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Ibrutinib

Phase 2

Lymphoma | Small molecule | Oncology |Karyopharm Therapeutics Inc.|Last Updated: Aug 11, 2026

Target and mechanism

Molecular targetBTK
Target classInhibitor
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLEDDMC
Total Trials1
Total Enrollment129

FDA Designations

No designations recorded

Clinical trial landscape

Ibrutinib · 1 trial · 1 indication

Phase 2 1
NCT02436707Novel Combination Therapy in the Treatment of Relapsed and Refractory Aggressive B-Cell LymphomaLymphoma
ACTIVE NOT_RECRUITING129 Analytics
PHASE2ACTIVE NOT_RECRUITING
Novel Combination Therapy in the Treatment of Relapsed and Refractory Aggressive B-Cell Lymphoma
LymphomaUnlock trial analytics

Study Endpoints

Primary Endpoints

Measure overall response rate
2 years

To determine the overall response rate (complete and partial response) to novel combination therapy in patients with relapsed and refractory aggressive B cell lymphoma

Secondary Endpoints

Number and severity of adverse events
2 years
Transplantation rate
2 years
Stem cell collection rate
2 years
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
R-GDPACTIVE_COMPARATORRituximab - 375 mg/m2 IV, 1.5 - 6 hours D1 (prior to cisplatin); Gemcitabine - 1000 mg/m2, IV 30 min D1, D8; Dexamethasone - 40 mg daily PO D1 - D4; Cisplatin - 75 mg/m2 IV, 1 hour D1;
Ibrutinib plus R-GDP (ACCRUAL COMPLETE)EXPERIMENTALIbrutinib 560 mg PO -- D1 - D21 Rituximab 375 mg/m2 IV 1.5 - 6 hours D1 (prior to cisplatin) Gemcitabine 1000 mg/m2 IV 30 min D1, D8 Dexamethasone 40 mg daily PO -- D1 - D4 Cisplatin 75 mg/m2 IV 1 hour D1
R-DICEP (ACCRUAL COMPLETE)EXPERIMENTALRituximab 375 mg/m2 IV 1.5-6hrs Day 1 and Day 5 prior to Cisplatin Mesna 1.75 g/m2 IV 24 hour Cycle 1, Day 2, Day 3 and Day 4 Cyclophosphamide, 1.75 g/m2 IV 2 hours, Day 2, Day 3 and Day 4 Etoposide 350 mg/m2 IV 2 hours, Day 2, Day 3 and Day 4 Cisplatin 35 mg/m2 IV, 2 hours, Day 2, Day 3 and Day 4 G-CSF 300 mcg (\<60kg); 480 mcg (60-90kg); 600 mcg (\>90kg); SC, Daily, starting Day 15 until apheresis completed.
Selinexor + R-GDPEXPERIMENTALSelinexor - 40mg PO, D1, D3, D8 Rituximab - 375 mg/m2 IV, 1.5 - 6 hours D1 (prior to cisplatin); Gemcitabine - 1000 mg/m2, IV 30 min D1, D8; Dexamethasone - 40 mg daily PO D1 - D4; Cisplatin - 75 mg/m2 IV, 1 hour D1;

Interventions

NameTypeDescription
IbrutinibDRUG -
RituximabDRUG -
GemcitabineDRUG -
DexamethasoneDRUG -
CisplatinDRUG -
MesnaDRUG -
CyclophosphamideDRUG -
EtoposideDRUG -
G-CSFDRUG -
SelinexorDRUG -
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Eligibility Criteria

Age Range16 Years to 65 Years
SexALL
Healthy VolunteersNo
Study Sites11

Inclusion Criteria: * Patients with histologic diagnosis for one of the following histologies according to the World Health Organization: documented at initial diagnosis or at relapse: * Diffuse large cell lymphoma, B-cell (includes primary mediastinal B-cell lymphoma, T-cell rich B-cell lymphom...

