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GSK2647544

Phase 1

Alzheimer's Disease | Small molecule | Neurology |GSK plc|Last Updated: Oct 18, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedPLACEBO_CONTROLLED
Total Trials1
Total Enrollment27

FDA Designations

No designations recorded

Clinical trial landscape

GSK2647544 · 1 trial · 1 indication

Phase 1 1
NCT01702467Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Single, Oral Escalating Doses of GSK2647544 in Healthy VolunteersAlzheimer's Disease
COMPLETED27 Analytics
PHASE1COMPLETED
Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Single, Oral Escalating Doses of GSK2647544 in Healthy Volunteers
Alzheimer's DiseaseUnlock trial analytics

Study Endpoints

Primary Endpoints

Safety and tolerability of GSK2647544 as assessed by number of subjects with adverse events (AE)s
5 days in each of the 4 dosing session

Safety and tolerability parameters will include recording of AEs

Safety and tolerability of GSK2647544 as assessed by change from Baseline in laboratory values
5 days in each of the 4 dosing session

Safety and tolerability parameters will include laboratory (haematology, clinical chemistry, urinalysis) values at Screening, Day -1, Day 3 and Follow-up (7-14 days post-last dose)

Safety and tolerability of GSK2647544 as assessed by change from Baseline in ECG readings
5 days in each of the 4 dosing session

Safety and tolerability parameter will include the electrocardiogram (ECG) readings at Screening, Day -1, Day 1, Day 2, Day 3 and Follow-up (7-14 days post-last dose)

Safety and tolerability of GSK2647544 as assessed by change from Baseline in Telemetry ECG parameters
3 Days in each of the 4 dosing session

Safety and tolerability parameter will include the Telemetry ECG readings from 30 minutes pre-dosing till 48 hours post-dosing

Safety and tolerability of GSK2647544 as assessed by change from Baseline in vital signs
5 days in each of the 4 dosing session

Vital signs measurement include systolic and diastolic blood pressure and pulse rate at Screening, Day -1, Day 1, Day 2, Day 3, Day 4 and Follow-up (7-14 days post-last dose)

Safety and tolerability of GSK2647544 as assessed by using the Columbia Suicide Severity Rating Scale (C-SSRS)
5 days in each of the 4 dosing session

C-SSRS will be measured at Screening, Day -1, Day 1 (conducted prior to discharge) and Follow-up (7-14 days post-last dose)

Secondary Endpoints

Peak plasma concentration (Cmax) of GSK2647544
4 Days in each of the 4 dosing session
Time of peak plasma concentration (tmax) of GSK2647544
4 Days in each of the 4 dosing session
Area under the time concentration curve (AUC) of GSK2647544
4 Days in each of the 4 dosing session
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Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
GSK2647544EXPERIMENTALThe starting dose of GSK2647544 is 0.5 mg. The escalating doses to be administered will be determined based on study results from previous dose (s).
PlaceboPLACEBO_COMPARATORMatching placebo

Interventions

NameTypeDescription
GSK2647544DRUGCapsules containing 0.5mg to 50mg of GSK2647544.
PlaceboDRUGMatching placebo capsules.
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Eligibility Criteria

Age Range18 Years to 55 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy males who are 18 to 55 years of age, inclusive * Healthy as determined by a responsible and experienced physician * aspartate aminotransferase (AST), Alanine transaminase (ALT), alkaline phosphatase and bilirubin \<= 1.5xUpper Limit of Normal (ULN) * Average of triplic...

Countries:Australia
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Frequently asked questions about GSK2647544

What is GSK2647544 used for?

GSK2647544 is an investigational small molecule being developed for Alzheimer's Disease. It is currently in Phase 1 clinical development, meaning it has not yet been approved and is still being studied for safety and tolerability in humans.

Who makes GSK2647544?

GSK2647544 is being developed by GSK plc, a global biopharma company listed on the stock exchange under the ticker GSK. The company is conducting clinical trials to evaluate the drug's safety and pharmacokinetics in healthy volunteers.

What phase is GSK2647544 in?

GSK2647544 is in Phase 1 clinical development. One Phase 1 trial has been completed, involving 27 participants. The drug is investigational and has not received regulatory approval for any use.

What clinical trials is GSK2647544 in?

GSK2647544 has one completed clinical trial, NCT01702467, titled 'Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of Single, Oral Escalating Doses of GSK2647544 in Healthy Volunteers.' This was a Phase 1, placebo-controlled study conducted in Australia with 27 healthy male participants.

Is GSK2647544 FDA approved?

GSK2647544 is not FDA approved. It is an investigational drug currently in Phase 1 clinical development. The completed trial focused on safety, tolerability, and pharmacokinetics in healthy volunteers, and further studies would be needed before any approval could be considered.

Is GSK2647544 the same as any other drug?

No alternative names for GSK2647544 have been reported. The drug is identified solely by its code name GSK2647544 in clinical trial registries and scientific literature.