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BAY1067197

Phase 2

Heart Failure | Small molecule | Cardiovascular |Bayer AG|Last Updated: Sep 19, 2019

Success Probability

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials2
Total Enrollment42

FDA Designations

No designations recorded

Clinical trial landscape

BAY1067197 · 2 trials · 1 indication

Phase 2 2
NCT02040233Multiple Dose Study in Heart Failure of BAY 1067197Heart Failure
COMPLETED31 Analytics
NCT01945606Study to Assess the Safety of BAY1067197 in Stable Heart Failure Patients on Standard Therapy Including ß-blockerHeart Failure
COMPLETED11 Analytics
PHASE2COMPLETED
Multiple Dose Study in Heart Failure of BAY 1067197
Heart FailureUnlock trial analytics
PHASE2COMPLETED
Study to Assess the Safety of BAY1067197 in Stable Heart Failure Patients on Standard Therapy Including ß-blocker
Heart FailureUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of Subjects With Relevant Changes in Heart Rate
From the start of study treatment up to Day 29

Heart rate was measured by monitor measurements after 30 minutes resting in a supine position. The relevant changes in heart rate were recorded and analysed.

Number of Subjects With Relevant Changes in Blood Pressure
From the start of study treatment up to Day 29

Blood pressure was measured by monitor measurements after 30 minutes resting in a supine position. The relevant changes in blood pressure were recorded and analysed.

Number of Subjects With More than First Degree Atrio-Ventricular (AV) Block
After 7 day tratment and day 28

A complete standard 12-lead ECG was recorded and evaluated parameters such as heart rate, PR/PQinterval, QRSD interval, QT interval (uncorrected). Clinically relevant findings in ECG such as a second degree AV-block Mobitz type I (Wenkebach), Mobitz type II - or any third-degree AV block were recorded and reported. A 24-hour Holter ECG was recorded with a standard Holter ECG recorder for the purpose of detecting AV blocks, no higher degree AV blocks \> 1 or clinically relevant effect on HR were observed during Holter monitoring periods.

Change From Baseline in Left Ventricular Ejection Fraction (LVEF)
Baseline to day 7

The change in LVEF between the post and the pre-treatment measurements were analyzed using Bayesian statistics to quantify the difference between BAY1067197 treatment and placebo measured by CMR. LVEF is the fraction of blood (in percent) pumped out of the heart's left ventricular chamber with each heart beat, and is a measure of cardiac output for the heart.

Maximum Observed Concentration of BAY84-3174 in Plasma (Cmax) After First Dose of BAY1067197
Day 1: pre-dose and 0.5, 1, 2, 3, 4, 6, 12 and 24 hours post-dose

Maximum observed BAY84-3174 concentration in plasma, directly taken from analytical data. Geometric mean and percentage geometric coefficient of variation (%CV) were reported.

Maximum Observed Concentration of BAY84-3174 in Plasma Divided by Dose (Cmax/D) After First Dose of BAY1067197
Day 1: pre-dose and 0.5, 1, 2, 3, 4, 6, 12 and 24 hours post-dose

Maximum observed drug concentration, directly taken from analytical data, divided by dose. Geometric mean and %CV were reported.

Area Under the Concentration Versus Time Curve of BAY84-3174 for the Dosing Interval (AUCtau) After First Dose of BAY1067197
Day 1: pre-dose and 0.5, 1, 2, 3, 4, 6, 12 and 24 hours post-dose

AUCtau is defined as area under the plasma concentration time profile from time zero to the end of the dosing interval after the first dose and dosing interval was 24 h for both arms. Geometric mean and %CV were reported.

Area Under the Concentration Versus Time Curve of BAY84-3174 for the Dosing Interval Divided by Dose (AUCtau/D) After First Dose of BAY1067197
Day 1: pre-dose and 0.5, 1, 2, 3, 4, 6, 12 and 24 hours post-dose

AUCtau/D is defined as area under the plasma concentration time profile from time zero to the end of the dosing interval divided by dose after the first dose and dosing interval was 24 h for both arms. Geometric mean and %CV were reported.

Maximum Observed Concentration of BAY84-3174 in Plasma (Cmax,md) After Multiple Dose Administration During a Dosing Interval
Day 7: pre dose and 0.5, 1, 2, 3, 4, 6 and 12 hours post dose; Day 8, Day 14, Day 22 and Day 29

Cmax,md is defined as maximum observed drug concentration in plasma after multiple-dose administrations during a dosing interval directly taken from analytical data.Geometric mean and %CV were reported.

