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GW870086X

Phase 2

Asthma | Small molecule | Respiratory |GSK plc|Last Updated: Feb 20, 2018

Success Probability

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Trial Design

RandomizedDouble-BlindCONTROLLED
Total Trials5
Total Enrollment129

FDA Designations

No designations recorded

Clinical trial landscape

GW870086X · 5 trials · 1 indication

Phase 2 2Phase 1 3
NCT00945932A Study to Evaluate the Effect of Repeat Doses of GW870086X in Mild to Moderate AsthmaticsAsthma
COMPLETED37 Analytics
NCT00857857A Study to Evaluate the Effect of GW870086X on Allergen Challenge in Mild AsthmaticsAsthma
COMPLETED24 Analytics
PHASE2COMPLETED
A Study to Evaluate the Effect of Repeat Doses of GW870086X in Mild to Moderate Asthmatics
AsthmaUnlock trial analytics
PHASE2COMPLETED
A Study to Evaluate the Effect of GW870086X on Allergen Challenge in Mild Asthmatics
AsthmaUnlock trial analytics

Study Endpoints

Primary Endpoints

Lung function as measured by FEV1
Day 28
Late Asthmatic Response (LAR): Minimum FEV1 Between 4-10 Hours After Allergen Challenge on Day 13 of Each Treatment Period
4-10 hours after allergen challenge on Day 13 of each treatment period

Analyzed using a mixed effects model including covariates for participant level Baseline FEV1 and period level Baseline FEV1. Participant level Baseline defined as the mean of Day 1 pre-dose values across periods for each participant and period level Baseline as the difference between the Day 1 pre-dose value and participant level Baseline for each period. Absolute change from saline Baseline was calculated for each participant and time point as value equal to highest challenge value minus highest saline value. Minimum FEV1 over 4-10 hours post allergen challenge was minimum value of all the post-saline time points between 4 to 10 hours (4, 4.5, 5, 5.5, 6, 6.5, 7, 7.5, 8, 8.5, 9, 9.5 and 10 hours). The adjusted mean is presented as least square mean (LSM).

Plasma concentrations of GW870086X and GW870086X pharmacokinetic parameters (including AUC, Cmax, t1/2 and tmax)
3 months
Effect of GW870086X on cortisol levels (naturally produced steroid hormone) in the body during a single dose and after 3 days of dosing
3 days
Change in lung function 2 hours after treatment on day 7
on day 7

Secondary Endpoints

Lung function as measured by FEV1
Day 7 and 14
Lung function as measured by PEFR
Twice daily over 28 days
Rescue medication usage
4-5 months
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
28 day repeat doseEXPERIMENTAL -
13 day repeat doseEXPERIMENTAL -
Treatment Period 1EXPERIMENTAL5mg of GW870086X or placebo will be given once daily for 14 days.
Treatment Period 2EXPERIMENTALGW870086X (5mg or 8.75mg) or placebo will be given once daily for 14 days. In a randomised dose escalating manor following on from treatment period 1.
Treatment Period 3EXPERIMENTAL8.75mg of GW870086X or placebo will be given once daily for 14 days.
GW870086XOTHER -
Cohort 1: Part AEXPERIMENTALSubjects in Cohort 1 will be randomized to receive 0.5, 2 and 6 mg GW870086X and placebo.
Cohort 2: Part AEXPERIMENTALSubjects in Cohort 2 will be randomized to receive 3 mg GW870086X or placebo.
Part BEXPERIMENTALSubjects will be randomized to receive 1 and 3 mg of GW870086X or placebo.

Interventions

NameTypeDescription
GW870086XDRUGInvestigational product
PlaceboDRUGPlacebo control
FPDRUGPositive control
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersNo
Study Sites8

Inclusion Criteria: * Male or female between 18 and 65 years of age inclusive, at the time of signing the informed consent. * A female subject is eligible to participate if she is of: Non-childbearing potential defined as pre-menopausal females with a documented tubal ligation or hysterectomy; or p...

Countries:GermanyAustraliaUnited Kingdom
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Frequently asked questions about GW870086X

What is GW870086X used for?

GW870086X is an investigational small molecule being developed for the treatment of asthma. It is administered by inhalation and has been studied in patients with mild to moderate asthma as well as in healthy volunteers. The drug is still in clinical development and has not been approved by regulatory authorities.

Who makes GW870086X?

GW870086X is being developed by GSK plc, a global biopharmaceutical company listed on the stock exchange under the ticker GSK. The company has conducted multiple clinical trials to evaluate the drug's safety, tolerability, and effects on lung function in asthmatic patients.

What phase is GW870086X in?

GW870086X is in Phase 2 clinical development for asthma. The drug has completed five clinical trials, including Phase 1 and Phase 2 studies, with a total enrollment of 129 participants. All trials have been completed, and the drug remains investigational.

What clinical trials is GW870086X in?

GW870086X has been studied in several completed clinical trials, including NCT00483899, NCT00549497, NCT00945932, and NCT01160003. These trials evaluated the drug's effects on lung function, steroid hormone levels, pharmacokinetics, safety, and tolerability in healthy volunteers and patients with asthma.

How does GW870086X work?

GW870086X is a small molecule administered by inhalation for the treatment of asthma. The specific molecular target of the drug has not been disclosed in the available clinical trial information. The drug is being studied for its effects on lung function and safety in asthmatic patients.