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ORIC-944

Phase 1

Metastatic Prostate Cancer | Small molecule | Oncology |Oric Pharmaceuticals, Inc.|Last Updated: Aug 11, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment250
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT05413421Study of ORIC-944 in Patients With Metastatic Prostate CancerPHASE1 RECRUITING 250Jun 1, 2022Sep 1, 2026Aug 11, 202527 United States, Australia +2
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Study Endpoints
Primary Endpoints
Recommended Phase 2 Dose (RP2D)
12 months

RP2D as determined by interval 3+3 dose escalation design

Maximum plasma concentration (Cmax)
28 Days

PK of ORIC-944 single agent and in combination with an ARPI

Time to maximum observed concentration (Tmax)
28 Days

PK of ORIC-944 single agent and in combination with an ARPI

Area under the curve (AUC)
28 Days

PK of ORIC-944 single agent and in combination with an ARPI

Apparent plasma terminal elimination half-life (t1/2)
28 Days

PK of ORIC-944 single agent and in combination with an ARPI

Secondary Endpoints
Clinical benefit rate (CBR)
36 months
Objective response rate (ORR)
36 months
Duration of response (DOR)
36 months
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Single Agent Dose EscalationEXPERIMENTALORIC-944 dosed orally on a continuous daily dosing regimen in 28-day cycles
Combination Dose EscalationEXPERIMENTALORIC-944 dosed orally on a continuous daily dosing regimen in 28-day cycles in combinations with abiraterone, apalutamide, darolutamide, or enzalutamide
Combination Dose OptimizationEXPERIMENTALCohort A and C: ORIC-944 dosed orally on a continuous daily dosing regimen in 28-day cycles in combination with apalutamide Cohort B and D: ORIC-944 dosed orally on a continuous daily dosing regimen in 28-day cycles in combination with darolutamide Combinations with abiraterone or enzalutamide may be conducted in the future
Interventions
NameTypeDescription
ORIC-944DRUGOral, once daily, continuous
Abiraterone acetate (Zytiga®) 250 mg or 500 mg tabletsDRUGOral, 1000 mg once daily, continuous
Apalutamide (Erleada™) 60 mg or 240 mg tabletsDRUGOral, 240 mg once daily, continuous
Darolutamide (Nubeqa®) 300 mg tabletsDRUGOral, 600 mg twice daily, continuous
Enzalutamide (Xtandi®) 40 mg capsules or 40 mg and 80 mg tabletsDRUGOral, 160 mg once daily, continuous
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Eligibility Criteria
Age Range18 Years — N/A
SexMALE
Healthy VolunteersNo
Study Sites27

Inclusion Criteria: * Patients with metastatic prostate cancer * Must have undergone bilateral orchiectomy or be willing to continue GnRH analogue or antagonist to maintain castrate levels of testosterone * Prior therapies: Part I (single agent ORIC-944 dose escalation): Any number of prior therap...

Countries:United StatesAustraliaSpainUnited Kingdom
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Competitive Landscape -Prostate Cancer 259 trials
CompanyTickerTrialsLead PhaseDrugs
Merck & Co., Inc.MRK7PHASE3Pembrolizumab, Enzalutamide, Ifinatamab deruxtecan, Docetaxel, Prednisone
AstraZeneca PLCAZN20PHASE3olaparib, abiraterone, Saruparib, Abiraterone, Darolutamide
Pfizer Inc.PFE12PHASE3Talazoparib with enzalutamide, PF-06821497, Docetaxel, Enzalutamide, Leuprolide Open Label
Johnson & JohnsonJNJ21PHASE3Apalutamide, Androgen Deprivation Therapy, Niraparib, Abiraterone, Prednisone
Eli Lilly and CompanyLLY9PHASE3Abemaciclib, Abiraterone, Prednisone or Prednisolone, -PNT2002, Enzalutamide
Amgen Inc.AMGN7PHASE3Xaluritamig, Abiraterone, Enzalutamide, Cabazitaxel, Docetaxel
Novartis AG Sponsored ADRNVS28PHASE3177Lu-PSMA-617, 68Ga-PSMA-11, ARDT, ADT, AAA617
Exelixis, Inc.EXEL4PHASE3Cabozantinib, Atezolizumab, Abiraterone, Enzalutamide, Prednisone
Candel Therapeutics, Inc.CADL3PHASE3Aglatimagene besadenovec + valacyclovir, aglatimagene besadenovec, valacyclovir, aglatimagene besadenovec + valacyclovir
Bristol-Myers Squibb CompanyBMY2PHASE3BMS-986365, Enzalutamide, Abiraterone, Docetaxel, Predinsone/Prednisolone
BioNTech SE Sponsored ADRBNTX1PHASE3BNT324, Docetaxel, Prednisone/prednisolone
Telix Pharmaceuticals Limited Sponsored ADRTLX3PHASE368Ga-PSMA-11, 177Lu-TLX591, Enzalutamide, Abiraterone, Docetaxel
Sanofi SA Sponsored ADRSNY2PHASE3abiraterone, Docetaxel, Cabazitaxel
Regeneron Pharmaceuticals, Inc.REGN4PHASE2REGN2810, Degarelix, Leuprolide, Docetaxel, BPX-601
Veracyte, Inc.VCYT2PHASE2Darolutamide, Zoladex, Zoladex LA, Decapeptyl sustained release, Depo-Eligard
Kyntra Bio, Inc.KYNB2PHASE2FG-3246, FOR46, Enzalutamide, Pegfilgrastim
Lantheus Holdings IncLNTH3PHASE3Undisclosed
IDEAYA Biosciences, Inc.IDYA3PHASE1IDE-161, Pembrolizumab, IDE034, IDE574, Fulvestrant
Xencor, Inc.XNCR1PHASE2vudalimab
GSK plc Sponsored ADRGSK2PHASE1GSK5471713, GSK5458514
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Recent Changes (Last 90 Days)
LOWMay 26, 2026NCT05413421primaryCompletionDate: changed
LOWMay 24, 2026NCT05413421studyFirstPostDate: changed