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400 µg Brimonidine

Phase 2

Macular Degeneration | Small molecule | Ophthalmology |AbbVie Inc.|Last Updated: Aug 21, 2018

Success Probability

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Trial Design

RandomizedDouble-BlindSHAM_CONTROLLED
Total Trials1
Total Enrollment119

FDA Designations

No designations recorded

Clinical trial landscape

400 µg Brimonidine · 3 trials · 3 indications

Phase 2 1Phase 1 2
NCT00658619Safety and Efficacy of Brimonidine Intravitreal Implant in Patients With Geographic Atrophy Due to Age-related Macular Degeneration (AMD)Macular Degeneration
COMPLETED119 Analytics
PHASE2COMPLETED
Safety and Efficacy of Brimonidine Intravitreal Implant in Patients With Geographic Atrophy Due to Age-related Macular Degeneration (AMD)
Macular DegenerationUnlock trial analytics

Study Endpoints

Primary Endpoints

Change From Baseline in Size of Geographic Atrophy Lesion Area in the Study Eye
Baseline, Month 12

Change from baseline in size of geographic atrophy lesion area in the study eye is based on fundus photography as read by an independent Reading Center. Photographs are taken with a specialized microscope with an attached camera to photograph the interior of the eye, including the retina and optic disc. A positive change from baseline indicates an increase in size of geographic atrophy lesion area (worsening; disease progression). Data are reported in disc area where 1 disc area = 1.767 millimeters squared (mm\^2).

Highest Vitreous Humor Level of Brimonidine in the Study Eye
60 Days

The highest level of brimonidine measured in the vitreous humor of the study eye in any patient is reported for each treatment arm. The vitreous humor is the clear gel that fills the space between the lens and the retina of the eye.

Change From Baseline in Best Corrected Visual Acuity (BCVA) in the Study Eye
Baseline, Month 6

BCVA is measured using an eye chart and is reported as the number of letters read correctly (ranging from 0 to 100 letters) in the study eye. The lower the number of letters read correctly on the eye chart, the worse the vision (or visual acuity). A positive change from baseline indicates an improvement and a negative change from baseline indicates a worsening.

Secondary Endpoints

Change From Baseline in Size of Geographic Atrophy Lesion Area in the Study Eye
Baseline, Month 3, Month 6, Month 9, Month 18, Month 24
Change From Baseline in Best Corrected Visual Acuity (BCVA) in the Study Eye
Baseline, 24 Months
Change From Baseline in Contrast Sensitivity in the Study Eye
Baseline, 24 Months
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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
400 µg Brimonidine Tartrate Implant Stage 1OTHERStage 1: 400 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1 and Month 6.
200 µg Brimonidine Tartrate Implant Stage 1OTHERStage 1: 200 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1 and Month 6.
400 µg Brimonidine Tartrate Implant Stage 2OTHERStage 2: 400 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1 and Month 6.
200 µg Brimonidine Tartrate Implant Stage 2OTHERStage 2: 200 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1 and Month 6.
Sham (no implant) Stage 2SHAM_COMPARATORStage 2: sham in both eyes on Day 1 and Month 6.
400 µg Brimonidine Tartrate ImplantEXPERIMENTAL400 µg brimonidine tartrate implant in the study eye on Day 1 (2, 4 or 8 weeks prior to undergoing a pars plana vitrectomy).
200 µg Brimonidine Tartrate ImplantEXPERIMENTAL200 µg brimonidine tartrate implant in the study eye on Day 1 (2, 4 or 8 weeks prior to undergoing a pars plana vitrectomy).
400 µg Brimonidine Tartrate Implant Group BEXPERIMENTAL400 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1.
200 µg Brimonidine Tartrate Implant Group BEXPERIMENTAL200 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1.
100 µg Brimonidine Tartrate Implant Group BEXPERIMENTAL100 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1.
100 µg Brimonidine Tartrate Implant Group AEXPERIMENTAL100 µg brimonidine tartrate implant in the study eye and sham in the fellow eye on Day 1.

Interventions

NameTypeDescription
400 µg Brimonidine Tartrate ImplantDRUG400 µg brimonidine tartrate implant in the study eye on Day 1 and Month 6.
200 µg Brimonidine Tartrate ImplantDRUG200 µg brimonidine tartrate implant in the study eye on Day 1 and Month 6.
Sham (no implant)OTHERSham in one or both eyes on Day 1 and Month 6.
100 µg Brimonidine Tartrate ImplantDRUG100 µg brimonidine tartrate implant in the study eye on Day 1.
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Eligibility Criteria

Age Range50 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites7

Inclusion Criteria: * Geographic atrophy in both eyes due to age-related macular degeneration * Visual acuity between 20/40 to 20/320 Exclusion Criteria: * Known allergy to brimonidine * Uncontrolled systemic disease or infection of the eye * Recent eye surgery or injections in the eye * Female p...

Countries:United StatesAustraliaGermanyItalyPhilippinesPortugalSouth KoreaCzechiaFrance
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Frequently asked questions about 400 µg Brimonidine

What is 400 µg Brimonidine used for?

400 µg Brimonidine is an investigational small molecule being studied for use in ophthalmology, specifically for retinitis pigmentosa, vitrectomy, and macular degeneration. It is delivered as an intravitreal implant. The drug is not approved and remains in clinical development.

Who makes 400 µg Brimonidine?

400 µg Brimonidine is being developed by AbbVie Inc., which trades under the ticker ABBV. The company is conducting clinical trials to evaluate the safety and efficacy of this intravitreal implant in patients with various eye conditions.

What phase is 400 µg Brimonidine in?

400 µg Brimonidine is in Phase 2 clinical development. One Phase 2 trial has been completed, along with two Phase 1 trials. The drug is investigational and has not received FDA approval.

What clinical trials is 400 µg Brimonidine in?

400 µg Brimonidine has been studied in three completed trials. NCT00658619 was a Phase 2 sham-controlled study in 119 patients with geographic atrophy due to age-related macular degeneration. NCT00661479 was a Phase 1 study in 21 patients with retinitis pigmentosa. NCT01229410 was a Phase 1 pharmacokinetic study in 24 patients undergoing vitrectomy.

Is 400 µg Brimonidine the same as Brimonidine?

400 µg Brimonidine is a specific dosage form of the drug brimonidine, delivered as an intravitreal implant. It is being studied for posterior segment eye diseases. The 400 µg dose refers to the amount of brimonidine in the implant.