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BMS-686117

Phase 1

Type 2 Diabetes | Small molecule | Metabolic |Bristol-Myers Squibb Company|Last Updated: Mar 16, 2009

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment36
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00508287Study to Evaluate the Safety, Pharmacokinetics, and Pharmacodynamics of BMS-686117 in Subjects With Type 2 DiabetesPHASE1 COMPLETED 36Aug 1, 2007Nov 1, 2007Mar 16, 20093 United States
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Study Endpoints
Primary Endpoints
Safety: incidence of adverse events
from subject enrollment to study discharge
Secondary Endpoints
PK parameters: Cmax, Tmax, AUC(0-24h), AUC(INF) and T-HALF
from pre-dose to 24 hrs post-dose
PD Measures: Fasting and postprandial serum glucose (AUC), serum insulin, and plasma glucagon concentrations. Acetaminophen plasma concentrations will be measured after a single dose of acetaminophen
from pre-dose to 9 hrs post-dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
AEXPERIMENTAL -
BACTIVE_COMPARATOR -
CPLACEBO_COMPARATOR -
Interventions
NameTypeDescription
BMS-686117DRUGInjection solution, Subcutaneous, 1 mg, Once daily, Single dose.
ByettaDRUGInjection solution, Subcutaneous, 5 mcg, Once daily, Single dose.
PlaceboDRUGInjection solution, Subcutaneous, 1 mg, Once daily, Single dose.
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersNo
Study Sites3

Inclusion Criteria: * Diagnosis of Type 2 diabetes for ≥ 3 months treated with metformin, thiazolidinedione, or sulfonylurea (either monotherapy or combination) or diet alone (drug naïve) * Fasting plasma glucose: 126 - 240 mg/dL * Hemoglobin A1c: 6 - 10% * Estimated CrCl ≥ 60 mL/min * ALT ≤ 1.5 x ...

Countries:United States
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