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VH4004280 Formulation A

Phase 1

HIV Infections | Small molecule | Infectious Disease |GSK plc|Last Updated: Aug 2, 2024

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment46
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT06168318A Study to Investigate the Relative Bioavailability and Food Effect of an Oral Capsid Inhibitor Tablet Formulation Compared With Other Oral Tablet Formulations in Male and Female Healthy ParticipantsPHASE1 COMPLETED 46Dec 18, 2023Jun 3, 2024Aug 2, 20241 United Kingdom
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Study Endpoints
Primary Endpoints
Area under the plasma concentration - time curve from time zero (pre-dose) to infinity time (AUC[0-inf]) of VH4004280 in fed conditions (after a high-fat or lower-fat meal)
From Day 1 to Day 49
Area under the plasma drug concentration - time curve from zero (pre-dose) to the end of the dosing interval at steady state (AUC[0-tlast) of VH4004280 in fed conditions (after a high-fat or lower-fat meal)
From Day 1 to Day 49
Maximum observed plasma drug concentration (Cmax) of VH4004280 in fed conditions(after a high-fat or lower-fat meal)
From Day 1 to Day 49
Time to maximum observed plasma concentration (Tmax) of VH4004280 in fed conditions (after a high-fat or lower-fat meal)
From Day 1 to Day 49
Secondary Endpoints
Number of participants with AEs (Adverse Events), by severity
From Day 1 to Day 49
Number of participants with maximum toxicity grade increase from baseline for liver laboratory parameters
From Day 1 to Day 49
Change from baseline in liver panel parameters: Total bilirubin and direct bilirubin (micromoles per liter)
From Day 1 to Day 49
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part 1 - Regimen AEXPERIMENTALVH4004280 Formulation A tablet administered in fed conditions.
Part 1 - Regimen BEXPERIMENTALVH4004280 Formulation B tablet administered in fed conditions.
Part 1 - Regimen CEXPERIMENTALVH4004280 Formulation C tablet administered in fed conditions.
Part 1 - Optional Regimen DEXPERIMENTALVH4004280 Formulation D tablet administered in fed conditions.
Part 1 - Optional Regimen EEXPERIMENTALVH4004280 Formulation E tablet administered in fed conditions.
Part 2 - Regimen AEXPERIMENTALVH4004280 Formulation A tablet administered in fasted conditions.
Part 2- Optional Regimen 1EXPERIMENTALVH4004280 Formulation B, C, D, or E tablet administered in fasted conditions.
Part 2- Optional Regimen 2EXPERIMENTALVH4004280 Formulation B, C, D, or E tablet administered in fasted conditions.
Part 2- Optional Regimen 3EXPERIMENTALVH4004280 Formulation B, C, D, or E tablet administered in fasted conditions.
Part 3 - Optional Regimen 1EXPERIMENTALVH4004280 Formulation A, B, C or D tablet administered in lower fat conditions.
Part 3- Optional Regimen 2EXPERIMENTALVH4004280 Formulation A, B, C or D tablet administered in lower fat conditions.
Part 3 - Optional Regimen 3EXPERIMENTALVH4004280 Formulation A, B, C or D tablet administered in lower fat conditions.
Part 3 - Optional Regimen 4EXPERIMENTALVH4004280 Formulation A, B, C or D tablet administered in lower fat conditions.
Interventions
NameTypeDescription
VH4004280 Formulation ADRUGOral administration of VH4004280 Formulation A in fasted or fed conditions.
VH4004280 Formulation BDRUGOral administration of VH4004280 Formulation B in fasted or fed conditions.
VH4004280 Formulation CDRUGOral administration of VH4004280 Formulation C in fasted or fed conditions.
VH4004280 Formulation DDRUGOral administration of VH4004280 Formulation D in fasted or fed conditions.
VH4004280 Formulation EDRUGOral administration of VH4004280 Formulation E in fasted or fed conditions.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Participants must be 18 to 55years of age. 2. Participants who are overtly healthy. 3. Negative (Severe Acute Respiratory Syndrome Coronavirus 2) SARs-CoV-2 test prior to dosing. 4. Has body mass index (BMI) within the range 19-32 (kg/m2). 5. Participants male at birth must u...

Countries:United Kingdom
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