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PS433540

Phase 2

Hypertension | Small molecule | Cardiovascular |Ligand Pharmaceuticals Incorporated|Last Updated: Sep 16, 2011

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials2
Total Enrollment541
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00635232A Study To Evaluate The Dose-Related Efficacy and Safety of PS433540 in Subjects With HypertensionPHASE2 COMPLETED 261Mar 1, 2008Dec 1, 2008Sep 16, 201140 United States
NCT00522925A Trial to Evaluate the Safety and Efficacy of PS433540 to Treat HypertensionPHASE2 COMPLETED 280Aug 1, 2007May 1, 2008Sep 16, 201115 United States
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Study Endpoints
Primary Endpoints
Change From Baseline in Mean Seated Systolic Blood Pressure (SBP) Following 12 Weeks of Treatment With PS433540 200 mg, 400 mg, 800 mg and Placebo.
12 weeks
Change From Baseline in Mean 24-hour Ambulatory Systolic Blood Pressure
4 weeks of treatment with PS43540
Secondary Endpoints
Change From Baseline in Mean Seated Diastolic Blood Pressure (DBP) Following 12 Weeks of Treatment With PS433540 200 mg, 400 mg, 800 mg and Placebo.
12 weeks
The Percentage of Patients Treated With Each Dose of PS433540 Who Achieved Blood Pressure Control, Defined as <140/90 mmHg, After 12 Weeks of Treatment.
12 weeks
Change From Baseline in Mean 24-hour Ambulatory Diastolic Blood Pressure
4 weeks of treatment with PS43540
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Irbesartan 300mgACTIVE_COMPARATORIrbesartan 300 mg once daily
PlaceboPLACEBO_COMPARATORBlinded Placebo Treatment
PS433540 200mgEXPERIMENTALPS433540 200mg once daily
PS433540 400mgEXPERIMENTALPS433540 400mg once daily
PS433540 800mgEXPERIMENTALPS433540 800mg once daily
1PLACEBO_COMPARATORMatching Placebo
2EXPERIMENTAL -
3EXPERIMENTAL -
Interventions
NameTypeDescription
irbesartanDRUG300 mg (2 x 150 mg capsules) once daily for 12 weeks
placeboDRUGplacebo capsules once daily for 12 weeks
PS433540DRUG200 mg (2 x 100 mg capsules) once daily for 12 weeks
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersNo
Study Sites40

Inclusion Criteria: * Males or females 18 - 70 years * Mean seated Systolic Blood Pressure (SBP) ≥ 140 mmHg and \< 180 mmHg and mean seated Diastolic Blood Pressure (DBP) \> 90 and \< 109 mmHg at two consecutive qualifying visits (Visits 3/3.5 and Visit 4). The mean difference in DBP between the tw...

Countries:United States
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