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Dolutegravir dispersible

Phase 1

HIV Infections | Small molecule | Infectious Disease |GSK plc|Last Updated: Jul 31, 2020

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment22

FDA Designations

No designations recorded

Clinical trial landscape

Dolutegravir dispersible · 1 trial · 1 indication

Phase 1 1
NCT03921723Dolutegravir Pediatric Liquid Formulation StudyHIV Infections
COMPLETED22 Analytics
PHASE1COMPLETED
Dolutegravir Pediatric Liquid Formulation Study
HIV InfectionsUnlock trial analytics

Study Endpoints

Primary Endpoints

Area Under the Plasma Concentration Time Curve From Time Zero to the Last Quantifiable Time Point (AUC[0-t]) for DTG
Pre-dose, 0.25, 0.5, 0.75, 1, 1.5, 2, 2.5, 3,3.5, 4, 5, 6, 8, 12, 16, 24, 48, and 72 hours post-dose

Blood samples were collected at indicated time points and pharmacokinetic (PK) analysis was performed. PK parameters were determined by non-compartmental methods.

AUC From Time Zero to Infinity (AUC[0-inf]) for DTG
Pre-dose, 0.25, 0.5, 0.75, 1, 1.5, 2, 2.5, 3,3.5, 4, 5, 6, 8, 12, 16, 24, 48, and 72 hours post-dose

Blood samples were collected at indicated time points and PK analysis was performed. PK parameters were determined by non-compartmental methods.

Maximum Observed Concentration (Cmax) for DTG
Pre-dose, 0.25, 0.5, 0.75, 1, 1.5, 2, 2.5, 3,3.5, 4, 5, 6, 8, 12, 16, 24, 48, and 72 hours post-dose

Blood samples were collected at indicated time points and PK analysis was performed. PK parameters were determined by non-compartmental methods.

Secondary Endpoints

Absorption Lag Time (Tlag) Following Administration of DTG
Pre-dose, 0.25, 0.5, 0.75, 1, 1.5, 2, 2.5, 3,3.5, 4, 5, 6, 8, 12, 16, 24, 48, and 72 hours post-dose
Time of Maximum Observed Concentration (Tmax) Following Administration of DTG
Pre-dose, 0.25, 0.5, 0.75, 1, 1.5, 2, 2.5, 3, 3.5, 4, 5, 6, 8, 12, 16, 24, 48, and 72 hours post-dose
Time of Last Quantifiable Concentration (Tlast) Following Administration of DTG
Pre-dose, 0.25, 0.5, 0.75, 1, 1.5, 2, 2.5, 3, 3.5, 4, 5, 6, 8, 12, 16, 24, 48, and 72 hours post-dose
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Subject receiving Dolutegravir 10 mgEXPERIMENTALSubject will receive a prototype equivalent to DTG 10 mg liquid formulation in period 1, a prototype equivalent to DTG 10 mg liquid formulation in period 2, a DTG 10 mg dispersible tablet in Period 3, each period will be separated by washout period of \>= 7 days, if required a prototype equivalent to DTG 10 mg liquid formulation in period 4, a prototype equivalent to DTG 10 mg liquid formulation in period 5, and a prototype equivalent to DTG 10 mg liquid formulation in period 6 will be evaluated.

Interventions

NameTypeDescription
Dolutegravir dispersible tabletDRUGDTG will be available as an oral tablet with dosing strength of 5 mg 2 tablet will be dispersed in water will be administered orally for prescribed regimen.
Dolutegravir oral suspensionDRUGDTG will be available as an oral suspension with dosing strength of 5 mg per milliliter (ml) or 2 mg per ml with miglyol 812N or ethyl cellulose in miglyol 812N as vehicle for suspension administered orally for prescribed regimen.
Dolutegravir oral solutionDRUGDTG will be available as an oral solution with dosing strength of 2 mg per ml will be administered orally for prescribed regimen.
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Eligibility Criteria

Age Range18 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Subject must be 18 to 55 years of age inclusive, at the time of signing the informed consent. * Subjects who are overtly healthy as determined by medical evaluation including medical history, physical examination, laboratory tests, and cardiac evaluation. * Body weight \>= 50 ...

Countries:United Kingdom
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Frequently asked questions about Dolutegravir dispersible

What is Dolutegravir dispersible used for?

Dolutegravir dispersible is a small molecule being developed for the treatment of HIV Infections. It is an investigational drug currently in Phase 1 clinical development. The dispersible formulation is designed for pediatric use, as indicated by the ongoing clinical trial studying this liquid formulation in the United Kingdom.

Who makes Dolutegravir dispersible?

Dolutegravir dispersible is being developed by GSK plc, which trades under the ticker GSK. The company is conducting clinical research on this investigational small molecule for the treatment of HIV Infections. The drug is currently in Phase 1 development.

What phase is Dolutegravir dispersible in?

Dolutegravir dispersible is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed, involving 22 participants in the United Kingdom.

What clinical trials is Dolutegravir dispersible in?

Dolutegravir dispersible has one completed clinical trial, NCT03921723, titled "Dolutegravir Pediatric Liquid Formulation Study." This Phase 1 study enrolled 22 participants with HIV Infections in the United Kingdom. The trial was uncontrolled, not randomized, and not double-blinded, and it included healthy volunteers.

Is Dolutegravir dispersible the same as Dolutegravir?

Dolutegravir dispersible is a formulation of the drug dolutegravir, specifically designed as a dispersible or liquid formulation for pediatric use. While the active ingredient is the same, the dispersible version is being studied separately in clinical trials for its suitability in treating HIV Infections in younger populations.