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Exenatide

Phase 3

Coronary Artery Disease | Small molecule | Cardiovascular |Eli Lilly and Company|Last Updated: Mar 9, 2021

Success Probability

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Trial Design

RandomizedNO_TREATMENT_CONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment38

FDA Designations

No designations recorded

Clinical trial landscape

Exenatide · 3 trials · 4 indications

Phase 3 1Phase 2 2
NCT01373216Glucagon-like Peptide 1 Agonist Exenatide for Improved Glucose Control and Cardiac Function in Patients With Aortocoronary BypassCoronary Artery Disease
COMPLETED38 Analytics
PHASE3COMPLETED
Glucagon-like Peptide 1 Agonist Exenatide for Improved Glucose Control and Cardiac Function in Patients With Aortocoronary Bypass
Coronary Artery DiseaseUnlock trial analytics

Study Endpoints

Primary Endpoints

Cardiac function - echocardiographic parameters
90 days after administration of exenatide

* cardiac chamber dimensions * left ventricular systolic function * left ventricular diastolic function * right ventricular systolic function

Percentage of patients spending more than 50 % of the time in the glycemic target range (100 to 140 mg/dl)
48 hours

The percentage of time spent achieving blood glucose control is defined as the ratio between the total time spent achieving blood glucose control and the total time under treatment. Blood glucose measurement will be done hourly. Blood glucose control is considered to be achieved between 2 blood glucose measurements if the first blood glucose value measured belongs to blood glucose target interval, defined as blood glucose level between 100 mg/dl l and 140 mg/dl l.

Variation of the SF-36 score value at 3-months
3 months

The SF-36 score is a self-administered questionnaire that assess both the physical and the psychosocial health-related quality of life. The use of the SF-36 score is recommended by the French Health Authority in coronary patients. The variation of the SF-36 score value at 3-months is defined as the difference between the SF36-score value at 3 months minus the preoperative SF-36 score value.

Secondary Endpoints

Number of participants with adverse effects
90 days after administration of exenatide
Hypoglycemia
48 hours
Severe hypoglycemia
48 hours
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Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ExenatideEXPERIMENTALPatients with decreased left ventricular function undergoing elective coronary artery by-pass grafting receiving perioperatively i.v. exenatide on top of standard treatment
ControlNO_INTERVENTIONPatients with decreased left ventricular function undergoing elective coronary artery by-pass grafting receiving standard treatment
Exenatide groupEXPERIMENTALExenatide. Exenatide: bolus of 0.05 µg/min infused during the 1st hour of treatment, followed by a continuous infusion of 0.025 µg/min until the end of treatment. The exenatide therapy will begin as soon as a blood glucose level is above 140 mg/dl will be measured. A of exenatide will be intravenously . The treatment will be administrated during the first postoperative 48 hours in the intensive care unit or until intensive care unit discharge if this event occurs earlier.
Insulin groupACTIVE_COMPARATORInsulin: Humalog (insulin lispro human analog). The insulin therapy will begin as soon as a blood glucose level is above 140 mg/dl will be measured. The dose of insulin intravenously infused will be adapted to blood glucose measurements, following the insulin therapy protocol used in our department. The insulin therapy protocol used in our department and prescribed as the benchmark treatment in the present study has been validated in a previous study. It has been derived from the protocol validated by Goldberg et al.

Interventions

NameTypeDescription
ExenatideDRUGPerioperative continuous i.v. administration of exenatide lasting for 72 hours - 40 ng/min for initial 30 min, 20 ng/min for remaining 71.5 hours
InsulinDRUG -
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Eligibility Criteria

Age Range18 Years to 85 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * elective coronary artery bypass grafting operation (CABG) * decreased left ventricular (LV) systolic function (EF LV ≤ 50%) * Age 18 to 85 * Signed informed consent * Females with childbearing potential have to use appropriate contraceptive measures during the whole study peri...

Countries:CzechiaFrance
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Frequently asked questions about Exenatide

What is Exenatide used for?

Exenatide is being studied for use in stress hyperglycemia, coronary artery disease, and quality of life in cardiac surgery patients. It is a small molecule in Phase 3 development for these cardiovascular-related conditions. The drug is being developed by Eli Lilly and Company.

What does Exenatide target?

Exenatide is a glucagon-like peptide 1 (GLP-1) agonist, as indicated in the clinical trial title. It targets the GLP-1 receptor to help improve glucose control and cardiac function in patients with coronary artery disease.

Who makes Exenatide?

Exenatide is being developed by Eli Lilly and Company, which trades under the ticker LLY. The company is conducting clinical trials to evaluate the drug for stress hyperglycemia, coronary artery disease, and quality of life improvements.

What phase is Exenatide in?

Exenatide is in Phase 3 clinical development for stress hyperglycemia, coronary artery disease, and quality of life. It is an investigational drug and has not been approved by the FDA for these indications. The drug is still undergoing clinical trials.

What clinical trials is Exenatide in?

Exenatide has been studied in three completed clinical trials: NCT01373216 for coronary artery disease and decreased left ventricular function, NCT01969149 for stress hyperglycemia, and NCT02432976 for quality of life in cardiac surgery patients. The trials were conducted in Czechia and France.

Is Exenatide the same as GLP-1 agonist?

Exenatide is a type of GLP-1 agonist, as described in the clinical trial title. It is specifically a glucagon-like peptide 1 agonist, which means it mimics the action of the natural GLP-1 hormone to regulate glucose levels.