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Fexofenadine New Formulation

Phase 3

Asthma | Small molecule | Respiratory |Sanofi|Last Updated: Sep 9, 2025

Target and mechanism

Molecular targetHRH1
Target classAntagonist
ModalitySmall molecule
ChEMBLCHEMBL914

Also known as Fexofenadine HCl New Formulation Tablet, Fexofenadine, Comparator = Montelukast, Fexofenadine, fexofenadine HCL (M016455), fexofenadine, Fexofenadine (loratadine if not available)

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindUNCONTROLLED
Total Trials3
Total Enrollment3,200

FDA Designations

No designations recorded

Clinical trial landscape

Fexofenadine New Formulation · 7 trials · 5 indications

Phase 3 5Phase 2 2
NCT05692154A Placebo-controlled Study of 2-day Pre-treatment With Fexofenadine in Seasonal Allergic RhinitisSeasonal Allergic Rhinitis
COMPLETED95 Analytics
NCT01306721Fexofenadine HCL - Pseudoephedrine HCL Combination Versus Allegra in Patients With Seasonal Allergic RhinitisRhinitis Seasonal
COMPLETED520 Analytics
NCT00044811Efficacy and Safety of Fexofenadine in Mild to Moderate Persistent AsthmaAsthma
COMPLETED1,000 Analytics
NCT00044824Efficacy and Safety of Fexofenadine in Mild to Moderate Persistent AsthmaAsthma
COMPLETED1,000 Analytics
NCT00045955Long-Term Safety Performance of Fexofenadine in AsthmaAsthma
COMPLETED1,200 Analytics
PHASE3COMPLETED
A Placebo-controlled Study of 2-day Pre-treatment With Fexofenadine in Seasonal Allergic Rhinitis
Seasonal Allergic RhinitisUnlock trial analytics
PHASE3COMPLETED
Fexofenadine HCL - Pseudoephedrine HCL Combination Versus Allegra in Patients With Seasonal Allergic Rhinitis
Rhinitis SeasonalUnlock trial analytics
PHASE3COMPLETED
Efficacy and Safety of Fexofenadine in Mild to Moderate Persistent Asthma
AsthmaUnlock trial analytics
PHASE3COMPLETED
Efficacy and Safety of Fexofenadine in Mild to Moderate Persistent Asthma
AsthmaUnlock trial analytics
PHASE3COMPLETED
Long-Term Safety Performance of Fexofenadine in Asthma
AsthmaUnlock trial analytics

Study Endpoints

Primary Endpoints

Area Under Curve (AUC) of the Total Nasal Symptoms Score (TNSS-3)
From 0 hour to 6 hours at Day 4

TNSS-3=composite score calculated as sum of rhinorrhea, sneezing, and nasal itching scores (TNSS-3: scale of each symptom is scored from 0 to 3), where 0 indicates no symptoms, a score of 1 for mild symptoms that are easily tolerated, 2 for awareness of symptoms which are bothersome but tolerable and 3 is reserved for severe symptoms that are hard to tolerate and interfere with daily activity. Individual scores were collected in e-diary. AUC of TNSS from time of the first observation to time of the last observation (AUC \[0-6 hr\]) was calculated by using the linear trapezoid method. Trapezoidal rule involves dividing the area into a number of strips of equal width. Then, approximating the area of each strip by the area of the trapezium formed when a chord replaces upper end. Sum of these approximations gives final numerical result of area under the curve. AUC range: Arm A=0.0-43.5; Arm B=2.1-39.9.

