX-3117 is being developed by Processa Pharmaceuticals, Inc., a biopharmaceutical company traded on the Nasdaq under the ticker symbol PCSA. The company is conducting clinical trials to evaluate the drug's safety and efficacy in oncology indications.

What phase is RX-3117 in?

RX-3117 is in Phase 1 clinical development. It is an investigational drug and has not received FDA approval. Two Phase 1 trials have been completed, including a dose-finding study in advanced malignancies and a combination study with Abraxane in metastatic pancreatic cancer.

What clinical trials is RX-3117 in?

RX-3117 has been studied in two completed Phase 1 trials. NCT02030067 was a dose-finding and safety study of oral single-agent RX-3117 in advanced malignancies, enrolling 127 patients. NCT03189914 evaluated RX-3117 in combination with Abraxane in metastatic pancreatic cancer, enrolling 46 patients.

Is RX-3117 the same as any other drug?

RX-3117 is not known to have any alternative names. It is being developed as a single agent and in combination with Abraxane for the treatment of solid tumors and metastatic pancreatic cancer. No other names for this drug have been reported.