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ertapenem

Phase 3

Infection | Small molecule | Infectious Disease |Merck & Company, Inc.|Last Updated: Aug 27, 2018

Target and mechanism

ModalitySmall molecule

Also known as ertapenem sodium (MK0826), ertapenem sodium, Ertapenem sodium

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials1
Total Enrollment599

FDA Designations

No designations recorded

Clinical trial landscape

ertapenem · 4 trials · 4 indications

Phase 3 4
NCT01370616Ertapenem Sodium (MK-0826) Versus Piperacillin/Tazobactam Sodium for the Treatment of Diabetic Foot Infections in Chinese Adults (MK-0826-061)Infection; Diabetic Foot
COMPLETED565 Analytics
NCT01254344Efficacy and Safety of Ertapenem Sodium (MK-0826) Following Colorectal Surgery in Chinese Adults (MK-0826-056)Infection
COMPLETED599 Analytics
NCT01014013Safety and Tolerability of Ertapenem Sodium in the Treatment of Complicated Urinary Tract Infections (0826-055)Urinary Tract Infection
COMPLETED271 Analytics
NCT00379951A Study to Assess the Safety, Tolerability and Efficacy of Ertapenem Sodium in the Treatment of Complicated Urinary Tract Infections (0826-048)Urinary Tract Infection
COMPLETED107 Analytics
PHASE3COMPLETED
Ertapenem Sodium (MK-0826) Versus Piperacillin/Tazobactam Sodium for the Treatment of Diabetic Foot Infections in Chinese Adults (MK-0826-061)
Infection; Diabetic FootUnlock trial analytics
PHASE3COMPLETED
Efficacy and Safety of Ertapenem Sodium (MK-0826) Following Colorectal Surgery in Chinese Adults (MK-0826-056)
InfectionUnlock trial analytics
PHASE3COMPLETED
Safety and Tolerability of Ertapenem Sodium in the Treatment of Complicated Urinary Tract Infections (0826-055)
Urinary Tract InfectionUnlock trial analytics
PHASE3COMPLETED
A Study to Assess the Safety, Tolerability and Efficacy of Ertapenem Sodium in the Treatment of Complicated Urinary Tract Infections (0826-048)
Urinary Tract InfectionUnlock trial analytics

Study Endpoints

Primary Endpoints

Percentage of Participants With Favorable Clinical Response Assessments at Discontinuation of Intravenous (IV) Study Therapy (DCIV)
Day 5 up to Day 28

The investigator assessed participants for a favorable clinical response, defined as clinical improvement or cure. Clinical improvement means that most pretherapy signs and symptoms of the index infection, in particular fever, lympangitis, and purulent drainage had resolved, and no further IV antibiotic therapy was required. Cure means that all pretherapy signs and symptoms of the index infection had resolved, and no further IV antibiotic therapy was required.

Percentage of Participants With Success of Prophylaxis
From study drug dose (day of surgery) up to 4 weeks post therapy

Percentage of participants who have no signs or symptoms of infection at the surgical site, do not require surgical intervention for infection, and have no need for further antimicrobial therapy

Microbiological Response Assessment Profile
5 to 9 days post-therapy

The difference in favorable microbiological response rates between the 2 treatment groups (MK0826 response rate minus ceftriaxone response rate) was assessed

The Number of Patients Who Experience Any Drug-related Adverse Experiences Leading to Discontinuation of Parenteral Study Drug and the Number of Patients With Any Drug-related Serious Adverse Experiences (AEs) During Parenteral Treatment
Adverse experiences that occurred during the study parenteral therapy period were analyzed. The period of parenteral therapy is from 3 days up to 14 days

Safety was assessed by statistical and/or clinical review of all safety parameters, including adverse experiences, physical examination, vital signs, and laboratory results during parenteral therapy. As per the primary safety hypothesis, it was expected that, at the end of the parenteral therapy only, MK0826 would be similar to ceftriaxone with respect to the proportion of patients with any drug-related clinical or laboratory adverse experiences leading to discontinuation of study drug and also with respect to the proportion of patients with any serious drug-related adverse experiences.

