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BIIB014

Phase 1

Healthy | Small molecule | Other |Biogen Inc.|Last Updated: Aug 23, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials3
Total Enrollment84
FDA Designations
No designations recorded
Clinical Trials (3)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01035515BIIB014 Cardiovascular Monitoring StudyPHASE1 COMPLETED 24Dec 1, 2009Apr 1, 2010Jun 22, 20101 United States
NCT01017666BIIB014 Effects on the Pharmacokinetics (PK) of Rosiglitazone, Warfarin, and MidazolamPHASE1 COMPLETED 28Nov 1, 2009Jun 2, 2010Aug 23, 20231 United Kingdom
NCT00531193Using PET Scans to Study Brain Receptor Occupancy of BIIB014 in Healthy Male VolunteersPHASE1 COMPLETED 32Sep 1, 2007Apr 1, 2008Jul 30, 20081 United Kingdom
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Study Endpoints
Primary Endpoints
Supine Blood pressure
24 hours
Pharmacokinetic profile of rosiglitazone (Cohort 1), midazolam & metabolites and s-warfarin (Cohort 2) during steady state exposure to BIIB014 or placebo
24 hours (Cohort 1); 144 hours (Cohort 2)
PET scanning with [11C]SCH442416 of the putamen, caudate, nucleus accumbens, thalamus, and cerebellum.
pre-dose and 24h following last dose
Secondary Endpoints
Adverse Events
Duration of subject participation
Concentrations of BIIB014 and its N-acetyl metabolite will be measured in blood plasma
up to 24h following last dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
Treatment Arms
ArmTypeDescription
Arm OneEXPERIMENTALArm 1 of 6 cross-over arms
Arm TwoEXPERIMENTALArm 2 of 6 cross-over arms
Arm ThreeEXPERIMENTALArm 3 of 6 cross-over arms
Arm FourEXPERIMENTALArm 4 of 6 cross-over arms
Arm FiveEXPERIMENTALArm 5 of 6 cross-over arms
Arm SixEXPERIMENTALArm 1 of 6 cross-over arms
Rosiglitazone 8mg POEXPERIMENTALCohort 1
Midazolam 2mg PO, Warfarin 25mg POEXPERIMENTALCohort 2
1OTHERVarious protocol-specified doses of BIIB014 will be used (doses to be determined by PET scan results)
Interventions
NameTypeDescription
PlaceboDRUGSingle dose oral capsule placebo comparator
BIIB014 50mgDRUGSingle dose oral capsule 50mg BIIB014
BIIB014 100mgDRUGSingle dose oral capsule 100mg BIIB014
BIIB014DRUGBIIB014 100mg PO Cohort 1 - 8d Cohort 2 - 14d
[11C]SCH442416OTHER11C\]SCH442416 is a radiolabelled tracer molecule that specifically binds to adenosine A2A sites and will be used to evaluate receptor occupancy. The target activity will be 370 MBq. \[11C\]SCH442416 will be administered IV as a bolus injection over 30 seconds following the start of each PET scan.
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Eligibility Criteria
Age Range18 Years — 50 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male or female subjects * Between the ages of 18 and 50, inclusive. * Must have a body mass index (BMI) between 19 kg/m2 and 30 kg/m2, inclusive Exclusion Criteria: * Clinically significant abnormalities (as determined by the Investigator) * Other unspecified reason ...

Countries:United StatesUnited Kingdom
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