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AZD0516

Phase 1

Metastatic Prostate Cancer | Small molecule | Oncology |AstraZeneca PLC|Last Updated: Aug 31, 2026

Success Probability

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment177

FDA Designations

No designations recorded

Clinical trial landscape

AZD0516 · 1 trial · 1 indication

Phase 1 1
NCT07181161Study of AZD0516 as Monotherapy and in Combination in Participants With Metastatic Prostate CancerMetastatic Prostate Cancer
RECRUITING283 Analytics
PHASE1RECRUITING
Study of AZD0516 as Monotherapy and in Combination in Participants With Metastatic Prostate Cancer
Metastatic Prostate CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Module 1 and 2: Parts A and B: Number of participants with Adverse Events (AEs), Serious Adverse Events (SAEs) and Adverse Event of Special Interests (AESIs)
From Day 1 up to approximately 3 years

Part A: To assess the safety and tolerability and to determine the Maximum Tolerated Dose (MTD) and/or Recommended Dose for Expansion (RDE) of AZD0516 as monotherapy and in combination with anti-cancer agents. Part B: To assess the safety and tolerability of AZD0516 as monotherapy and in combination with anti-cancer agents.

Module 1 and 2: Part A: Number of participants with Dose Limiting Toxicities (DLTs)
From Day 1 up to end of DLT period (approximately 21 days)

To assess the safety and tolerability of AZD0516 as monotherapy and in combination with anti-cancer agents.

Module 1: Parts B and C and Module 2: Part B: Percentage of participants with Prostate-Specific Antigen (PSA) 50 response rate
Up to approximately 2 years

The PSA50 response rate is defined as the percentage of participants achieving ≥ 50% decrease in PSA from baseline to the lowest post-baseline PSA result.

Secondary Endpoints

Module 1 and 2: Part A: Percentage of participants with PSA50 response rate
Up to approximately 2 years
Module 1 and 2: Parts A, B and C: Percentage of participants with PSA90 response rate
Up to approximately 2 years
Module 1 and 2: Parts A, B and C: Time to PSA 50 response (TTPSA50)
Up to approximately 2 years
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Arm 1: AZD0516 monotherapyEXPERIMENTALParticipants with mCRPC will receive AZD0516 monotherapy.
Arm 2: AZD0516 + AZD9574EXPERIMENTALParticipants with mCRPC will receive AZD0516 in combination with AZD9574.

Interventions

NameTypeDescription
AZD0516DRUGAZD0516 will be administered via intravenous infusion.
AZD9574DRUGAZD9574 will be administered orally.
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Eligibility Criteria

Age Range18 Years to 130 Years
SexMALE
Healthy VolunteersNo
Study Sites52

Main Inclusion Criteria: * Histologically or cytologically confirmed diagnosis of metastatic adenocarcinoma of the prostate. Focal high grade neuroendocrine features are permitted. * Measurable PSA ≥ 1 μg/L (≥ 1 ng/mL). * Surgically or medically castrated with serum testosterone levels ≤ 50 ng/dL (...

Countries:United StatesBrazilChinaFranceItalyJapanPolandSouth KoreaSpainUnited Kingdom
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Competitive Landscape -Prostate Cancer 254 trials (matched to "Metastatic Prostate Cancer")

Recent Changes (Last 90 Days)

LOWAug 31, 2026NCT07181161Enrollment: 177 → 283
LOWAug 31, 2026NCT07181161Enrollment: 177 → 283
LOWJul 15, 2026NCT07181161lastUpdatePostDate: changed
LOWJul 15, 2026NCT07181161lastUpdatePostDate: changed
LOWJun 12, 2026NCT07181161lastUpdatePostDate: changed
LOWJun 12, 2026NCT07181161lastUpdatePostDate: changed

Frequently asked questions about AZD0516

What is AZD0516 used for in metastatic prostate cancer?

AZD0516 is an investigational small molecule being studied for the treatment of metastatic prostate cancer. It is currently in Phase 1 clinical development as a monotherapy and in combination with other agents. The drug is being evaluated in a clinical trial enrolling male participants aged 18 years and older.

Who makes AZD0516?

AZD0516 is being developed by AstraZeneca PLC, a biopharmaceutical company listed on the stock exchange under the ticker symbol AZN. The company is conducting a Phase 1 clinical trial of AZD0516 in participants with metastatic prostate cancer across multiple countries.

What phase is AZD0516 in?

AZD0516 is in Phase 1 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities. The ongoing Phase 1 trial is actively recruiting participants to evaluate the safety and efficacy of AZD0516 as a monotherapy and in combination for metastatic prostate cancer.

What clinical trials is AZD0516 in?

AZD0516 is being studied in a Phase 1 clinical trial with the identifier NCT07181161. This trial, titled 'Study of AZD0516 as Monotherapy and in Combination in Participants With Metastatic Prostate Cancer,' is currently recruiting participants and has a target enrollment of 283 patients.

Is AZD0516 being tested in a randomized controlled trial?

Yes, the Phase 1 clinical trial of AZD0516 is randomized and controlled. The trial is not double-blind, meaning participants and investigators know which treatment is being administered. The study is designed to evaluate AZD0516 as a monotherapy and in combination with other treatments for metastatic prostate cancer.

Where is the AZD0516 clinical trial being conducted?

The AZD0516 Phase 1 clinical trial is being conducted in multiple countries, including the United States, Brazil, China, France, Italy, Japan, Poland, South Korea, Spain, and the United Kingdom. The trial is actively recruiting male participants aged 18 years and older with metastatic prostate cancer.