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Nintedanib

Phase 1

Idiopathic Pulmonary Fibrosis | Small molecule | Respiratory |GSK plc|Last Updated: Feb 18, 2025

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment50

FDA Designations

No designations recorded

Clinical trial landscape

Nintedanib · 1 trial · 1 indication

Phase 1 1
NCT06625489A Study to Evaluate the Safety, Tolerability and Blood Levels of GSK3915393 Administered to Healthy Participants of Chinese, Japanese and European Ancestry and to Assess Effects of GSK3915393 on NintedanibIdiopathic Pulmonary Fibrosis
COMPLETED50 Analytics
PHASE1COMPLETED
A Study to Evaluate the Safety, Tolerability and Blood Levels of GSK3915393 Administered to Healthy Participants of Chinese, Japanese and European Ancestry and to Assess Effects of GSK3915393 on Nintedanib
Idiopathic Pulmonary FibrosisUnlock trial analytics

Study Endpoints

Primary Endpoints

Part A: Number of Participants with Adverse Events (AEs)
Up to Day 10

An AE is any untoward medical occurrence in a clinical study participant, temporally associated with the use of a study intervention, whether or not considered related to the study intervention.

Part A: Number of Participants with Serious Adverse Events (SAEs)
Up to Day 10

An SAE is defined as any untoward medical occurrence that, at any dose, meets one or more of the criteria: results in death; is life threatening; requires hospitalization or prolongation of existing hospitalization; results in persistent or significant disability/incapacity; is a congenital anomaly/birth defect in the offspring of a study participant; abnormal pregnancy outcome; or is a suspected transmission of any infectious agent via an authorized medicinal product.

Part A: Number of Participants with Clinically Significant Changes in Clinical Laboratory Values
Up to Day 10

Number of participants with clinically significant changes in clinical laboratory values (hematology, clinical chemistry, and routine urinalysis) will be assessed.

Part A: Number of Participants with Clinically Significant Changes in Vital Signs
Up to Day 10

Number of participants with clinically significant changes in Vital signs (temperature, systolic and diastolic blood pressure \[BP\], pulse rate and respiratory rate \[RR\]) will be assessed.

Part A: Number of Participants with Clinically Significant Changes in 12-Lead Electrocardiogram (ECG)
Up to Day 10

Number of participants with clinically significant changes in 12-lead ECG will be assessed.

Part A: Area Under the Plasma Concentration Versus Time Curve From Time Zero To t (AUC [0-t]) of GSK3915393
Up to 36 hours post dose

Blood sample will be collected to evaluate plasma concentration of GSK3915393.

Part A: Area Under the Plasma Concentration Versus Time Curve From Time Zero To Infinity (AUC [0-inf]) of GSK3915393
Up to 36 hours post dose

Blood sample will be collected to evaluate plasma concentration of GSK3915393.

Part A: Maximum Observed Plasma Concentration (Cmax) of GSK3915393
Up to 36 hours post dose

Blood sample will be collected to evaluate plasma concentration of GSK3915393.

Part A: Time to Cmax (Tmax) of GSK3915393
Up to 36 hours post dose

Blood sample will be collected to evaluate time of maximum plasma concentration of GSK3915393.

Part A: Apparent Terminal Half-life (T1/2) of GSK3915393
Up to 36 hours post dose

Blood sample will be collected to evaluate plasma concentration of GSK3915393.

Part B: AUC (0-t) of Nintedanib
Up to 48 hours post dose

Blood sample will be collected to evaluate plasma concentration of Nintedanib.

Part B: AUC (0-inf) of Nintedanib
Up to 48 hours post dose

Blood sample will be collected to evaluate plasma concentration of Nintedanib.

Part B: Cmax of Nintedanib
Up to 48 hours post dose

An AE is any untoward medical occurrence in a clinical study participant, temporally associated with the use of a study intervention, whether or not considered related to the study intervention

Secondary Endpoints

Part B: Number of Participants with AEs
Up to Day 17
Part B: Number of Participants with SAEs
Up to Day 17
Part B: Number of Participants with Clinically Significant Changes in Clinically Laboratory Values
Up to Day 17
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part A: GSK3915393EXPERIMENTALParticipants from Chinese, Japanese, and European ancestries will be randomized to receive GSK3915393 under fasting condition.
Part A: PlaceboPLACEBO_COMPARATORParticipants from Chinese, Japanese, and European ancestries will be randomized to receive placebo under fasting condition.
Part B: Nintedanib followed by Nintedanib plus GSK3915393EXPERIMENTALMale participants will be randomized to receive Nintedanib in Period 1 followed by co-administration of Nintedanib and GSK3915393 in Period 2 under fed conditions. There will be a washout period of minimum 5 days post last dose between Period 1 and Period 2.
Part B: Nintedanib plus GSK3915393 followed by NintedanibEXPERIMENTALMale participants will be randomized to receive co-administration of Nintedanib and GSK3915393 in Period 1 followed by Nintedanib in Period 2 under fed conditions. There will be a washout period of minimum 5 days post last dose between Period 1 and Period 2.

Interventions

NameTypeDescription
Part A: PlaceboDRUGPlacebo will be administered.
NintedanibDRUGNintedanib will be administered.
GSK3915393DRUGGSK3915393 will be administered.
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Eligibility Criteria

Age Range18 Years to 50 Years
SexALL
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: For Part A and Part B: Participants who are generally healthy as determined by medical evaluation based on screening medical history, physical examination, vital signs, electrocardiogram (ECG) assessments, and laboratory tests Body weight at least 50.0 kilograms (kg) (110 pound...

Countries:United States
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Frequently asked questions about Nintedanib

What is Nintedanib used for in Idiopathic Pulmonary Fibrosis?

Nintedanib is a small molecule being studied for Idiopathic Pulmonary Fibrosis (IPF). It is currently in Phase 1 clinical development as an investigational drug. A completed trial evaluated its safety, tolerability, and blood levels when administered to healthy participants of Chinese, Japanese, and European ancestry, with a focus on its effects on IPF.

Who makes Nintedanib?

Nintedanib is being developed by GSK plc, a pharmaceutical company listed on the stock exchange under the ticker symbol GSK. The company is conducting clinical research on this small molecule for the treatment of Idiopathic Pulmonary Fibrosis.

What phase is Nintedanib in?

Nintedanib is in Phase 1 clinical development. It is an investigational drug, not yet approved, and is being studied for Idiopathic Pulmonary Fibrosis. One Phase 1 trial has been completed, involving 50 participants.

What clinical trials is Nintedanib in?

Nintedanib has one completed clinical trial registered under NCT06625489. This Phase 1 study evaluated the safety, tolerability, and blood levels of GSK3915393 when administered to healthy participants of Chinese, Japanese, and European ancestry, and assessed its effects on Nintedanib. The trial was conducted in the United States.

Is Nintedanib the same as GSK3915393?

Nintedanib is the drug being studied, while GSK3915393 appears to be a related compound investigated in the same clinical trial. The completed Phase 1 study (NCT06625489) evaluated the safety, tolerability, and blood levels of GSK3915393 and assessed its effects on Nintedanib in healthy participants.