Maximum Observed Concentration of BAY84-3174 in Plasma Divided by Dose (Cmax,md/D) After Multiple Dose Administration During a Dosing Interval
Day 7: pre dose and 0.5, 1, 2, 3, 4, 6 and 12 hours post dose; Day 8, Day 14, Day 22 and Day 29

Maximum observed drug concentration, directly taken from analytical data divided by dose after multiple doses. Geometric mean and %CV were reported.

Area Under the Concentration Versus Time Curve of BAY84-3174 During any Dosing Interval (AUCtau,md) After Multiple Dose Administration
Day 7: pre-dose and 0.5, 1, 2, 3, 4, 6, 12 and 24 hours post-dose

AUCtau,md is defined as area under the plasma concentration time profile from time zero during the dosing interval after multiple-dose administrations and dosing interval was 24 h for both arms. Geometric mean and %CV were reported.

Area Under the Concentration Versus Time Curve of BAY84-3174 During any Dosing Interval Divided by Dose (AUCtau,md/D) After Multiple Dose Administration
Day 7: pre-dose and 0.5, 1, 2, 3, 4, 6, 12 and 24 hours post-dose

AUCtau,md/D is defined as area under the plasma concentration time profile from time zero to the end of the dosing interval after multiple dose of administrations divided by dose and dosing interval was 24 h for both arms. Geometric mean and %CV were reported.

Number of patients with occurrence of AV-Block > I°
up to 48 hours

Secondary Endpoints

Changes From Baseline for Wall Motion Score Index at Day (WMSI) as Measured by Cardiac Magnetic Resonance at Day 7
Baseline to day 7
Number of Subjects With Clinically Relevant Changes Observed in Echocardiography Parameters
Baseline, Day 6 and 15
Number of Subjects With Clinically Relevant Changes Observed in Biomarkers
Baseline up to Day 15
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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BAY1067197 (10 mg)ACTIVE_COMPARATOR -
BAY1067197ACTIVE_COMPARATOR -
Placebo (10 mg)PLACEBO_COMPARATOR -
PlaceboPLACEBO_COMPARATOR -
Placebo and BAY1067197EXPERIMENTALPatients will get both treatment 1 and 2

Interventions

NameTypeDescription
BAY1067197 (10 mg)DRUG10 mg BAY1067197 for 7 d treatment once daily as oral application
BAY1067197DRUGThe dose escalation to the second dose step will proceed only if the previous dose step has shown acceptable safety and tolerability 5 mg / or 10 mg / or 20 mg BAY1067197 for 7 d treatment as oral application.
Placebo (10 mg)DRUG10 mg Placebo for 7 d treatment once daily as oral application
PlaceboDRUG5 mg / or 10 mg / or 20 mg Placebo for 7 d treatment once daily as oral application
Placebo (treatment 1)DRUGOral administration of placebo tablets
BAY1067197 (treatment 2)DRUGOral administration of a single dose of 30 mg (3×10 mg Tablet) BAY1067197
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Eligibility Criteria

Age Range18 Years to 75 Years
SexALL
Healthy VolunteersNo
Study Sites6

* Inclusion Criteria: * Clinical diagnosis of chronic systolic heart failure of ischemic or non-ischemic etiology:(New York Heart Association)NYHA class I-III and treatment with standard pharmacological therapy for the treatment of systolic heart failure including β-blocker ≥ 4 weeks prior to random...

Countries:GermanyItalyNetherlandsPoland
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Frequently asked questions about BAY1067197

What is BAY1067197 used for?

BAY1067197 is an investigational small molecule being developed for heart failure. It is being studied in patients with stable heart failure who are on standard therapy including a beta-blocker. The drug is in Phase 2 clinical development and is not yet approved by regulatory authorities.

Who makes BAY1067197?

BAY1067197 is being developed by Bayer AG, a German pharmaceutical company. Bayer's stock is traded on the OTC market under the ticker symbol BAYRY. The company is conducting clinical trials to evaluate the safety and efficacy of this drug in heart failure patients.

What phase is BAY1067197 in?

BAY1067197 is in Phase 2 clinical development. Two Phase 2 trials have been completed, both in heart failure patients. The drug is still investigational and has not received regulatory approval. It is being studied for its safety and potential therapeutic effects in this patient population.

What clinical trials is BAY1067197 in?

BAY1067197 has completed two Phase 2 clinical trials. NCT01945606 assessed safety in stable heart failure patients on standard therapy including a beta-blocker, enrolling 11 participants in the Netherlands. NCT02040233 was a multiple dose study in heart failure, enrolling 31 participants across Germany, Italy, Netherlands, and Poland.

Is BAY1067197 the same as BAY 1067197?

Yes, BAY1067197 and BAY 1067197 refer to the same drug. The compound is identified by the same name in both clinical trial registrations, with the spacing in the name varying. Both trials listed under these names are Phase 2 studies in heart failure patients.