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VH4011499 Dose A

Phase 1

HIV Infections | Small molecule | Infectious Disease |GSK plc|Last Updated: Feb 18, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment60
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT06368986A Study to Investigate the Effect of Food on the Bioavailability of a Capsid Inhibitor (CAI) in Male and Female Healthy ParticipantsPHASE1 COMPLETED 60Apr 17, 2024Oct 2, 2024Feb 18, 20251 United States
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Study Endpoints
Primary Endpoints
Area under the plasma concentration - time curve from time zero (pre-dose) to infinity time (AUC[0-inf]) of VH4011499
From Day 1 (pre-dose) to Day 28
Area under the plasma drug concentration - time curve from zero (pre-dose) to the end of the dosing interval at steady state (AUC[0-tlast) of VH4011499
From Day 1 (pre-dose) to Day 28
Maximum observed plasma drug concentration (Cmax) of VH4011499
From Day 1 (pre-dose) to Day 28
Time to maximum observed plasma concentration (Tmax) of VH4011499
From Day 1 (pre-dose) to Day 28
Secondary Endpoints
Number of participants with AEs (Adverse Events), by severity
From Day 1 (pre-dose) to Day 28
Number of participants with maximum toxicity grade increase from baseline for liver laboratory parameters
From Day 1 (pre-dose) to Day 28
Change from baseline in liver panel parameters: total bilirubin and direct bilirubin (micromoles per liter)
From Day 1 (pre-dose) to Day 28
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeOTHER
Treatment Arms
ArmTypeDescription
Part 1 Dose A - Fasted conditionEXPERIMENTALVH4011499 Dose A tablet administered in fasted condition.
Part 1 Dose A- Fed condition (high fat meal)EXPERIMENTALVH4011499 Dose A tablet administered in fed condition (high fat meal).
Part 2 Dose B - Optional - Fed condition (low fat meal)EXPERIMENTALVH4011499 Dose B tablet administered in fed condition (low fat meal).
Part 3 Dose B - Fasted conditionEXPERIMENTALVH4011499 Dose B tablet administered in fasted condition.
Part 3 Dose B - Fed condition (high fat meal)EXPERIMENTALVH4011499 Dose B tablet administered in fed condition (high fat meal).
Interventions
NameTypeDescription
VH4011499 Dose ADRUGVH4011499 administered in fasted or fed conditions.
VH4011499 Dose BDRUGVH4011499 Dose B administered in fasted or fed conditions.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Participants who are 18 to 55 years of age. * Participants who are overtly healthy. * One SARs-CoV-2 negative test is required prior to dosing * Body weight within 50-100 kg and body mass index (BMI) within the range 19-32 kg/m2 (inclusive). * Capable of giving signed informed...

Countries:United States
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