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MEDI-4166

Phase 1

Type 2 Diabetes | Monoclonal antibody | Metabolic |AstraZeneca PLC|Last Updated: Mar 13, 2019

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment103
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02524782A Phase 1, Single- and Multiple Dose Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of MEDI4166 in Subjects With Type 2 DiabetesPHASE1 COMPLETED 103Oct 7, 2015Apr 14, 2017Mar 13, 201911 United States
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Study Endpoints
Primary Endpoints
Part A: Number of subjects with adverse events as a measure of safety and tolerability of MEDI4166
43 days post dosing

Treatment emergent adverse events (TEAEs) and serious adverse events (TESAEs)

Part B: Change in glucose AUC measured up to 240 minutes after mixed meal tolerance test (MMTT) from baseline to Day 36
36 days post dosing
Part B: Change in LDL-C from baseline to Day 36
36 days post dosing
Secondary Endpoints
Part A: Pharmacokinetics of MEDI4166, maximum plasma concentration (Cmax)
43 days post dosing
Part A: Pharmacokinetics of MEDI4166, area under the curve concentration (AUC)
43 days post dosing
Part A: Change from baseline in LDL-C
43 days post dosing
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
MEDI-4166EXPERIMENTALMEDI-4166 administered subcutaneously
PlaceboPLACEBO_COMPARATORPlacebo administered subcutaneously
Interventions
NameTypeDescription
MEDI-4166BIOLOGICALMEDI-4166 administered subcutaneously
PlaceboBIOLOGICALPlacebo administered subcutaneously
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersNo
Study Sites11

Inclusion Criteria: * Type 2 Diabetes, ages 18-65 * Must provide written informed consent * BMI\>=25 and =\<42 * Venous access suitable for multiple cannulations * Vital signs within normal specified ranges * Females must be non-lactating and non-childbearing potential * Males must practice 2 effec...

Countries:United States
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