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Nebivolol 1 Percent

Phase 2

Open-Angle Glaucoma | Small molecule | Ophthalmology |Summit Therapeutics Inc.|Last Updated: Apr 17, 2024

Success Probability

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials1
Total Enrollment226

FDA Designations

No designations recorded

Clinical trial landscape

Nebivolol 1 Percent · 1 trial · 2 indications

Phase 2 1
NCT04910100Nebivolol 0.5, 1.0, or Timolol 0.5 Suspension Compared to Timolol 0.5 Solution to Treat Glaucoma/Ocular HypertensionOpen-Angle Glaucoma
COMPLETED226 Analytics
PHASE2COMPLETED
Nebivolol 0.5, 1.0, or Timolol 0.5 Suspension Compared to Timolol 0.5 Solution to Treat Glaucoma/Ocular Hypertension
Open-Angle GlaucomaUnlock trial analytics

Study Endpoints

Primary Endpoints

Intraocular Pressure Over 84 Days
Over 84 days

Measured utilizing a calibrated Goldmann tonometer; two consecutive IOP measurements of each eye will be performed. If the 2 measurements differ by more than 2 mm Hg, a third measurement will be taken. The primary efficacy analysis will be the between-group comparison of the mean IOP values in the study eye at 10AM, 2 hours postdose, and 4PM, at each of the Visit 4/Day 15, Visit 5/Day 42, and Visit 6/Day 84 visits (ie, a total of 9 between-group comparisons). A hierarchical analysis will be conducted to compare each of the investigational products against the comparator, timolol 0.5% ophthalmic solution, as follows: (1) nebivolol 1% ophthalmic suspension, (2) nebivolol 0.5% ophthalmic suspension, and (3) timolol ophthalmic suspension.

Secondary Endpoints

Intraocular Pressure: Change From Baseline in Diurnal IOP at Each Visit
Day 15: 8 AM ± 30 minutes, 2 hours post-dose ± 30 minutes, 4 PM ± 30 minutes; Day 42: 8 AM ± 30 minutes, 2 hours post-dose ± 30 minutes, 4 PM ± 30 minutes; Day 84: 8 AM ± 30 minutes, 2 hours post-dose ± 30 minutes, 4 PM ± 30 minutes
Intraocular Pressure: Change From Baseline at All Time Points at Each Visit
Day 15: 8 AM ± 30 minutes, 2 hours post-dose ± 30 minutes, 4 PM ± 30 minutes; Day 42: 8 AM ± 30 minutes, 2 hours post-dose ± 30 minutes, 4 PM ± 30 minutes; Day 84: 8 AM ± 30 minutes, 2 hours post-dose ± 30 minutes, 4 PM ± 30 minutes
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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Nebivolol Ophthalmic Suspension 1 PercentEXPERIMENTALAdministered twice daily to both eyes for 84 days (12 weeks)
Nebivolol Ophthalmic Suspension 0.5 PercentEXPERIMENTALAdministered twice daily to both eyes for 84 days (12 weeks)
Timolol Ophthalmic Suspension 0.5 PercentEXPERIMENTALAdministered twice daily to both eyes for 84 days (12 weeks)
Timolol Ophthalmic Solution 0.5 PercentACTIVE_COMPARATORAdministered twice daily to both eyes for 84 days (12 weeks)

Interventions

NameTypeDescription
Nebivolol Ophthalmic Suspension 1 PercentDRUG1 drop instilled into each eye twice daily
Nebivolol Ophthalmic Suspension 0.5 PercentDRUG1 drop instilled into each eye twice daily
Timolol Ophthalmic Suspension 0.5 PercentDRUG1 drop instilled into each eye twice daily
Timolol Ophthalmic Solution 0.5 PercentDRUG1 drop instilled into each eye twice daily
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Eligibility Criteria

Age Range18 Years to 100 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. Willing and able to understand and sign an informed consent form prior to any study related procedures. 2. Able to administer or have a caregiver accurately administer an eye drop. 3. Have POAG or OHT in both eyes that requires therapy for IOP and is adequately controlled, in...

Countries:United States
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Competitive Landscape -Open-Angle Glaucoma 9 trials

Frequently asked questions about Nebivolol 1 Percent

What is Nebivolol 1 Percent used for?

Nebivolol 1 Percent is an investigational small molecule being developed for the treatment of open-angle glaucoma and ocular hypertension. It is a topical ophthalmic formulation intended to lower intraocular pressure in patients with these conditions. The drug is currently in Phase 2 clinical development.

What does Nebivolol 1 Percent target?

Nebivolol 1 Percent is a beta-blocker, a class of drugs that works by blocking beta-adrenergic receptors. In the eye, this reduces the production of aqueous humor, thereby lowering intraocular pressure. This mechanism is relevant for treating open-angle glaucoma and ocular hypertension.

Who makes Nebivolol 1 Percent?

Nebivolol 1 Percent is being developed by Summit Therapeutics Inc., a biopharmaceutical company. Summit Therapeutics is publicly traded under the ticker symbol SMMT on the stock market.

What phase is Nebivolol 1 Percent in?

Nebivolol 1 Percent is in Phase 2 clinical development. It is an investigational drug and has not been approved by regulatory authorities. A Phase 2 clinical trial has been completed to evaluate its safety and efficacy in patients with open-angle glaucoma and ocular hypertension.

What clinical trials is Nebivolol 1 Percent in?

Nebivolol 1 Percent has been studied in a completed Phase 2 clinical trial with the identifier NCT04910100. This trial compared Nebivolol 0.5% and 1.0% suspensions to Timolol 0.5% solution in 226 patients with open-angle glaucoma or ocular hypertension. The study was conducted in the United States.

Is Nebivolol 1 Percent the same as Timolol?

No, Nebivolol 1 Percent is not the same as Timolol. Nebivolol is a distinct beta-blocker being developed by Summit Therapeutics, while Timolol is an established beta-blocker used as a comparator in clinical trials. In the Phase 2 trial, Nebivolol was compared directly against Timolol 0.5% solution.