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Ciclesonide/Formoterol Combination

Phase 3

Asthma | Small molecule | Respiratory |AstraZeneca PLC|Last Updated: Apr 26, 2017

Success Probability

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials19
Total Enrollment6,995

FDA Designations

No designations recorded

Clinical trial landscape

Ciclesonide/Formoterol Combination · 19 trials · 1 indication

Phase 3 18Phase 2 1
NCT00392288Efficacy and Safety of Ciclesonide (CIC) Administered Twice Daily in Pediatric Patients With Asthma.Asthma
COMPLETED528 Analytics
NCT00384189A Comparative Study of Inhaled Ciclesonide Versus Placebo in Children (6-11 Years) With AsthmaAsthma
COMPLETED1,080 Analytics
NCT00306163Responsiveness of Lower Airways in Adult Patients (18-60 Years) With Stable Asthma After Treatment With Ciclesonide and Fluticasone Propionate (BY9010/NL-101)Asthma
COMPLETED37 Analytics
NCT00305461Effect of Ciclesonide on Quality of Life in Patients With Moderate Persistent Asthma (21 to 65 y) (BY9010/AR-101)Asthma
COMPLETED101 Analytics
NCT00163449Efficacy and Safety of Ciclesonide in Preschool Children With Asthma (2 to 6 Years) (BY9010/M1-207)Asthma
COMPLETED1,000 Analytics
NCT00163371Effects of Inhaled Ciclesonide Versus Fluticasone Propionate Versus Placebo on Lower Leg Growth in Prepubertal Children With Mild Persistent Asthma (6 to 12 y) (BY9010/M1-208)Asthma
COMPLETED28 Analytics
NCT00163436Efficacy and Safety of Ciclesonide Administered With or Without Different Spacers in Patients With Asthma (12 to 75 y) (BY9010/M1-145)Asthma
COMPLETED450 Analytics
NCT00163293Efficacy of Ciclesonide Inhaled Once Daily Versus Other Corticosteroids Used for Treatment of Mild Asthma in Children (4 to 11 Years) (BY9010/CA-101)Asthma
COMPLETED240 Analytics
NCT00163319Efficacy of Ciclesonide and Fluticasone Propionate in Adult Patients With Moderate and Severe Persistent Asthma (18 to 75 y) (BY9010/IT-101)Asthma
COMPLETED500 Analytics
NCT00163423Efficacy of Ciclesonide Versus Fluticasone Propionate in Patients With Mild to Moderate Asthma (12 to 75 y) (BY9010/M1-142)Asthma
COMPLETED480 Analytics
PHASE3COMPLETED
Efficacy and Safety of Ciclesonide (CIC) Administered Twice Daily in Pediatric Patients With Asthma.
AsthmaUnlock trial analytics
PHASE3COMPLETED
A Comparative Study of Inhaled Ciclesonide Versus Placebo in Children (6-11 Years) With Asthma
AsthmaUnlock trial analytics
PHASE3COMPLETED
Responsiveness of Lower Airways in Adult Patients (18-60 Years) With Stable Asthma After Treatment With Ciclesonide and Fluticasone Propionate (BY9010/NL-101)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Effect of Ciclesonide on Quality of Life in Patients With Moderate Persistent Asthma (21 to 65 y) (BY9010/AR-101)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Efficacy and Safety of Ciclesonide in Preschool Children With Asthma (2 to 6 Years) (BY9010/M1-207)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Effects of Inhaled Ciclesonide Versus Fluticasone Propionate Versus Placebo on Lower Leg Growth in Prepubertal Children With Mild Persistent Asthma (6 to 12 y) (BY9010/M1-208)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Efficacy and Safety of Ciclesonide Administered With or Without Different Spacers in Patients With Asthma (12 to 75 y) (BY9010/M1-145)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Efficacy of Ciclesonide Inhaled Once Daily Versus Other Corticosteroids Used for Treatment of Mild Asthma in Children (4 to 11 Years) (BY9010/CA-101)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Efficacy of Ciclesonide and Fluticasone Propionate in Adult Patients With Moderate and Severe Persistent Asthma (18 to 75 y) (BY9010/IT-101)
AsthmaUnlock trial analytics
PHASE3COMPLETED
Efficacy of Ciclesonide Versus Fluticasone Propionate in Patients With Mild to Moderate Asthma (12 to 75 y) (BY9010/M1-142)
AsthmaUnlock trial analytics

Study Endpoints

Primary Endpoints

Change From Baseline in Forced Expiratory Volume in One Second (FEV1) at Week 12.
Baseline and Week 12

Change in FEV1 (Percent of predicted) from baseline to week 12. FEV1 was measured only in children between 6 to \<12 years only. Least Squares Mean were adjusted for Baseline FEV1, age \[yrs\], pooled center, previous corticosteroid therapy and holding chamber.

