Recent Updates
Recently added Catalysts

Teriflunomide HMR1726

Phase 3

Multiple Sclerosis | Small molecule | Immunology |Sanofi|Last Updated: Mar 13, 2015

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
NO_TREATMENT_CONTROLLEDBiomarker
Total Trials2
Total Enrollment82
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01863888Effect of Teriflunomide on Immune Cell Subsets in the Blood of Patients With Multiple SclerosisPHASE3 COMPLETED 70Oct 1, 2013Jan 1, 2015Mar 13, 201510 Belgium, Germany +1
NCT02046629A Study to Evaluate the Pharmacokinetic Profiles of Single 14 mg Teriflunomide Tablet in Healthy Chinese VolunteersPHASE1 COMPLETED 12May 1, 2014Jul 1, 2014Aug 21, 20141 China
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Change from baseline in Lymphocyte subset parameters as measured by flow cytometry
At 12 weeks and 24 weeks
Pharmacokinetic parameters for teriflunomide determined from plasma concentration
5 weeks
Secondary Endpoints
Change from baseline in biased T cell clonal repertoire based T cell receptor (TCR) spectratyping
At 12 weeks and 24 weeks
Change from baseline in serum cytokine as measured by multicytokine array tool
At 12 weeks and 24 weeks
Change from baseline in Mitogen/TCR-specific T cell proliferation as measured by flow cytometry
At 12 weeks and 24 weeks
Unlock Study Endpoints
Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
teriflunomide (HMR1726)EXPERIMENTALParticipants administered 14mg Teriflunomide once daily, oral. For participants who permanently discontinue Teriflunomide, an accelerated elimination procedure with either cholestyramine or charcoal will be administered.
Reference populationNO_INTERVENTIONUntreated healthy subjects
teriflunomide dose 1EXPERIMENTALTeriflunomide 14mg tablet, oral single dose, fast condition Cholestyramine power, 8 gram,oral three times a day for 4 days, fed condition
Interventions
NameTypeDescription
teriflunomide HMR1726DRUGPharmaceutical form:tablet Route of administration: oral
cholestyramineDRUGPharmaceutical form:powder Route of administration: oral
charcoalDRUGPharmaceutical form:granule Route of administration: oral
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites10

Inclusion criteria: Patients (male and female) with relapsing forms of multiple sclerosis meeting McDonald criteria for MS at the screening visit and having either one of the following treatment status: * Naïve to disease modifying (DM) treatment or no DM treatment for more than 2 years * Or curre...

Countries:BelgiumGermanyNetherlandsChina
Unlock Eligibility Criteria