Recent Updates
Recently added Catalysts

GS-5745

Phase 1

Rheumatoid Arthritis | Small molecule | Immunology |Gilead Sciences, Inc.|Last Updated: Jun 29, 2015

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment18

FDA Designations

No designations recorded

Clinical trial landscape

GS-5745 · 2 trials · 2 indications

Phase 1 2
NCT02176876Safety, Tolerability, and Pharmacokinetics of GS-5745 in Subjects With Rheumatoid ArthritisRheumatoid Arthritis
COMPLETED18 Analytics
NCT02209987Absolute Bioavailability, Safety, and Tolerability of Subcutaneous GS-5745 in Healthy AdultsUlcerative Colitis
COMPLETED28 Analytics
PHASE1COMPLETED
Safety, Tolerability, and Pharmacokinetics of GS-5745 in Subjects With Rheumatoid Arthritis
Rheumatoid ArthritisUnlock trial analytics
PHASE1COMPLETED
Absolute Bioavailability, Safety, and Tolerability of Subcutaneous GS-5745 in Healthy Adults
Ulcerative ColitisUnlock trial analytics

Study Endpoints

Primary Endpoints

Incidence of adverse events, changes in laboratory tests and vital signs from baseline, and development of immunogenicity after dosing
Up to 100 days

This composite endpoint will measure the safety and tolerability profile of GS-5745.

PK profile of GS-5745
Predose and postdose on Days 1 and Day 11, and Weeks 2, 3, 4, 6, and 8

This composite endpoint will measure the plasma PK profile of GS-5745. The following parameters will be measured, where applicable: * Cmax: maximum observed concentration of drug in plasma * AUClast: concentration of drug from time zero to the last quantifiable concentration * AUC0-inf: area under the plasma concentration versus time curve starting with time zero to infinity

Secondary Endpoints

PK profile of GS-5745
Pre-infusion, 30 minutes, 4 hours, and 24 hours post-infusion on Day 1; pre-infusion and 30 minutes post-infusion on Days 15 and 29; Days 4, 8, 36, and 43
Incidences of adverse events and laboratory abnormalities
Up to 8 weeks
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
GS-5745EXPERIMENTALParticipants will receive GS-5745 every 2 weeks for a total of 3 infusions.
Placebo to match GS-5745PLACEBO_COMPARATORParticipants will receive placebo to match GS-5745 every 2 weeks for a total of 3 infusions.
GS-5745 SCEXPERIMENTALParticipants will receive a single dose of GS-5745 by SC injection.
GS-5745 IVEXPERIMENTALParticipants will receive a single dose of GS-5745 by IV infusion.

Interventions

NameTypeDescription
GS-5745DRUGGS-5745 400 mg administered intravenously
Placebo to match GS-5745DRUGPlacebo to match GS-5745 administered intravenously
GS-5745 SCDRUGGS-5745 150 mg administered by SC injection formulated as a sterile, aqueous buffered solution in a single-use pre-filled syringe
GS-5745 IVDRUGGS-5745 150 mg administered by IV infusion formulated as a sterile, aqueous buffered solution in single-use glass vials
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 70 Years
SexALL
Healthy VolunteersNo
Study Sites4

Inclusion Criteria: * 18 to 70 years of age, inclusive, at time of screening * Weight: ≥ 45 to \< 120 kg * Males or non-pregnant, non-lactating females * Diagnosis of RA according to the 1987 revised American College of Rheumatology (ACR) for the classification of RA * Active disease, defined as a ...

Countries:CzechiaHungaryNew Zealand
Unlock Eligibility Criteria

Frequently asked questions about GS-5745

What is GS-5745 used for?

GS-5745 is an investigational small molecule being developed for ulcerative colitis and rheumatoid arthritis. It is in Phase 1 clinical development and is not yet approved by the FDA. The drug is being studied for its safety, tolerability, and pharmacokinetics in these conditions.

Who makes GS-5745?

GS-5745 is developed by Gilead Sciences, Inc., a biopharmaceutical company traded on NASDAQ under the ticker GILD. The drug is currently in Phase 1 clinical trials for ulcerative colitis and rheumatoid arthritis.

What phase is GS-5745 in?

GS-5745 is in Phase 1 clinical development. It is an investigational drug and has not received FDA approval. Clinical trials have been completed for rheumatoid arthritis and healthy adults, with the drug being studied for ulcerative colitis.

What clinical trials is GS-5745 in?

GS-5745 has completed two Phase 1 trials. NCT02176876 studied the drug in 18 subjects with rheumatoid arthritis in Czechia and Hungary. NCT02209987 assessed subcutaneous GS-5745 in 28 healthy adults in New Zealand, with conditions listed as ulcerative colitis.

Is GS-5745 the same as any other drug?

GS-5745 is the primary name for this investigational small molecule developed by Gilead Sciences. No alternative names have been reported for this drug in clinical development for ulcerative colitis and rheumatoid arthritis.