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Paroxetine 12.5 milligrams

Phase 1

Depressive Disorder | Small molecule | Psychiatry |GSK plc|Last Updated: Jun 19, 2018

Target and mechanism

ModalitySmall molecule

Also known as Paroxetine 12.5 milligrams tablet

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment18

FDA Designations

No designations recorded

Clinical trial landscape

Paroxetine 12.5 milligrams · 1 trial · 1 indication

Phase 1 1
NCT00938184Single Dose Study of Controlled-Release Paroxetine Tablets in Healthy Japanese Male SubjectsDepressive Disorder
COMPLETED18 Analytics
PHASE1COMPLETED
Single Dose Study of Controlled-Release Paroxetine Tablets in Healthy Japanese Male Subjects
Depressive DisorderUnlock trial analytics

Study Endpoints

Primary Endpoints

Pharmacokinetic parameters of plasma paroxetine after single doses of paroxetine CR at 12.5mg, 25mg and 50mg in healthy Japanese male volunteers
up to 120 hours after a single dose in all dosing sessions

Secondary Endpoints

Safety and tolerability after single doses of paroxetine CR at 12.5mg, 25mg and 50mg in healthy Japanese male volunteers
up to 120 hours after a single dose in all dosing sessions
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Treatment sequence A/B/CEXPERIMENTALEligible subjects will be randomized in sequence A/B/C and will receive A: single tablet of paroxetine 12.5 milligrams, B: single tablet of paroxetine 25 milligrams and C: two tablets of paroxetine 25 milligrams administered orally in the morning. Subjects will be fasting since 10 hours before dosing in each period.
Treatment sequence A/C/BEXPERIMENTALEligible subjects will be randomized in sequence A/C/B and will receive A: single tablet of paroxetine 12.5 milligrams, C: two tablets of paroxetine 25 milligrams and B: single tablet of paroxetine 25 milligrams administered orally in the morning. Subjects will be fasting since 10 hours before dosing in each period.
Treatment sequence B/A/CEXPERIMENTALEligible subjects will be randomized in sequence B/A/C and will receive B: single tablet of paroxetine 25 milligrams, A: single tablet of paroxetine 12.5 milligrams and C: two tablets of paroxetine 25 milligrams administered orally in the morning. Subjects will be fasting since 10 hours before dosing in each period.
Treatment sequence B/C/AEXPERIMENTALEligible subjects will be randomized in sequence B/C/A and will receive B: single tablet of paroxetine 25 milligrams, C: two tablets of paroxetine 25 milligrams and A: single tablet of paroxetine 12.5 milligrams administered orally in the morning. Subjects will be fasting since 10 hours before dosing in each period.
Treatment sequence C/A/BEXPERIMENTALEligible subjects will be randomized in sequence C/A/B and will receive C: two tablets of paroxetine 25 milligrams, A: single tablet of paroxetine 12.5 milligrams and B: single tablet of paroxetine 25 milligrams administered orally in the morning. Subjects will be fasting since 10 hours before dosing in each period.
Treatment sequence C/B/AEXPERIMENTALEligible subjects will be randomized in sequence C/B/A and will receive C: two tablets of paroxetine 25 milligrams, B: single tablet of paroxetine 25 milligrams and A: single tablet of paroxetine 12.5 milligrams administered orally in the morning. Subjects will be fasting since 10 hours before dosing in each period.

Interventions

NameTypeDescription
Paroxetine 12.5 milligrams tabletDRUGSingle dose of paroxetine 12.5 milligrams controlled release tablet will be administered orally.
Paroxetine 25 milligrams tabletDRUGSingle dose of paroxetine 25 milligrams controlled release tablet will be administered orally.
Paroxetine 50 milligrams tabletDRUGSingle dose of paroxetine 50 milligrams controlled release tablet (as two tablets of 25 milligrams) will be administered orally.
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Eligibility Criteria

Age Range20 Years to 64 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy Japanese adult males between 20 and 64 years of age inclusive * BMI 18.50 or higher and \< 25.00 kg/m2, and bodyweight 50 kg or higher * Non-smokers * AST, ALT, ALP, gamma-GTP and total-bilirubin are below the upper limit of normal range * QTc(B) interval \<450 msec * ...

Countries:Japan
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