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Cabotegravir IR Formulation

Phase 1

HIV Infections | Small molecule | Infectious Disease |GSK plc|Last Updated: Dec 13, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment24
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT05776108A Study to Assess the Food Effect and the Relative Bioavailability of the Cabotegravir (CAB) Pediatric Dispersible Tablet (DT) FormulationPHASE1 COMPLETED 24Mar 23, 2023Jun 8, 2023Dec 13, 20231 United States
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Study Endpoints
Primary Endpoints
Area under the concentration-time curve from time zero (pre-dose) extrapolated to infinite time (AUC[0-inf]) following administration of CAB DT after a high fat meal
Up to 168 hours
Area under the concentration time curve from time zero (pre-dose) extrapolated to last time of quantifiable concentration (AUC[0-last]) following administration of CAB DT after a high fat meal
Up to 168 hours
Maximum observed concentration (Cmax) following administration of CAB DT after a high fat meal
Up to 168 hours
AUC(0-inf) following administration of CAB DT in fasted state
Up to 168 hours
AUC(0-last) following administration of CAB DT in fasted state
Up to 168 hours
Cmax following administration of CAB DT in fasted state
Up to 168 hours
AUC(0-inf) following administration of CAB IR in fasted state
Up to 168 hours
AUC(0-last) following administration of CAB IR in fasted state
Up to 168 hours
Cmax following administration of CAB IR in fasted state
Up to 168 hours
Secondary Endpoints
Apparent terminal phase half-life (T1/2) following administration of CAB DT
Up to 168 hours
Lag time before observation of drug concentrations in sampled matrix (tlag) following administration of CAB DT
Up to 168 hours
Time of occurrence of Cmax (Tmax) following administration of CAB DT
Up to 168 hours
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
CAB IR Formulation (reference)/CAB DT Formulation (Test 1)/CAB DT Formulation (Test 2)EXPERIMENTALParticipants will receive CAB IR Formulation (reference) under fasted conditions in treatment period 1 followed by CAB DT Formulation (test 1) under fasted conditions in treatment period 2 followed by CAB DT Formulation (test 2) under fed conditions in treatment period 3. There will be a minimum washout period of 14 days between each treatment .
CAB DT Formulation (Test 1)/CAB IR Formulation (reference)/CAB DT Formulation (test 2)EXPERIMENTALParticipants will receive CAB DT Formulation (test 1) under fasted conditions in treatment period 1 followed by CAB IR Formulation (reference) under fasted conditions in treatment period 2 followed by CAB DT Formulation (test 2) under fed conditions in treatment period 3. There will be a minimum washout period of 14 days between each treatment.
CAB DT Formulation (test 2)/CAB IR Formulation (reference)/CAB DT Formulation (test 1)EXPERIMENTALParticipants will receive CAB DT Formulation (test 2) under fed conditions in treatment period 1 followed by CAB IR Formulation (reference) under fasted conditions in treatment period 2 followed by CAB DT Formulation (test 1) under fasted conditions in treatment period 3. There will be a minimum washout period of 14 days between each treatment.
CAB IR Formulation (reference)/CAB DT Formulation (test 2)/CAB DT Formulation (test 1)EXPERIMENTALParticipants will receive CAB IR Formulation (reference) under fasted conditions in treatment period 1 followed by CAB DT Formulation (test 2) under fed conditions in treatment period 2 followed by CAB DT Formulation (test 1) under fasted conditions in treatment period 3. There will be a minimum washout period of 14 days between each treatment.
CAB DT Formulation (test 1)/CAB DT Formulation (test 2)/CAB IR Formulation (reference)EXPERIMENTALParticipants will receive CAB DT Formulation (test 1) under fasted conditions in treatment period 1 followed by CAB DT Formulation (test 2) under fed conditions in treatment period 2 followed by CAB IR Formulation (reference) under fasted conditions in treatment period 3. There will be a minimum washout period of 14 days between each treatment.
CAB DT Formulation (test 2)/CAB DT Formulation (test 1)/CAB IR Formulation (reference)EXPERIMENTALParticipants will receive CAB DT Formulation (test 2) under fed conditions in treatment period 1 followed by CAB DT Formulation (test 1) under fasted conditions in treatment period 2 followed by CAB IR Formulation (reference) under fasted conditions in treatment period 3. There will be a minimum washout period of 14 days between each treatment.
Interventions
NameTypeDescription
Cabotegravir IR Formulation (reference)DRUGCabotegravir IR Formulation (reference) will be administered.
Cabotegravir DT Formulation (test 1)DRUGCabotegravir DT Formulation (test 1) will be administered.
Cabotegravir DT Formulation (test 2)DRUGCabotegravir DT Formulation (test 2) will be administered.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion criteria: * Participant must be 18 to 55 years of age inclusive, at the time of signing the informed consent form (ICF). * Participants who are healthy as determined by the investigator or medically qualified designee based on a medical evaluation including medical history, physical exami...

Countries:United States
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