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Relacatib

Phase 1

Osteoarthritis | Small molecule | Musculoskeletal |GSK plc|Last Updated: Oct 4, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment32
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00411190Study To Determine The Effects Of Doses Of Relacatib On The Metabolism Of Acetaminophen, Ibuprofen And AtorvastatinPHASE1 COMPLETED 32Oct 19, 2006Dec 15, 2006Oct 4, 20172 Belgium
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Study Endpoints
Primary Endpoints
The primary objective of this study is to characterize the effect of relacatib at steady-state on the pharmacokinetics of a single oral dose of acetaminophen, ibuprofen and atorvastatin in healthy postmenopausal females.
Up to Day 17
Secondary Endpoints
To assess the safety and tolerability of the concomitant administration of oral doses of relacatib and acetaminophen, ibuprofen and atorvastatin. To describe the changes from baseline in serum CTXI levels for each relacatib dose tested.
Up to Day 17
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeDIAGNOSTIC
Treatment Arms
ArmTypeDescription
Session 1EXPERIMENTALSubjects will receive 500 mg acetaminophen on Day 1, 400 mg ibuprofen on Day 2, 40 mg atorvastatin on Day 3.
Session 2EXPERIMENTALSubjects will be randomized to receive relacatib 60 mg or 120 mg from Day 1-14. On Day 15 subjects will receive 500 mg acetaminophen, 400 mg ibuprofen on Day 16 and 40 mg atorvastatin on Day 17 with usual dose of relacatib.
Interventions
NameTypeDescription
RelacatibDRUGSubjects will administer 60 or 120 mg tablets in Session 2
AcetaminophenDRUGAcetaminophen will be administered orally
IbuprofenDRUGIbuprofen will be administered orally
AtorvastatinDRUGAtorvastatin will be administered orally
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Eligibility Criteria
Age Range18 Years — 70 Years
SexFEMALE
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * Healthy * Postmenopausal * Body weight \> 50 kg * Body mass index (BMI) between 19 and 30 * The subject is willing and able to give a signed and dated written informed consent prior to admission to the study * The subject is able to understand and comply with protocol requirem...

Countries:Belgium
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