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ABT-335 and rosuvastatin

Phase 3

Dyslipidemia | Small molecule | Cardiovascular |AstraZeneca PLC|Last Updated: Oct 3, 2012

Target and mechanism

ModalitySmall molecule

Also known as ABT-335, ABT-335 and rosuvastatin calcium

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials1
Total Enrollment280

FDA Designations

No designations recorded

Clinical trial landscape

ABT-335 and rosuvastatin · 3 trials · 4 indications

Phase 3 2Phase 1 1
NCT0068001730 Week Study of the Combination of ABT-335 and Rosuvastatin Compared to Rosuvastatin Monotherapy for Subjects With Dyslipidemia and Stage 3 Chronic Kidney DiseaseDyslipidemia
COMPLETED280 Analytics
NCT00463606A Multicenter Study Comparing the Safety and Efficacy of ABT-335 and Rosuvastatin Calcium Combination Therapy to Monotherapy in Subjects With DyslipidemiaHypercholesterolemia
COMPLETED760 Analytics
PHASE3COMPLETED
30 Week Study of the Combination of ABT-335 and Rosuvastatin Compared to Rosuvastatin Monotherapy for Subjects With Dyslipidemia and Stage 3 Chronic Kidney Disease
DyslipidemiaUnlock trial analytics
PHASE3COMPLETED
A Multicenter Study Comparing the Safety and Efficacy of ABT-335 and Rosuvastatin Calcium Combination Therapy to Monotherapy in Subjects With Dyslipidemia
HypercholesterolemiaUnlock trial analytics

Study Endpoints

Primary Endpoints

Median Percent Change in Triglycerides From Baseline to Week 8.
Baseline to 8 weeks

Triglycerides were measured in milligrams/deciliter.

Mean Percent Change From Baseline to the Final Visit in High-density Lipoprotein Cholesterol (HDL-C) (Full Analysis Set)
Baseline to 12 Weeks

The mean percent change from baseline to the final visit in High-density lipoprotein cholesterol (HDL-C), with ABT-335 135 mg in combination with rosuvastatin 5 mg versus rosuvastatin 5 mg monotherapy.

Mean Percent Change From Baseline to the Final Visit in Triglycerides (Full Analysis Set)
Baseline to 12 Weeks

The mean percent change from baseline to the final visit in triglycerides, with ABT-335 135 mg in combination with rosuvastatin 5 mg versus rosuvastatin 5 mg monotherapy.

Mean Percent Change From Baseline to the Final Visit in Low-density Lipoprotein Cholesterol (LDL-C) (Full Analysis Set)
Baseline to 12 Weeks

The mean percent change from baseline to the final visit in low-density lipoprotein cholesterol (LDL-C), with ABT-335 135 mg in combination with rosuvastatin 5 mg versus ABT-335 135 mg monotherapy.

Blood concentrations of the active ingredients and metabolites of ABT-335 and rosuvastatin
Days 1, 8, 9, and 10

Secondary Endpoints

Mean Percent Change in High-Density Lipoprotein Cholesterol From Baseline to Week 8.
Baseline to 8 weeks
Mean Percent Change From Baseline to the Final Visit in Non-high-density Lipoprotein Cholesterol (Non-HDL-C), With ABT-335 135 mg in Combination With Rosuvastatin 5 mg Versus ABT-335 135 mg Monotherapy (Full Analysis Set)
Baseline to 12 Weeks
Mean Percent Change From Baseline to the Final Visit in Non-high-density Lipoprotein Cholesterol (Non-HDL-C), With ABT-335 135 mg in Combination With Rosuvastatin 5 mg Versus Rosuvastatin 5 mg Monotherapy (Full Analysis Set)
Baseline to 12 Weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
ABT-335 plus rosuvastatinEXPERIMENTALABT-335 45 mg plus rosuvastatin 5 mg for 8 weeks, then ABT-335 45 mg plus rosuvastatin 10 mg for 8 weeks
RosuvastatinACTIVE_COMPARATORRosuvastatin 5 mg for 8 weeks then rosuvastatin 10 mg for 8 weeks
ABT-335 and Rosuvastatin CalciumEXPERIMENTALABT-335 135mg in combination with rosuvastatin calcium 5mg administered orally, once daily for 12 weeks
ABT-335ACTIVE_COMPARATORABT-335 135mg monotherapy administered orally, once daily for 12 weeks
Rosuvastatin CalciumACTIVE_COMPARATORRosuvastatin calcium 5mg monotherapy administered orally, once daily for 12 weeks
1EXPERIMENTAL -

Interventions

NameTypeDescription
ABT-335 plus rosuvastatinDRUGABT-335 45 mg plus rosuvastatin 5 mg for 8 weeks, then ABT-335 45 mg plus rosuvastatin 10 mg for 8 weeks
RosuvastatinDRUGRosuvastatin 5 mg for 8 weeks then rosuvastatin 10 mg for 8 weeks
ABT-335 and rosuvastatin calciumDRUGABT-335 135 mg in combination with rosuvastatin calcium 5 mg administered orally, once daily for 12 weeks
ABT-335DRUGABT-335 135 mg monotherapy administered orally, once daily for 12 weeks
rosuvastatin calciumDRUGRosuvastatin calcium 5 mg monotherapy administered orally, once daily for 12 weeks
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites114

Inclusion Criteria * Dyslipidemic participants with Chronic Kidney Disease Stage 3 * For entry into the Treatment Phase (Visit 3), the participant satisfied the following laboratory criteria (measured at the Screening Visit\[s\]): * Estimated glomerular filtration rate between 30 and 59 mL/min/1...

Countries:United StatesPuerto Rico
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Frequently asked questions about ABT-335 and rosuvastatin

What is ABT-335 used for?

ABT-335 is an investigational small molecule being developed for cardiovascular conditions including dyslipidemia and hypercholesterolemia. It has been studied in patients with dyslipidemia, including those with renal insufficiency or stage 3 chronic kidney disease. The drug is not approved and remains in clinical development.

Who makes ABT-335?

ABT-335 is being developed by AstraZeneca PLC, a biopharmaceutical company traded on the NASDAQ under the ticker symbol AZN. The company has sponsored clinical trials evaluating the drug for the treatment of dyslipidemia and related cardiovascular conditions.

What phase is ABT-335 in?

ABT-335 is an investigational drug that has completed Phase 1 and Phase 3 clinical trials. It is not FDA approved and remains in clinical development. The most advanced completed studies were Phase 3 trials evaluating the drug in combination with rosuvastatin for dyslipidemia.

What clinical trials is ABT-335 in?

ABT-335 has been studied in three completed clinical trials. NCT00463606 was a Phase 3 study comparing ABT-335 and rosuvastatin combination therapy to monotherapy in 760 subjects with dyslipidemia. NCT00585143 was a Phase 1 pharmacokinetic study in 37 subjects with renal impairment. NCT00680017 was a Phase 3 study in 280 subjects with dyslipidemia and stage 3 chronic kidney disease.

Is ABT-335 the same as a combination therapy with rosuvastatin?

ABT-335 has been studied as a combination therapy with rosuvastatin calcium in clinical trials for dyslipidemia. The trials compared the safety and efficacy of the combination to rosuvastatin monotherapy. ABT-335 itself is the investigational drug being evaluated in these combination regimens.