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MK0518

Phase 1

HIV-1 Infection | Small molecule | Infectious Disease |Merck & Company, Inc.|Last Updated: Mar 21, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment18
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01000818A Study to Evaluate the Effect of Famotidine and Omeprazole on MK0518 (Raltegravir) Pharmacokinetics in Human Immunodeficiency Virus (HIV)-Infected Patients (0518-054)PHASE1 COMPLETED 18Jun 1, 2008Mar 1, 2009Mar 21, 2017 -
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Study Endpoints
Primary Endpoints
Plasma Area Under Curve (AUC 0-12 hr ) for Raltegravir
12 hours postdose

Area Under the Plasma Concentration-Time Curve and peak concentration

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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Period 1EXPERIMENTALMK0518
Period 2EXPERIMENTALfamotidine + MK0518
Period 3EXPERIMENTALomeprazole + MK0518
Interventions
NameTypeDescription
MK0518 (Raltegravir)DRUG400 mg oral tablet of MK0518 once every 12 hours. Period 1 duration is one day, Period 2 duration is one day, Period 3 duration is five days.
famotidineDRUGSingle 20 mg famotidine oral tablet taken 2 hours prior to administration of AM dose of MK0518
omeprazoleDRUG20 mg oral tablet of omeprazole, once daily for 5 days
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo

Inclusion Criteria: * Patient is Human immunodeficiency virus (HIV) positive * Patient is taking an MK0518 (Raltegravir) containing regimen * Patient has not had any changes to his/her antiviral regimen in the last 2 weeks * Patient who is of reproductive potential agrees to use an acceptable metho...

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