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GSK1265744

Phase 1

HIV Infection | Small molecule | Infectious Disease |GSK plc|Last Updated: Apr 2, 2012

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials2
Total Enrollment103
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00812318Healthy Volunteer Study To Assess The Bioavailability of GSK1265744 When Administered Orally Either When Fasted or Following a Meal.PHASE1 COMPLETED 45Jun 1, 2008Aug 1, 2008Apr 2, 20121 United States
NCT00659191A Healthy Volunteer And Patient Study To Assess The Safety, Tolerability And Pharmacokinetics Of GSK1265744PHASE1 COMPLETED 58Feb 1, 2008Nov 1, 2008Oct 15, 20105 United States
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Study Endpoints
Primary Endpoints
Composite of pharmacokinetic parameters
6 days

Plasma GSK1265744 Area under the concentration-time curve from time zero (pre-dose) extrapolated to infinite time \[AUC(0-infinity)\], Area under the concentration-time curve over the dosing interval \[AUC(0-t)\], and Maximum observed concentration (Cmax).

Safety evaluations (labs, ECG, blood pressure), and blood sampling for PK, Continuous AE monitoring through study conclusion and follow up, 7-14 days after last dose. For Part C only: anti-viral activity through study conclusion and follow-up.
through study conclusion and follow up, 7-14 days after last dose
Secondary Endpoints
Safety and tolerability parameters, including the collection adverse events
6 days
Composite of pharmacokinetic parameters
6 days
Safety and tolerability parameters including the change from baseline in clinical laboratory assessments
6 days
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Treatment AEXPERIMENTALGSK1265744 10mg oral solution
Treatment BEXPERIMENTALGSK1265744 5mg tablet, fasted
Treatment CEXPERIMENTALGSK1265744 5mg tablet, fed
Interventions
NameTypeDescription
GSK1265744 10 mg oral solutionDRUGGSK1265744
GSK1265744 5 mg tabletDRUGGSK1265744 5mg tablet, fasted
GSK1265744DRUG -
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy as determined by a responsible physician, based on a medical evaluation including medical history, physical examination, laboratory tests and 12-lead ECG. A subject with a clinical abnormality or laboratory parameters outside the reference range for the population bein...

Countries:United States
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