Recent Updates
Recently added Catalysts

SCH 58235

Phase 1

Hypercholesterolemia | Small molecule | Metabolic |Organon & Co.|Last Updated: Feb 16, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
RandomizedACTIVE_CONTROLLED
Total Trials1
Total Enrollment18
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00653913Evaluation of Potential for Drug Interaction Between SCH 58235 (Ezetimibe) and Pitavastatin (Study P03962)(COMPLETED)PHASE1 COMPLETED 18Mar 1, 2004Sep 1, 2004Feb 16, 2022 -
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Compare plasma concentrations of SCH 58235 (ezetimibe) and pitavastatin after administration of each drug alone and in combination, using Cmax and AUC(0-24h).
Day 7 of each period
Secondary Endpoints
Compare plasma concentrations of SCH 58235 (ezetimibe) and pitavastatin administration of each drug alone and in coadministration, using Tmax, plasma concentration 24 h after last dose, and AUC(I).
Day 7 of each period
Adverse events, laboratory tests results, and vital signs.
Throughout study
Unlock Study Endpoints
Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Group AACTIVE_COMPARATORSCH 58235 (Period 1) Pitavastatin (Period 2) Coadministration (Period 3)
Group BACTIVE_COMPARATORSCH 58235 (Period 1) Coadministration (Period 2) Pitavastatin (Period 3)
Group CACTIVE_COMPARATORPitavastatin (Period 1) SCH 58235 (Period 2) Coadministration (Period 3)
Group DACTIVE_COMPARATORPitavastatin (Period 1) Coadministration (Period 2) SCH 58235 (Period 3)
Group EACTIVE_COMPARATORCoadministration (Period 1) SCH 58235 (Period 2) Pitavastatin (Period 3)
Group FACTIVE_COMPARATORCoadministration (Period 1) Pitavastatin (Period 2) SCH 58235 (Period 3)
Interventions
NameTypeDescription
SCH 58235DRUGSCH 58235 10 mg (once daily)
pitavastatinDRUGPitavastatin 2 mg (once daily)
Unlock Study Design Details
Eligibility Criteria
Age Range20 Years — 65 Years
SexMALE
Healthy VolunteersYes

Inclusion Criteria: * Healthy adult male subjects meeting all the criteria below or adult male subjects having no obvious disease other than high cholesterol levels. * Aged 20 years or over and 65 years or below when the informed consent is obtained. * Weighing 50 kg or over and 80 kg or below on t...

Unlock Eligibility Criteria