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Fursemide for administration

Phase 2

Heart Failure | Small molecule | Cardiovascular |MannKind Corporation|Last Updated: Dec 2, 2022

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment23

FDA Designations

No designations recorded

Clinical trial landscape

Fursemide for administration · 1 trial · 1 indication

Phase 2 1
NCT02329834Crossover Study to Compare the Pharmacokinetics and Bioavailability of a Novel Furosemide Regimen Administered Subcutaneously vs. the Same Dose Administered Intravenously in Subjects With Chronic Heart FailureHeart Failure
COMPLETED23 Analytics
PHASE2COMPLETED
Crossover Study to Compare the Pharmacokinetics and Bioavailability of a Novel Furosemide Regimen Administered Subcutaneously vs. the Same Dose Administered Intravenously in Subjects With Chronic Heart Failure
Heart FailureUnlock trial analytics

Study Endpoints

Primary Endpoints

Cmax
0, 5 min, 15 min, 30 min, 45 min, 60 min, 1.5 hours, 2 hours, 2:05 min, 2:15 min, 2:30 min, 2:45 min, 3 hours, 3:30 min, 4, 5, 6, 8, 10, 12, 14, and 16 hours post-dose

Maximum observed plasma concentration of Furosemide

Tmax
0, 5 min, 15 min, 30 min, 45 min, 60 min, 1.5 hours, 2 hours, 2:05 min, 2:15 min, 2:30 min, 2:45 min, 3 hours, 3:30 min, 4, 5, 6, 8, 10, 12, 14, and 16 hours post-dose

Time to achieve maximum observed Furosemide plasma concentration

AUClast
0, 5 min, 15 min, 30 min, 45 min, 60 min, 1.5 hours, 2 hours, 2:05 min, 2:15 min, 2:30 min, 2:45 min, 3 hours, 3:30 min, 4, 5, 6, 8, 10, 12, 14, and 16 hours post-dose

The area under the plasma concentration versus time curve from time 0 (pre-dose) to the last quantifiable time point.

AUCinf
0, 5 min, 15 min, 30 min, 45 min, 60 min, 1.5 hours, 2 hours, 2:05 min, 2:15 min, 2:30 min, 2:45 min, 3 hours, 3:30 min, 4, 5, 6, 8, 10, 12, 14, and 16 hours post-dose

The area under the plasma concentration-time curve from time 0 (pre-dose) to time of last measurable plasma concentration.

AUCext
0, 5 min, 15 min, 30 min, 45 min, 60 min, 1.5 hours, 2 hours, 2:05 min, 2:15 min, 2:30 min, 2:45 min, 3 hours, 3:30 min, 4, 5, 6, 8, 10, 12, 14, and 16 hours post-dose

The percentage of AUC that is extrapolated beyond the last measurable concentration

λz
24 hours

Apparent plasma terminal-phase elimination rate constant

t 1/2
24 hours

Terminal-phase half life

Volume of Distribution, Terminal Phase
24 hours

Systemic Volume of distribution, terminal phase for IV furosemide and Apparent Volume of distribution, terminal phase for SC furosemide

CL
24 hours

Systemic Clearance for IV furosemide and Apparent Systemic Clearance for SC furosemide

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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Treatment Sequence 1EXPERIMENTALFurosemide Injection Solution for subcutaneous administration (80mg) over 5 hours followed by i.v. Furosemide Injection, USP (80 mg)by i.v. bolus in second period
Treatment Sequence 2EXPERIMENTALFurosemide Injection, USP (80 mg) by i.v. bolus, followed by Furosemide Injection Solution for subcutaneous administration (80mg) over 5 hours in second period.

Interventions

NameTypeDescription
Fursemide Injection Solution for subcutaneous administration (80 mg)DRUGFurosemide Injection Solution, 10mL of undiluted buffered furosemide solution (8mg/mL)
Furosemide Injection, USPDRUGFurosemide Injection, USP (10mg/mL), 80 mg by intravenous administration.
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * An Institutional Review Board (IRB) approved informed consent is signed and dated prior to any study-related activities. * Male and female subjects ≥18 years of age, with body volume and weight \<130 kg and body mass index (BMI) \<38 kg/m2 * Females will be non-pregnant, non-l...

Countries:United States
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