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icovamenib

Phase 2

Type 2 Diabetes | Small molecule | Metabolic |Biomea Fusion, Inc.|Last Updated: Aug 28, 2026

Target and mechanism

Target class-Nib (Kinase)
ModalitySmall molecule

Also known as icovamenib 100mg

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLEDDMC
Total Trials2
Total Enrollment124

FDA Designations

No designations recorded

Clinical trial landscape

icovamenib · 3 trials · 2 indications

Phase 2 2Phase 1 1
NCT07502508Phase 2 Trial of Icovamenib in Participants With Type 2 Diabetes Mellitus Who Are Not Achieving Glycemic Targets While Using GLP-1-Based TherapyType 2 Diabetes
RECRUITING60 Analytics
NCT07502495Phase 2 Trial of Icovamenib in Participants With Type 2 Diabetes Who Are Not Achieving Glycemic TargetsType 2 Diabetes
ACTIVE NOT_RECRUITING64 Analytics
PHASE2RECRUITING
Phase 2 Trial of Icovamenib in Participants With Type 2 Diabetes Mellitus Who Are Not Achieving Glycemic Targets While Using GLP-1-Based Therapy
Type 2 DiabetesUnlock trial analytics
PHASE2ACTIVE NOT_RECRUITING
Phase 2 Trial of Icovamenib in Participants With Type 2 Diabetes Who Are Not Achieving Glycemic Targets
Type 2 DiabetesUnlock trial analytics

Study Endpoints

Primary Endpoints

To demonstrate that icovamenib 100 mg once daily for 12 weeks is superior to placebo for glycemic control
26 weeks

Mean change in HbA1c from baseline

Evaluate food effect and PK profile of icovamenib capsule formulation in fed and fasted states
Every other day for a max of 2 weeks

Tmax

Secondary Endpoints

To demonstrate that icovamenib 100 mg once daily for 12 weeks is superior to placebo for glycemic control
12 weeks
To compare the change in fasting plasma glucose with icovamenib versus placebo during the off-treatment Follow-up Period
26 weeks
To compare the safety and tolerability of icovamenib versus placebo
52 weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Arm A: icovamenib 100 mgEXPERIMENTALStarting on Day 1, participants will receive icovamenib 100 mg QD in addition to their currently prescribed Ozempic (semaglutide injection)-based regimen. Treatment will last for 12 weeks. At Week 12, participants will continue on a stable dose of their baseline Ozempic-based regimen. The total duration of the trial is approximately 56 weeks (including screening and follow-up)
Arm B: matching placebo 100 mgPLACEBO_COMPARATORStarting on Day 1, participants will receive matching placebo QD in addition to their currently prescribed Ozempic (semaglutide injection)-based regimen. Treatment will last for 12 weeks. At Week 12, participants will continue on a stable dose of their baseline Ozempic-based regimen. The total duration of the trial is approximately 56 weeks (including screening and follow-up).
Arm B: placebo matching 100 mgPLACEBO_COMPARATORplacebo matching 100mg QD in addition to their currently prescribed antihyperglycemic medication(s) for 12 weeks. At Week 12, participants will continue on their currently prescribed antihyperglycemic medication(s). The total duration of the trial is approximately 56 weeks
Regimen AEXPERIMENTALA - icovamenib capsule 100mg in fasted state
Regimen BEXPERIMENTALB - icovamenib capsule 100mg in the fed state (0.5 h after initiation of low-fat breakfast)
Regimen CEXPERIMENTALC - icovamenib capsule 100mg in the fed state (1 h after initiation of a low-fat breakfast)
Regimen DEXPERIMENTALD - icovamenib capsule 100mg in the fed state (0.5 h after initiation of a high-fat breakfast)
Regimen EEXPERIMENTALE - icovamenib capsule 100mg in the fed state (1 h after initiation of a high-fat breakfast)
Regimen FEXPERIMENTALF - icovamenib HPMC capsule 100mg in the fed state (0.5 h after initiation of a high-fat breakfast)
Regimen GEXPERIMENTALG - icovamenib HPMC capsule 100mg in the fed state (1h after initiation of a high-fat breakfast)
Regimen HEXPERIMENTALH - icovamenib HPMC capsule 100mg in the fed state (0.5 h after initiation of a low-fat breakfast)
Regimen IEXPERIMENTALI - icovamenib HPMC capsule 100mg in the fed state (1 h after initiation of a low-fat breakfast)

Interventions

NameTypeDescription
icovamenib 100 mgDRUGicovamenib 100 mg
PlaceboDRUGMatching placebo
icovamenib 100mgDRUGicovamenib 100mg
IcovamenibDRUGInvestigational Product
Icovamenib HPMCDRUGInvestigational Product
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Eligibility Criteria

Age Range18 Years to 70 Years
SexALL
Healthy VolunteersNo
Study Sites17

Key Inclusion Criteria: 1. Males or females, age ≥18 years and ≤70 years 2. Have been diagnosed with T2D 3. Taking Ozempic (semaglutide injection) and have been treated with lifestyle management and 0 to 2 additional antihyperglycemic medications (metformin and/or SGLT2 inhibitor) with a stable dos...

Countries:United States
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Recent Changes (Last 90 Days)

MEDIUMAug 28, 2026NCT07502495Status: RECRUITING → ACTIVE_NOT_RECRUITING
MEDIUMAug 28, 2026NCT07502495Status: RECRUITING → ACTIVE_NOT_RECRUITING
LOWAug 7, 2026NCT07502495primaryCompletionDate: changed
LOWAug 7, 2026NCT07502495primaryCompletionDate: changed
LOWJun 16, 2026NCT07502508startDate: changed
LOWJun 16, 2026NCT07502508startDate: changed
LOWJun 16, 2026NCT07502508startDate: changed
LOWJun 16, 2026NCT07502508startDate: changed

Frequently asked questions about icovamenib

What is Icovamenib used for?

Icovamenib is an investigational small molecule being studied for Type 2 Diabetes. It is also being evaluated in healthy volunteers for a food effect study. The drug is in clinical development by Biomea Fusion, Inc. and is not yet approved.

What does Icovamenib target?

Icovamenib is a kinase inhibitor, as indicated by its '-nib' suffix. It is being studied for its potential role in treating Type 2 Diabetes. The specific molecular target has not been disclosed in clinical trial information.

Who makes Icovamenib?

Icovamenib is being developed by Biomea Fusion, Inc., a biopharmaceutical company traded under the ticker symbol BMEA. The company is conducting clinical trials of Icovamenib in the United States for Type 2 Diabetes and in healthy volunteers.

What phase is Icovamenib in?

Icovamenib is in Phase 2 clinical development for Type 2 Diabetes. A Phase 1 food effect study in healthy volunteers has been completed. The drug is investigational and has not received FDA approval.

What clinical trials is Icovamenib in?

Icovamenib is being studied in two Phase 2 trials: NCT07502495 in participants with Type 2 Diabetes not achieving glycemic targets, and NCT07502508 in those not achieving targets while using GLP-1-based therapy. A Phase 1 food effect study, NCT07254286, has been completed.

Is Icovamenib the same as icovamenib 100mg?

Yes, Icovamenib is also known as icovamenib 100mg or icovamenib 100 mg. These names refer to the same drug substance being developed by Biomea Fusion, Inc. for Type 2 Diabetes.