Change From Baseline in Morning Peak Expiratory Flow (PEF)
Baseline and Week 12

PEF is the maximum speed of expiration. A portable electronic PEF meter was used for the home PEF readings. The patients recorded PEF daily, in the morning immediately after getting up. Readings were done preferably at least 4 hours after use of rescue medication and before inhalation of the study medication. At each measurement, three readings were obtained in the standing position. All three values were recorded in the diary; the highest value was used for evaluation. The higher change from Baseline values are the best. Analysis of covariance (ANCOVA) model with the baseline value and age as covariates was used for analysis. Last observation carried forward.

PC20 AMP (Post-treatment Compared to Baseline)
Baseline and 5 weeks

Mean change of Provocative concentration of Adenosine-5'-monophosphate (PC20 AMP) leading to a 20 percent decrease in Forced expiratory volume in one second (FEV1) between post-treatment and baseline using two different particle sizes. - Small particles = Mass mean aerodynamic diameter (MMAD) of approximately 1.04-1.08 micron - Large particles = MMAD of approximately 9.9-10.6 micron

differences in Quality of Life from AQLQ(S) (T end versus T0)
8 weeks
time to first exacerbation
8 weeks
differences in FEV1 and FVC from spirometry (T end vs T0).
8 weeks
time to first moderate or severe asthma exacerbation.
24 weeks
growth velocity of the right lower leg as measured by knemometry.
FEV1.
Time to First Asthma Exacerbation
Up to 12 months

Time to first asthma exacerbation is defined as the time in days until the first asthma exacerbation, or to the end of treatment visit. In the absence of an exacerbation, an early treatment discontinuation is treated as a censored observation on the day following the last use of study drug.

Exacerbations (Post-hoc Analysis of Annual Rates)
Up to 12 months

A model-based analysis of asthma exacerbation was performed to adjust to important covariables. The distribution of the data suggested a Poisson regression modeling (zero inflated) strategy. After a variable selection process considering also variable-by-treatment interactions, the variables centre, age \[years\] and race were identified to be important beside treatment. The parameters centre and age \[years\] were allocated to zero-model part and the variables treatment and race to the Poisson model part. The estimates of the per-treatment rates are based on a negative-binomial distribution.

number of patients with candidiasis of the oropharynx or hoarseness.
FEV1
time to the first asthma exacerbation.
FEV1 absolute values
PD20FEV1 from methacholine challenge.
FEV1 absolute values.
time until the first severe asthma exacerbation occurs
number of poorly controlled asthma days.
variables of primary interest are FVC% at PC20 MCh, SVC% at PC20 MCh
FVC% at PC20 AMP, SVC% at PC20 AMP
regional air trapping
bronchial and alveolar exhaled NO
lung function variables
non-cellular inflammatory markers.
AUC(0-24h)/24 h of serum cortisol level
24 h urinary cortisol excretion adjusted for creatinine.
PC20FEV1 (AMP)
Time to the first experience of lack of efficacy
AUC (FEV1) over a 24 h dosing interval.

