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AZD5069

Phase 1

Healthy | Small molecule | Other |AstraZeneca PLC|Last Updated: Jun 25, 2015

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials4
Total Enrollment280
FDA Designations
No designations recorded
Clinical Trials (4)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01332903Open Label, Healthy Volunteers, ADME Study With Single Oral Administration of [14C] AZD5069PHASE1 COMPLETED 6May 1, 2011Jul 1, 2011Jun 25, 20151 United Kingdom
NCT01100047Japanese Single and Multiple Ascending Dose (JSMAD), Safety, Tolerability, Pharmacokinetics (PK) and Pharmacodynamics (PD) Study of AZD5069PHASE1 COMPLETED 63May 1, 2010Feb 1, 2011Jun 25, 20151 United Kingdom
NCT01051505A Study to Assess the Safety, Tolerability, Pharmacokinetics (PK) and Pharmacodynamics (PD) of Multiple Ascending Doses of AZD5069 in Healthy VolunteersPHASE1 COMPLETED 8Jan 1, 2010Apr 1, 2010Jun 25, 20151 United Kingdom
NCT00953888Study to Investigate the Safety, Tolerability and Activity of AZD5069 When Given as a Single Dose to Healthy Male and/or Female SubjectsPHASE1 COMPLETED 203Jul 1, 2009Dec 1, 2009Jun 25, 20151 United Kingdom
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Study Endpoints
Primary Endpoints
To investigate the absorption, distribution, metabolism and excretion of AZD5069 in human subjects by measuring the amount of [14C] radioactivity in plasma and whole blood
From pre-dose until 168 hours post last dose

To investigate the absorption, distribution, metabolism and excretion of AZD5069 in human subjects by measuring the amount of \[14C\] radioactivity in plasma and whole blood and the resulting area under the concentration-time curve from zero extrapolated to infinity (AUC), to the last measurable concentration (AUC(0 t)).

To investigate the absorption, distribution, metabolism and excretion of AZD5069 in human subjects by measuring Plasma [14C] AZD5069:AZD5069 (cold) ratios for concentrations and selected pharmacokinetic parameters (AUCs and Cmax).
From pre-dose until 168hours post last dose
To investigate the excretion of AZD5069 in human subjects by measuring the amount and percentage of radioactive dose recovered in urine, faeces, and renal clearance.
From pre-dose until 168hours post last dose
Adverse events, electrocardiograms (ECGs), laboratory variables, blood pressure, pulse rate, body temperature, QT interval and continuous cardiac monitoring using telemetry
From screening period to follow-up visit 42 days (Maximum)
Safety and tolerability of AZD5069 assessing vitals signs (blood pressure, pulse rate,body temperature), ECG,laboratory variables (including high sensitivity C-reactive protein, circulating neutrophils), continuous cardiac monitoring using telemetry.
Baselines assessments at Visit 1 (enrolment). Assessments pre-dose at Visit 2 and at protocol defined time-points post-dose. Follow up assessments at Visit 3.
Secondary Endpoints
To investigate the safety and tolerability of AZD5069 given orally
From screening visit, Day 12, up to follow up visit
Assessment of ex vivo GROa stimulated CD11b expression on neutrophils in whole blood
Samples collected at Visit 2 from pre-dose and at regular protocol defined intervals up to 96 hours post-dose
Measurement of the effect of AZD5069 on blood cells
Samples collected at Visit 2 from pre-dose and at regular protocol defined intervals up to 96 hours post-dose
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Study Design & Arms
AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
1EXPERIMENTAL\[14C\] AZD5069
2PLACEBO_COMPARATOR -
ActiveEXPERIMENTALAZD5069 oral solution
PlaceboPLACEBO_COMPARATORPlacebo oral solution
Interventions
NameTypeDescription
[14C] AZD5069DRUGSingle 120 mg oral dose administered on Day 1
AZD5069DRUGOral suspension
PlaceboDRUGOral suspension
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Eligibility Criteria
Age Range50 Years — N/A
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Have a body mass index (BMI) of ≥18 and ≤30 kg/m2 and weight of ≥50 kg and ≤100 kg. * Regular daily bowel movements (ie, production of at least 1 stool per day). * Non-smoker or ex-smoker who has not used tobacco or nicotine products for ≥6 months prior to Visit 1 * Healthy Ma...

Countries:United Kingdom
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