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Amlodipine

Phase 3

Hypertension | Small molecule | Cardiovascular |Novartis AG|Last Updated: Aug 4, 2020

Target and mechanism

ModalitySmall molecule

Also known as Amlodipine (Optional)

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindCONTROLLED
Total Trials5
Total Enrollment4,745

FDA Designations

No designations recorded

Clinical trial landscape

Amlodipine · 5 trials · 1 indication

Phase 3 5
NCT00797862Aliskiren and the Calcium Channel Blocker Amlodipine Combination as an Initial Treatment Strategy for HypertensionHypertension
COMPLETED1,254 Analytics
NCT00778921Study to Evaluate the Efficacy and Safety of Combination Aliskiren/Amlodipine in Patients With Hypertension Not Adequately Responding to Amlodipine AloneHypertension
COMPLETED847 Analytics
NCT00699192Safety, Tolerability, and Efficacy of Once Daily Amlodipine/Valsartan 5/80 as Compared to Amlodipine/Valsartan 5/40 or to Amlodipine 5 mg Monotherapy in Patients 65 Years of Age and Older With Essential HypertensionHypertension
COMPLETED965 Analytics
NCT00523744Efficacy and Safety of Valsartan and Amlodipine (± HCTZ) in Adults With Moderate, Inadequately Controlled HypertensionHypertension
COMPLETED257 Analytics
NCT00171366A Study Comparing the Response of Patients With Hypertension to Amlodipine or Amlodipine Plus Benazepril.Hypertension
COMPLETED1,422 Analytics
PHASE3COMPLETED
Aliskiren and the Calcium Channel Blocker Amlodipine Combination as an Initial Treatment Strategy for Hypertension
HypertensionUnlock trial analytics
PHASE3COMPLETED
Study to Evaluate the Efficacy and Safety of Combination Aliskiren/Amlodipine in Patients With Hypertension Not Adequately Responding to Amlodipine Alone
HypertensionUnlock trial analytics
PHASE3COMPLETED
Safety, Tolerability, and Efficacy of Once Daily Amlodipine/Valsartan 5/80 as Compared to Amlodipine/Valsartan 5/40 or to Amlodipine 5 mg Monotherapy in Patients 65 Years of Age and Older With Essential Hypertension
HypertensionUnlock trial analytics
PHASE3COMPLETED
Efficacy and Safety of Valsartan and Amlodipine (± HCTZ) in Adults With Moderate, Inadequately Controlled Hypertension
HypertensionUnlock trial analytics
PHASE3COMPLETED
A Study Comparing the Response of Patients With Hypertension to Amlodipine or Amlodipine Plus Benazepril.
HypertensionUnlock trial analytics

Study Endpoints

Primary Endpoints

Overall Mean Change From Baseline in Mean Sitting Systolic Blood Pressure (msSBP) Over 8, 16 and 24 Weeks
Baseline, 8 weeks, 16 weeks, and 24 weeks

Systolic Blood Pressure was measured in a sitting position using a validated automated blood pressure monitor (the Omron device) according to Guidelines of the British Hypertension Society, at Baseline and over 8, 16 and 24 weeks of study treatment. The overall mean change in msSBP from baseline was estimated over three time points: Week 8, Week 16, and Week 24. Analysis used a repeated measures Analysis of Covariance (ANCOVA) model with treatment, visit, and region as factors, treatment by visit interaction and baseline msSBP as a covariate.

Change From Baseline in Mean Sitting Systolic Blood Pressure (msSBP) at Week 24
Baseline to 24 weeks

Systolic Blood pressure was measured in a sitting position using a validated automated blood pressure monitor (the Omron device) according to Guidelines of the British Hypertension Society, at Baseline and 24 weeks of study treatment. Analysis used a repeated measures ANCOVA model with treatment, visit and region as factors, treatment by visit interaction and baseline msSBP as a covariate.