Countries:Canada
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Competitive Landscape -Lymphoma 338 trials

Top 20 of 66 competitors

CompanyTickerTrialsLead PhaseDrugs
Regeneron Pharmaceuticals, Inc.REGN7PHASE3Odronextamab, Rituximab, Cyclophosphamide, Doxorubicin, Vincristine
Eli Lilly and CompanyLLY12PHASE3Pirtobrutinib, Idelalisib, Bendamustine, Rituximab
AstraZeneca PLCAZN14PHASE3Surovatamig, R-CHOP, R-CVP, BR
Merck & Co., Inc.MRK16PHASE3Nemtabrutinib, Fludarabine, Cyclophosphamide, Bendamustine, Rituximab
AbbVie, Inc.ABBV11PHASE3Venetoclax
Novartis AG Sponsored ADRNVS8PHASE3Tisagenlecleucel, Lenalidomide and rituximab in 28-day cycles for up to 12 cycles, Rituximab, cyclophosphamide, doxorubicin, vincristine and prednisone or prednisolone in 21-day cycles for 6 to 8 cycles, Lymphodepleting chemotherapy
Incyte CorporationINCY16PHASE3Tafasitamab, Lenalidomide
BeOne Medicines Ltd. Sponsored ADRONC20PHASE3BGB-16673, Bendamustine, Rituximab, Methylprednisolone, Chlorambucil
Gilead Sciences, Inc.GILD7PHASE3Axicabtagene Ciloleucel, Cyclophosphamide, Fludarabine, Lenalidomide, Rituximab
Genmab A/S Sponsored ADRGMAB18PHASE3Epcoritamab, Rituximab, Lenalidomide
Bristol-Myers Squibb CompanyBMY17PHASE3Golcadomide, Rituximab, Cyclophosphamide, Doxorubicin, Vincristine
Johnson & JohnsonJNJ11PHASE3Ibrutinib
Pfizer Inc.PFE4PHASE3Brentuximab vedotin, Rituximab, Lenalidomide
Nurix Therapeutics, Inc.NRIX6PHASE3NX-5948, Pirtobrutinib
ADC Therapeutics LtdADCT4PHASE3Loncastuximab Tesirine, Rituximab, Gemcitabine, Oxaliplatin
Corvus Pharmaceuticals, Inc.CRVS2PHASE3Soquelitinib, Belinostat, Pralatrexate
Grifols, S.A. Sponsored ADR Class BGRFS1PHASE3Xembify
HUTCHMED (China) Limited Sponsored ADRHCM2PHASE3HMPL-760, R-GemOx
Nuvalent, Inc. Class ANUVL1PHASE3Neladalkib, Alectinib
Takeda Pharmaceutical Co. Ltd. Sponsored ADRTAK6PHASE2Brentuximab Vedotin, Cyclophosphamide, Doxorubicin, Prednisone
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Recent Changes (Last 90 Days)

MEDIUMAug 11, 2026NCT02436707primaryCompletionDate: changed
MEDIUMAug 11, 2026NCT02436707primaryCompletionDate: changed

Frequently asked questions about Ibrutinib

What is Ibrutinib used for in lymphoma?

Ibrutinib is an investigational small molecule being studied for the treatment of lymphoma, specifically in a Phase 2 clinical trial for relapsed and refractory aggressive B-cell lymphoma. It is being developed by Karyopharm Therapeutics Inc. and is not yet approved by the FDA.

What does Ibrutinib target?

Ibrutinib is a kinase inhibitor, as indicated by its '-tinib' suffix, which denotes a class of drugs that target kinases. Kinases are enzymes involved in cell signaling and growth, and inhibiting them can help slow or stop cancer cell proliferation.

Who makes Ibrutinib?

Ibrutinib is being developed by Karyopharm Therapeutics Inc., a biopharmaceutical company traded under the ticker symbol KPTI. The company is conducting clinical research on this drug for the treatment of lymphoma.

What phase is Ibrutinib in?

Ibrutinib is currently in Phase 2 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities and is still undergoing clinical trials to evaluate its safety and efficacy in patients with lymphoma.

What clinical trials is Ibrutinib in?

Ibrutinib is being studied in a single Phase 2 clinical trial with the identifier NCT02436707, titled 'Novel Combination Therapy in the Treatment of Relapsed and Refractory Aggressive B-Cell Lymphoma.' This active, non-recruiting trial is enrolling 129 participants in Canada and is open to individuals aged 16 years and older.

Is Ibrutinib the same as ibrutinib?

Yes, Ibrutinib is the same as ibrutinib. The drug is commonly referred to by its generic name, ibrutinib, and is being developed by Karyopharm Therapeutics Inc. for the treatment of lymphoma.