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INCB057643

Phase 1

Healthy Volunteers | Small molecule | Other |Incyte Corporation|Last Updated: Jun 11, 2025

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment48
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT06941077A Study to Evaluate the Relative Bioavailability of New Formulations of INCB057643 Tablets Administered Orally in Healthy ParticipantsPHASE1 COMPLETED 48May 12, 2025Jun 3, 2025Jun 11, 20251 United States
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Study Endpoints
Primary Endpoints
Pharmacokinetics Parameter (PK): Cmax of INCB057643
Up to Day 10

Defined as maximum observed plasma concentration of INCB057643.

Pharmacokinetics Parameter: AUC(0-last) of INCB057643
Up to Day 10

Defined as area under the single-dose serum concentration-time curve from time = 0 to the last measurable concentration at time of INCB057643.

Pharmacokinetics Parameter: AUC 0-∞ of INCB057643
Up to Day 10

Defined as the area under the single-dose serum concentration-time curve extrapolated to time of infinity of INCB057643.

Secondary Endpoints
Number of participants with Treatment-emergent Adverse Events (TEAEs)
Up to Day 26
Pharmacokinetics Parameter: Tmax of INCB057643
Up to Day 10
Pharmacokinetics Parameter: t1/2 of INCB057643
Up to Day 10
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Cohort 1: Dose Treatment AEXPERIMENTALINCB057643 will be administered at protocol defined dose.
Cohort 2: Dose Treatment BEXPERIMENTALINCB057643 will be administered at protocol defined dose.
Cohort 3: Dose Treatment CEXPERIMENTALINCB057643 will be administered at protocol defined dose.
Cohort 4: Dose Treatment DEXPERIMENTALINCB057643 will be administered at protocol defined dose.
Cohort 4: Dose Treatment EEXPERIMENTALINCB057643 will be administered at protocol defined dose.
Interventions
NameTypeDescription
INCB057643DRUGTablet
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Ability to comprehend and willingness to sign a written ICF for the study. * Aged 18 to 55 years, inclusive, at the time of signing the ICF. * BMI within the range of 18.0 to 30.0 kg/m2 inclusive. Note: Up to 25% of the participants in each cohort may be enrolled with a BMI \>...

Countries:United States
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