Change in Mean Sitting Diastolic Blood Pressure (msDBP) From Baseline to End of Study
Baseline and Week 8
Change in Mean Sitting Systolic Blood Pressure (msSBP) From Baseline to End of Study (Week 8)
Baseline to end of study (Week 8)

At study entry, blood pressure (BP) was measured in both arms with an automatic BP monitor. The arm with the higher systolic BP reading was used for all measurements throughout the study. At each study visit, 3 separate sitting BPs were obtained 23-26 hours post-dose with at least 2 minutes between measurements and with the cuff fully deflated. Mean BP was automatically calculated from the 3 readings. A negative change from baseline indicates lowered BP.

Change in Mean Sitting Diastolic Blood Pressure (msDBP) During the Core Phase of the Study
Baseline Phase 2 (Week 4) to end of Phase 2 (Week 8)

The arm in which the highest sitting diastolic pressures were found at study entry was the arm used for all subsequent readings. A calibrated sphygmomanometer and appropriate size cuff were used to measure arterial sitting blood pressure (BP) at trough with the arm supported at the level of the heart. At each study visit, after having the patient in a sitting position for at least 5 minutes, systolic/diastolic blood pressure were measured 3 times at 1-2 minute intervals. A mean was calculated from the 3 measurements. A negative change indicates improvement.

Change in Mean Sitting Diastolic Blood Pressure (msDBP) During the Extension Phase of the Study
Baseline Phase 3 (Week 8) to end of Phase 3 (Week 12)

The arm in which the highest sitting diastolic pressures were found at study entry was the arm used for all subsequent readings. A calibrated sphygmomanometer and appropriate size cuff were used to measure arterial sitting blood pressure (BP) at trough with the arm supported at the level of the heart. At each study visit, after having the patient in a sitting position for at least 5 minutes, systolic/diastolic blood pressure were measured 3 times at 1-2 minute intervals. A mean was calculated from the 3 measurements. A negative change indicates improvement.

Change from baseline in mean sitting diastolic blood pressure at week 6

Secondary Endpoints

Change From Baseline in Mean Sitting Diastolic Blood Pressure (msDBP) at Week 32
Baseline to 32 weeks
Overall Mean Change From Baseline in Mean Sitting Diastolic Blood Pressure (msDBP) Over 8, 16, and 24 Weeks
Baseline, 8 weeks, 16 weeks and 24 weeks
Change From Baseline in Mean Sitting Diastolic Blood Pressure (msDBP) at Week 24
Baseline to 24 weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeDIAGNOSTIC

Treatment Arms

ArmTypeDescription
Aliskiren + AmlodipineEXPERIMENTALEligible participants received oral aliskiren 150 mg + amlodipine 5 mg daily from week 1-8. From week 8 - 16, the dose of the combination treatment increased to aliskiren 300 mg + amlodipine 10 mg daily. From week 16-24, participants in this group continued combination treatment (aliskiren 300 mg + amlodipine 10 mg) for 8 weeks. At week 24, if blood pressure was not adequately controlled (systolic blood pressure \>140 mmHg or diastolic blood pressure \>90 mmHg) hydrochlorothiazide 12.5 mg was added to the combination (aliskiren 300 mg + amlodipine 10 mg) for an additional 8 weeks. Total treatment period =32 weeks.
Aliskiren Start - Amlodipine Add-OnEXPERIMENTALEligible participants received oral aliskiren 150 mg daily from week 1-8. From week 8 - 16, the dose of aliskiren increased to 300 mg daily. From week 16-24, amlodipine 10 mg was added to the aliskiren 300 mg for 8 weeks (aliskiren 300 mg + amlodipine 10 mg). At week 24, if blood pressure was not adequately controlled (systolic blood pressure \>140 mmHg or diastolic blood pressure \>90 mmHg) hydrochlorothiazide 12.5 mg was added to the combination (aliskiren 300 mg + amlodipine 10 mg) for an additional 8 weeks. Total treatment period =32 weeks.
Amlodipine Start- Aliskiren Add-OnEXPERIMENTALEligible participants received oral amlodipine 5 mg daily from week 1-8. From week 8 - 16, the dose of amlodipine increased to 10 mg daily. From week 16-24, aliskiren 300 mg was added to the amlodipine 10 mg for 8 weeks (amlodipine 10 mg + aliskiren 300 mg). At week 24, if blood pressure was not adequately controlled (systolic blood pressure \>140 mmHg or diastolic blood pressure \>90 mmHg) hydrochlorothiazide 12.5 mg was added to the combination (amlodipine 10 mg + aliskiren 300 mg) for an additional 8 weeks. Total treatment period =32 weeks.
Amlodipine 10 mgEXPERIMENTALAmlodipine 10 mg
Aliskiren/Amlodipine 150/10 mgEXPERIMENTALAliskiren/Amlodipine 150/10 mg
Aliskiren/Amlodipine 300/10 mgEXPERIMENTALAliskiren/Amlodipine 300/10 mg
Amlodipine/Valsartan 5/80 mgEXPERIMENTAL1 capsule amlodipine 5 mg, 1 capsule valsartan 80 mg once daily
Amlodipine/Valsartan 5/40 mgACTIVE_COMPARATOR1 capsule amlodipine 5 mg, 1 capsule valsartan 40 mg once daily
Amlodipine 5 mgACTIVE_COMPARATOR1 capsule amlodipine 5 mg, 1 capsule placebo to match valsartan once daily
Amlodipine(AML)+olmesartan, AML+valsartan, AML+valsartan+HCTZEXPERIMENTALDuring the Treatment Phase 1, participants received 1 week of treatment with olmesartan 10 mg and amlodipine 5 mg once daily in free combination, followed by three weeks of treatment with olmesartan 20 mg plus amlodipine 10 mg once daily in free combination. During the treatment Phase 2 of the study participants received amlodipine 10 mg plus valsartan 160 mg for 4 weeks. During the Extension Phase, participants received 4 weeks treatment with amlodipine 10 mg plus valsartan 160 mg plus hydrochlorothiazide (HCTZ) 12.5 mg.

Interventions

NameTypeDescription
AmlodipineDRUGAmlodipine (5 mg and 10 mg) was provided as capsules taken orally once daily.
hydrochlorothiazideDRUGHydrochlorothiazide 12.5 mg capsules were taken orally once daily
AliskirenDRUGAliskiren 150 mg and aliskiren 300 mg were provided as film-coated tablets, taken orally once daily.
Amlodipine 10 mgDRUGAmlodipine 10 mg
Aliskiren 150DRUGAliskiren/Amlodipine 150/10 mg
Amlodipine 300DRUGAliskiren/Amlodipine 300/10 mg
Amlodipine 5 mgDRUG1 capsule amlodipine 5 mg orally once daily
Valsartan 80 mgDRUG1 capsule valsartan 80 mg orally once daily
Valsartan 40 mgDRUG1 capsule valsartan 40 mg orally once daily
PlaceboDRUG1 capsule placebo to match valsartan orally once daily
Olmesartan medoxomilDRUGOlmesartan medoxomil supplied as 10 mg tablets taken once a day during Treatment Phase 1 only.
Amlodipine+valsartanDRUGFixed-dose combination of amlodipine 10 mg plus valsartan 160 mg tablet taken orally once a day during Treatment Phase 2 and Extension Phase.
amlodipine/benazeprilDRUG -
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites10

Inclusion Criteria: * Male or female outpatients ≥ 18 years of age * Participants with essential hypertension: * Naive participants must have a mean sitting Systolic Blood Pressure (msSBP) ≥ 150 mmHg and \< 180 mmHg at Visit 1 and Visit 2. (Participants are considered 'naïve' if they have never ...

Countries:CanadaCosta RicaFranceGermanyGreeceGuatemalaSouth AfricaSwitzerlandUnited KingdomVenezuelaArgentinaNorwayPolandSlovakiaSwedenTurkey (Türkiye)CzechiaFinlandHungaryItalySpainUnited States
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