Secondary Endpoints

Change From Baseline in Total Daily Asthma Symptom Score at Week 12.
Baseline and Week 12
Change From Baseline in Use of Albuterol/Salbutamol at Week 12.
Baseline and Week 12
Time to First Event of Lack of Efficacy (LOE) by Week 12
12 weeks
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Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Placebo MDIPLACEBO_COMPARATORdouble-blind
Ciclesonide MDI 40 µg BIDEXPERIMENTALdouble-blind
Ciclesonide MDI 80 µg BIDEXPERIMENTALdouble-blind
Ciclesonide 40 µgACTIVE_COMPARATORPlacebo-matching ciclesonide, inhaled via a metered-dose inhaler (MDI) with 1,1,1,2-hydrofluoroalkane (HFA)-134a as propellant, once daily, in the evening for 2 to 4 weeks in the Baseline period followed by ciclesonide 40 µg, inhaled via a MDI with HFA-134a as propellant, once daily in the evening for 12 weeks. Salbutamol 100 μg/puff was available to be used as rescue medication if needed.
Ciclesonide 80 µgACTIVE_COMPARATORPlacebo-matching ciclesonide, inhaled via a MDI with HFA-134a as propellant, once daily, in the evening for 2 to 4 weeks in the Baseline period followed by ciclesonide 80 µg, inhaled via a MDI with HFA-134a as propellant, once daily in the evening for 12 weeks. Salbutamol 100 μg/puff was available to be used as rescue medication if needed.
Ciclesonide 160 µgACTIVE_COMPARATORPlacebo-matching ciclesonide, inhaled via a MDI with HFA-134a as propellant, once daily, in the evening for 2 to 4 weeks in the Baseline period followed by ciclesonide 160 µg, inhaled via a MDI with HFA-134a as propellant, once daily in the evening for 12 weeks. Salbutamol 100 μg/puff was available to be used as rescue medication if needed.
PlaceboPLACEBO_COMPARATORPlacebo-matching Ciclesonide, inhaled via a MDI with HFA-134a as propellant, once daily in the evening for 2 to 4 week in the Baseline period followed by placebo-matching ciclesonide, inhaled via a MDI with HFA-134a as propellant, once daily in the evening for 12 weeks. Salbutamol 100 μg/puff was available to be used as rescue medication if needed.
1ACTIVE_COMPARATORCiclesonide 160 µg
2ACTIVE_COMPARATORFluticasone 100 µg
3ACTIVE_COMPARATORCiclesonide 160 µg
4PLACEBO_COMPARATORPlacebo
Ciclesonide 100 µgACTIVE_COMPARATORCiclesonide 100 µg, metered-dose inhaler, two puffs once daily, in the evening, for up to 12 months.
Ciclesonide 200 µgACTIVE_COMPARATORCiclesonide 200 µg, metered-dose inhaler, two puffs once daily, in the evening, for up to 12 months.

Interventions

NameTypeDescription
CiclesonideDRUGCiclesonide MDI 40 µg BID over twelve weeks
PlaceboDRUGPlacebo MDI over twelve weeks
SalbutamolDRUGSalbutamol inhalation powder
FluticasoneDRUGinhaled Fluticasone 100 µg, twice daily
Ciclesonide/Formoterol CombinationDRUG -
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Eligibility Criteria

Age Range4 Years to 11 Years
SexALL
Healthy VolunteersNo
Study Sites6

Inclusion Criteria: * History of persistent bronchial asthma for at least 3 months prior to screening; * For patients with persistent bronchial asthma and being treated with a controller therapy: Documented use of an inhaled steroid or Singulair® 5mg once daily; * For patients with persistent bronc...

Countries:United StatesHungaryMexicoPolandRussiaSouth AfricaBulgariaGermanyRomaniaSpainUkraineNetherlandsArgentinaBrazilIndiaSwitzerlandDenmarkCanadaFranceItalyBelgiumUnited KingdomAustriaPortugalMalaysiaTaiwanSouth KoreaAustraliaCzechia
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Frequently asked questions about Ciclesonide/Formoterol Combination

What is Ciclesonide used for?

Ciclesonide is an investigational small molecule in Phase 3 development for asthma, bronchial asthma, rhinitis, allergic, seasonal, seasonal allergic rhinitis, hay fever, and perennial allergic rhinitis. It is being studied in the respiratory therapeutic area. The drug has been evaluated in 19 completed clinical trials with a total enrollment of 6,995 participants.

Who makes Ciclesonide?

Ciclesonide is being developed by AstraZeneca PLC, which trades under the ticker AZN. The company is conducting clinical research on this respiratory drug candidate for asthma and allergic rhinitis indications. AstraZeneca has completed 19 trials involving the drug, with all trials now closed.

What phase is Ciclesonide in?

Ciclesonide is in Phase 3 clinical development for respiratory conditions including asthma and allergic rhinitis. It is an investigational drug and has not been reported as FDA approved. All 19 clinical trials listed for Ciclesonide are completed, with no active trials currently enrolling patients.

What clinical trials is Ciclesonide in?

Ciclesonide has completed 19 clinical trials, including NCT00163345, NCT00163397, NCT00306163, and NCT00314509. These Phase 3 and Phase 2 studies evaluated the drug in asthma patients across countries such as the Netherlands, Malaysia, Taiwan, France, Germany, Hungary, and South Africa. The trials were randomized, double-blind, and active-controlled.

Is Ciclesonide the same as Alvesco?

Ciclesonide is the generic name for the drug also known by the brand name Alvesco. The data provided does not list alternative names, so this relationship is not confirmed in the available information. Ciclesonide is being studied for asthma and allergic rhinitis indications.