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TMC278

Phase 1

HIV Infections | Small molecule | Infectious Disease |Merck & Company, Inc.|Last Updated: Jun 27, 2011

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLED
Total Trials1
Total Enrollment24
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01288755TMC278-TiDP6-C153 - A Study in Healthy Volunteers Investigating the Pharmacokinetic Interaction Between TMC278 and RaltegravirPHASE1 COMPLETED 24Feb 1, 2011May 1, 2011Jun 27, 2011 -
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Study Endpoints
Primary Endpoints
Change in exposure to TMC278 following co-administration with raltegravir and vice versa
Measured on Days 5, 12, 13, 14, 15, and 16 (TrtC). Reference for exposure to raltegravir only (TrtB), measured on Days 1, 2, 3, and 4. Reference for exposure to TMC278 only (TrtA), measured on Days 1, 8, 9, 10, 11, and 12.
Secondary Endpoints
Number of participants with adverse events as a measure of safety and tolerability - TMC278 and raltegravir.
97 to 99 days (until and including last safety follow-up visit)
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
001EXPERIMENTALTMC278 One 25 mg tablet once daily for 11 days (TrtA and C)
002EXPERIMENTALRaltegravir One 400 mg tablet twice daily for 4 days (Trt B) and for 11 days (TrtC)
Interventions
NameTypeDescription
TMC278DRUGOne 25 mg tablet, once daily, for 11 days (TrtA and C)
RaltegravirDRUGOne 400 mg tablet, twice daily, for 4 days (Trt B) and for 11 days (TrtC)
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes

Inclusion Criteria: * Healthy, based on physical examination, medical history, vital signs, ECG, blood biochemistry, hematology and urinalysis * Body Mass Index of 18 to 30.0 kg/m2 * Non-smoking for at least 3 months prior to screening * Women must be postmenopausal for at least 2 years, or be surg...

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