Safety and tolerability
14 Days

Secondary Endpoints

Percentage of Participants With Favorable Clinical Response Assessments at Day 5 of IV Study Therapy
Day 5
Percentage of Participants With Favorable Clinical Response Assessments at Follow-up Assessment (FUA) Day 10 of Post-antibiotic Study Therapy
Day 15 up to Day 38
Percentage of Participants With Favorable Microbiological Response Assessments at FUA Day 10 of Post-antibiotic Study Therapy
Day 15 up to Day 38
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Ertapenem sodiumEXPERIMENTALParticipants received 1.0 g intravenous (IV) ertapenem sodium as a single daily dose at Hour 0 infused over a 30-minute interval , and IV piperacillin/tazobactam-matching placebo at Hours 8 and 16 infused over a 30-minute interval, for 5 to 28 days. Participants may be switched to Amoxicillin/clavulunate potassium 625 mg administered orally, twice daily, from Day 6 to Day 28
Piperacillin/tazobactam sodiumACTIVE_COMPARATORParticipants received 4.5 g IV piperacillin/tazobactam at Hours 0, 8, and 16 infused over a 30-minute interval, for 5 to 28 days. Participants may be switched to Amoxicillin/clavulunate potassium 625 mg administered orally, twice daily, from Day 6 to Day 28
Ertapenem sodium 1 gEXPERIMENTALErtapenem sodium 1 g administered intravenously (IV) as a single dose followed by matching placebo to metronidazole administered IV as a single dose
Ceftriaxone sodium 2 gACTIVE_COMPARATORCeftriaxone sodium 2 g administered intravenously (IV) as a single dose followed by metronidazole 500 mg administered IV as a single dose
ertapenem sodium (MK0826)EXPERIMENTALertapenem sodium
ceftriaxone sodiumACTIVE_COMPARATORceftriaxone sodium
1EXPERIMENTALArm 1: ertapenem sodium

Interventions

NameTypeDescription
Ertapenem sodiumDRUGErtapenem sodium, 1.0 g IV daily over 30 minutes at Hour 0 for 5 to 28 days
Piperacillin/tazobactam sodiumDRUGPiperacillin/tazobactam sodium, 4.5 g, IV every 8 hours, given over 30 minutes at Hours 0, 8, and 16 for 5 to 28 days
Piperacillin/tazobactam-matching placeboDRUGPlacebo, IV over 30 minutes, 2 times per day at Hours 8 and 16 for 5 to 28 days
Amoxicillin/clavulunate potassiumDRUGIf clinically indicated, participants may be switched to Amoxicillin/clavulunate potassium 625 mg administered orally, twice daily, from Day 6 to Day 28
ceftriaxone sodiumDRUGCeftriaxone sodium 2 g administered IV as a single dose over 30 minutes within 2 hours prior to the initial surgical incision
placebo to metronidazoleDRUGPlacebo (0.9% sodium chloride) administered IV as a single dose over 30 minutes within 2 hours prior to the initial surgical incision
metronidazoleDRUGMetronidazole 500 mg administered IV as a single dose over 30 minutes within 2 hours prior to the initial surgical incision
ertapenem sodium (MK0826)DRUGa single daily dose of ertapenem sodium 1.0g IV infused over 30 minutes, for 7-14 days (patients may be switched to oral ciprofloxacin after 3 doses of IV therapy if needed)
Comparator: ceftriaxone sodiumDRUGa single daily dose of ceftriaxone 2.0g IV infused over 30 minutes, for 7-14 days (patients may be switched to oral ciprofloxacin after 3 doses of IV therapy)
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Eligibility Criteria

Age Range18 Years to 80 Years
SexALL
Healthy VolunteersNo

Inclusion Criteria: Participant is Chinese with: * Type I diabetes mellitus (IDDM) or Type II diabetes mellitus (NIDDM) treated with diet and/or medication * Clinically- or bacteriologically-documented moderate-to-severe (non life-threatening) diabetic foot infection that requires treatment with I...

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