Changes in the nasal congestion score based on the patient's symptom diary
over 2 treatment weeks (from baseline to end of treatment)
Change from baseline in Forced expiratory volume FEV1.
Change from baseline in Forced Expiratory Volume FEV1
Safety evaluation
Number of patients with adverse events
4 weeks
The number of clinically significant abnormalities for laboratory findings
4 weeks

Secondary Endpoints

AUC of Total Ocular Symptoms Score (TOSS) (H0-H6 at Day 4)
From 0 hour to 6 hours at Day 4
AUC of Total Nasal Symptoms Score (TNSS-3) (H0-H12 at Day 4)
From 0 hour to 12 hours at Day 4
AUC of Total Ocular Symptoms Score (TOSS) (H0-H12 at Day 4)
From 0 hour to 12 hours at Day 4
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Arm A (active-active)EXPERIMENTALTwo days of pre-treatment with Fexofenadine 180 mg each day in the morning on Day 2 and Day 3, then Fexofenadine180 mg after the pollen challenge on Day 4.
Arm B (placebo-active)EXPERIMENTALTwo days of pre-treatment with tablet of matching placebo each day in the morning on Day 2 and Day 3, then Fexofenadine180 mg after the pollen challenge on Day 4.
FEX 60 mgACTIVE_COMPARATORStudy medications is administered one hour before or two hours after a meal twice a day. Placebo lead-in period: 1 placebo tablet of fexofenadine 60 mg + 2 placebo tablets of fexofenadine 60 mg/pseudoephedrine 60 mg (fixe dose combination) Double-blind treatment period: 1 tablet of fexofenadine 60 mg + 2 placebo tablets of fexofenadine 60 mg /pseudoephedrine 60 mg (fixe dose combination)
FEX 60 mg/PSE 60 mgEXPERIMENTALStudy medications is administered one hour before or two hours after a meal twice a day. Placebo lead-in period: 1 placebo tablet of fexofenadine 60 mg + 2 placebo tablets of fexofenadine 60 mg/pseudoephedrine 60 mg (fixe dose combination Double-blind treatment period: 1 tablet of fexofenadine 60 mg/pseudoephedrine 60 mg (fixe dose combination) + 1 placebo tablet of fexofenadine 60 mg / pseudoephedrine 60 mg (fixe dose combination)
FEX 60 mg/PSE 120 mgEXPERIMENTALStudy medications is administered one hour before or two hours after a meal twice a day. Placebo lead-in period: 1 placebo tablet of fexofenadine 60 mg + 2 placebo tablets of fexofenadine 60 mg/pseudoephedrine 60 mg (fixe dose combination) Double-blind treatment period: 2 tablets of fexofenadine 30 mg/pseudoephedrine 60 mg (fixe dose combination) + 1 placebo tablet of fexofenadine 30 mg
Age 6 months - 2 yearsEXPERIMENTALPatients between 6 months and 2 years old - Type: Experimental
Age 2 - 11 yearsEXPERIMENTALPatients between 2 and 11 years (and under 10.5 kg)
Age 2 - 11 years (and over 10.5 kg)EXPERIMENTALPatients between 2 and 11 years (and over 10.5 kg)

Interventions

NameTypeDescription
FexofenadineDRUGFexofenadine oral tablet
PlaceboDRUGFexofenadine matching placebo oral tablet
fexofenadine HCL (M016455)DRUGPharmaceutical form:tablet Route of administration: oral
pseudoephedrineDRUGPharmaceutical form:tablet Route of administration: oral
fexofenadine HCL matching placeboDRUGPharmaceutical form:tablet Route of administration: oral
pseudoephedrine matching placeboDRUGPharmaceutical form:tablet Route of administration: oral
Fexofenadine, Comparator = MontelukastDRUG -
fexofenadine/Allegra (M016455)DRUGPharmaceutical form:dry syrup formulation to be suspended in water Route of administration: oral
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Eligibility Criteria

Age Range18 Years to 80 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Participants are eligible to be included in the study only if all of the following criteria apply: * Participant is willing to provide written informed consent. * Adult participants (18 to 80 years old) suffering from seasonal allergic rhinitis (SAR) provoked by Ragweed pollen...

Countries:CanadaJapanUnited StatesCosta RicaGuatemalaHungaryMexicoPolandRussia
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