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Olaparib

Phase 1

Ovarian Cancer | Small molecule | Oncology |Novartis AG|Last Updated: Oct 3, 2024

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment70

FDA Designations

No designations recorded

Clinical trial landscape

Olaparib · 1 trial · 2 indications

Phase 1 1
NCT05258747A Crossover Bioequivalence Study of Olaparib Tablets, 150 mg (Lek Pharmaceuticals d.d.) and Lynparza® (Olaparib) Tablets 150 mg (AstraZeneca Pharmaceuticals LP), in Patients With Breast Cancer Gene (BRCA) Mutated Ovarian Cancer, Recurrent Ovarian Cancer or Metastatic Breast CancerOvarian Cancer
COMPLETED70 Analytics
PHASE1COMPLETED
A Crossover Bioequivalence Study of Olaparib Tablets, 150 mg (Lek Pharmaceuticals d.d.) and Lynparza® (Olaparib) Tablets 150 mg (AstraZeneca Pharmaceuticals LP), in Patients With Breast Cancer Gene (BRCA) Mutated Ovarian Cancer, Recurrent Ovarian Cancer or Metastatic Breast Cancer
Ovarian CancerUnlock trial analytics

Study Endpoints

Primary Endpoints

Maximum Plasma Concentration During the Dosing Interval at Steady State (CmaxSS)
Pre-dose (0.00 hr) on day 1,6,7,8,14,15 and 16 and Post-dose on day 8 and day 16

To assess the pharmacokinetics and establish bioequivalence of the Test Product (Olaparib tablets, 150 mg) relative to that of Reference Product (Lynparza® (olaparib) tablets 150 mg) in patients with Breast Cancer Gene (BRCA) mutated ovarian cancer, recurrent ovarian cancer or metastatic breast cancer.

Area Under the Plasma Concentration Versus Time Curve for One Dosing Interval at Steady State (AUC(0-t)ss)
Pre-dose (0.00 hr) on day 1,6,7,8,14,15 and 16 and Post-dose on day 8 and day 16

To assess the pharmacokinetics and establish bioequivalence of the Test Product (Olaparib tablets, 150 mg) relative to that of Reference Product (Lynparza® (olaparib) tablets 150 mg) in patients with BRCA mutated ovarian cancer, recurrent ovarian cancer or metastatic breast cancer.

Secondary Endpoints

Number of Serious Adverse Events
up to Day 24
Number of Adverse Events
up to Day 24
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER

Treatment Arms

ArmTypeDescription
Olaparib tablets, 150 mg, then Lynparza® (olaparib) tablets 150 mgOTHERparticipants will receive 2 x 150 mg Olaparib tablets twice daily for 16 days in a crossover design
Lynparza® (olaparib) tablets 150 mg, then Olaparib tablets, 150 mgOTHERparticipants will receive 2 x 150 mg Olaparib tablets twice daily for 16 days in a crossover design

Interventions

NameTypeDescription
Olaparib tablets, 150 mgDRUGOlaparib tablets, 150 mg of Lek Pharmaceuticals d.d., Slovenia
Lynparza® (olaparib) tablets 150 mgDRUGLynparza® (olaparib) tablets 150 mg Manufactured for: AstraZeneca Pharmaceuticals LP, Wilmington, Delaware (DE).
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Eligibility Criteria

Age Range18 Years to 85 Years
SexFEMALE
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: \- First-Line Maintenance Treatment of BRCA-mutated Advanced Ovarian Cancer maintenance treatment of adult patients with deleterious or suspected deleterious germline or somatic BRCA-mutated advanced epithelial ovarian, fallopian tube or primary peritoneal cancer who are in comp...

Countries:India
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Competitive Landscape -Ovarian Cancer 176 trials

Top 20 of 59 competitors

CompanyTickerTrialsLead PhaseDrugs
Merck & Co., Inc.MRK5PHASE3Pembrolizumab, Paclitaxel, Bevacizumab, Docetaxel
AstraZeneca PLCAZN19PHASE3Olaparib
GSK plc Sponsored ADRGSK4PHASE3Niraparib
Eli Lilly and CompanyLLY8PHASE3Sofetabart Mipitecan, Paclitaxel, Topotecan, Gemcitabine, Pegylated liposomal doxorubicin
AbbVie, Inc.ABBV13PHASE3Mirvetuximab soravtansine plus Bevacizumab, Bevacizumab
Bristol-Myers Squibb CompanyBMY4PHASE3Rucaparib, Nivolumab
Genmab A/S Sponsored ADRGMAB5PHASE3Rina-S, Paclitaxel, Topotecan, Pegylated liposomal doxorubicin, Gemcitabine
Pfizer Inc.PFE4PHASE3Avelumab, Lorlatanib, Talazoparib, Pemetrexed, Axitinib
Corcept Therapeutics Incorporated.CORT2PHASE3Nab-paclitaxel/m^2, Relacorilant once daily
Verastem, Inc.VSTM4PHASE3avutometinib, Defactinib, Pegylated liposomal doxorubicin, Paclitaxel, Letrozole
Zentalis Pharmaceuticals, Inc.ZNTL3PHASE3Azenosertib
Imunon, Inc.IMNN3PHASE3IMNN-001, Paclitaxel, Carboplatin, Olaparib, Niraparib
Incyte CorporationINCY2PHASE3INCB123667
Genelux Corp.GNLX1PHASE3olvimulogene nanivacirepvec, Platinum chemotherapy: carboplatin or cisplatin, Non-platinum chemotherapy: Physician's Choice of gemcitabine, taxane or pegylated liposomal doxorubicin, Bevacizumab
Regeneron Pharmaceuticals, Inc.REGN4PHASE2Ubamatamab, Bevacizumab, Cemiplimab, Fianlimab, PLD
Novartis AG Sponsored ADRNVS4PHASE2Dabrafenib, Trametinib
BeOne Medicines Ltd. Sponsored ADRONC2PHASE3Pamiparib
IQVIA Holdings IncIQV1PHASE3Oregovomab, Paclitaxel, Carboplatin
Xencor, Inc.XNCR3PHASE2vudalimab
Exelixis, Inc.EXEL2PHASE2Cabozantinib
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Frequently asked questions about Olaparib

What is Olaparib used for in Ovarian Cancer?

Olaparib is an investigational small molecule being studied for use in ovarian cancer, specifically in patients with BRCA-mutated ovarian cancer, recurrent ovarian cancer, or metastatic breast cancer. It is currently in Phase 1 clinical development and is not yet approved for any indication.

Who makes Olaparib?

Olaparib is being developed by Novartis AG, which trades under the ticker NVS. The drug is currently in Phase 1 clinical development for ovarian cancer and is not yet approved.

What phase is Olaparib in?

Olaparib is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and the drug is not yet available for commercial use.

What clinical trials is Olaparib in?

Olaparib has one completed clinical trial, NCT05258747, a Phase 1 crossover bioequivalence study of olaparib tablets in patients with BRCA-mutated ovarian cancer, recurrent ovarian cancer, or metastatic breast cancer. The trial enrolled 70 female participants in India.

Is Olaparib the same as Lynparza?

Olaparib is being studied as a generic version of Lynparza (olaparib) tablets. The Phase 1 trial compared olaparib tablets from Lek Pharmaceuticals d.d. with Lynparza tablets from AstraZeneca Pharmaceuticals LP to assess bioequivalence.