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BAY1000394

Phase 1

Neoplasms | Small molecule | Oncology |Bayer AG|Last Updated: Jun 24, 2019

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials2
Total Enrollment22

FDA Designations

No designations recorded

Clinical trial landscape

BAY1000394 · 2 trials · 1 indication

Phase 1 2
NCT02047890Japanese BAY1000394 Monotherapy Phase I StudyNeoplasms
COMPLETED12 Analytics
NCT01335256Clinical Study to Evaluate Safety and Maximum Tolerated Dose of BAY1000394 Given in a 4 Week on / 2 Week Off Schedule in Subjects With Advanced MalignanciesNeoplasms
COMPLETED10 Analytics
PHASE1COMPLETED
Japanese BAY1000394 Monotherapy Phase I Study
NeoplasmsUnlock trial analytics
PHASE1COMPLETED
Clinical Study to Evaluate Safety and Maximum Tolerated Dose of BAY1000394 Given in a 4 Week on / 2 Week Off Schedule in Subjects With Advanced Malignancies
NeoplasmsUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of participants with adverse events as a measure of safety and tolerability
6 months
Number of participants with abnormal lab parameters based on descriptive statistics
6 months
Maximum observed drug concentration (Cmax) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose). Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Cmax divided by dose per body weight (Cmax,norm) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose). Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Cmax divided by dose (Cmax/D) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose). Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Area under the concentration versus time curve from zero to infinity after single dose (AUC) for BAY1000394 and its metabolite M-1
= Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose)
AUC from time 0 to 12 hours after single dose (AUC(0-12) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8 and 12 hours
AUC divided by dose per body weight (AUCnorm) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose)
AUCnorm from time 0 to 12 hours after single dose (AUC(0-12),norm) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8 and 12 hours
AUC divided by dose (AUC/D) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose)
Time to reach Cmax (tmax) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose). Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Terminal half-life (t½) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 1: 0 (pre dose), 0.5, 1, 2, 4, 6, 8, 12 and 24 hours (Day 2, before morning dose). Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Maximum observed drug concentration after multiple dosing (Cmax,md) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Cmax divided by dose per body weight after multiple dosing (Cmax,norm,md) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Cmax divided by dose (Cmax,md/D) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
AUC from time 0 to 12 hours after multiple dosing (AUC(0-12),md) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
AUCnorm from time 0 to 12 hours after multiple dosing (AUC(0-12),norm,md) for BAY1000394 and its metabolite M-1
Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
AUC from time 0 to 12 hours divided by dose after multiple dosing for BAY1000394 and its metabolite M-1
Cycle 1 / Day 10 : 0 (before morning dose), 0.5, 1, 2, 4, 6, 8 and 12 hours (before evening dose)
Number of subjects with Adverse Events as a measure safety
Up to 3 years or longer if indicated
Maximum tolerated dose: Measured by adverse event profile
Up to 3 years or longer if indicated

Secondary Endpoints

Tumor response
Screening and on Day 21 of even numbered cycle
Biomarkers evaluation measured by Enzyme-linked immunosorbent assay (ELISA)
Up to 3 years or longer if indicated
Tumor Response evaluation measured by Response Evaluation Criteria in Solid Tumors (RECIST 1.1)
Up to 3 years or longer if indicated
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BAY1000394EXPERIMENTALApproximately 12 subjects will be included: 3 to 6 evaluable subjects for each cohort. The cycle length will be 3 weeks (21 days).
Arm 1EXPERIMENTAL -

Interventions

NameTypeDescription
BAY1000394 (2.5mg)DRUGBAY1000934 2.5mg twice a day (bid) in a 3 days on and 4 days off schedule. (Cohort 1)
BAY1000394 (5mg)DRUGBAY1000934 5mg twice a day (bid) in a 3 days on and 4 days off schedule. (Cohort 2)
BAY1000394DRUGBAY1000394 will be administered orally twice a day (bid) in a 4 week on / 2 week off schedule.
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Eligibility Criteria

Age Range20 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites2

Inclusion Criteria: * Japanese male or female subjects aged ≥20 years * Eastern Cooperative Oncology Group (ECOG) performance status of 0 - 1 * Life expectancy of at least 12 weeks * Subjects with advanced, histologically or cytologically confirmed solid tumors, not amenable to any standard therapy...

Countries:JapanUnited States
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Frequently asked questions about BAY1000394

What is BAY1000394 used for?

BAY1000394 is an investigational small molecule being studied for the treatment of neoplasms, which are abnormal growths of tissue that can be benign or malignant. It is being evaluated in oncology clinical trials for patients with advanced malignancies. The drug is currently in Phase 1 clinical development.

Who makes BAY1000394?

BAY1000394 is being developed by Bayer AG, a multinational pharmaceutical company. Bayer's stock is traded over-the-counter under the ticker symbol BAYRY. The company is conducting clinical trials to evaluate the safety and tolerability of this investigational oncology drug.

What phase is BAY1000394 in?

BAY1000394 is in Phase 1 clinical development. Two Phase 1 trials have been completed, but no active trials are currently ongoing. The drug is investigational and has not been approved by regulatory authorities. It remains in early-stage clinical testing for the treatment of neoplasms.

What clinical trials is BAY1000394 in?

BAY1000394 has been studied in two completed Phase 1 clinical trials. NCT01335256 evaluated safety and maximum tolerated dose in subjects with advanced malignancies in the United States. NCT02047890 was a Japanese monotherapy Phase I study. Both trials enrolled a total of 22 participants.

Is BAY1000394 the same as any other drug?

No alternative names for BAY1000394 have been disclosed in the clinical trial information. The drug is identified solely by its code name BAY1000394 in the registered clinical studies. It is an investigational small molecule being developed by Bayer AG for oncology indications.